Employees – University of Copenhagen

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Department of Drug Design and Pharmacology > Employees

Hans Bräuner-Osborne

Hans Bräuner-Osborne

Professor


  1. 2005
  2. Published

    Chemoenzymatic synthesis of a series of 4-substituted glutamate analogues and pharmacological characterization at human glutamate transporters subtypes 1-3. / Alaux, Sebastien; Kusk, Mie; Sagot, Emanuelle; Bolte, Jean; Jensen, Anders A.; Bräuner-Osborne, Hans; Gefflaut, Thierry; Bunch, Lennart.

    In: Journal of Medicinal Chemistry, Vol. 48, No. 25, 2005, p. 7980-92.

    Research output: Research - peer-reviewJournal article

  3. Published

    Azetidinic amino acids : stereocontrolled synthesis and pharmacological characterization as ligands for glutamate receptors and transporters. / Bräuner-Osborne, Hans; Bunch, Lennart; Chopin, Nathalie; Couty, François; Evano, Gwilherm; Jensen, Anders A.; Kusk, Mie Lindskov; Nielsen, Birgitte; Rabasso, Nicolas.

    In: Organic & Biomolecular Chemistry, Vol. 3, No. 21, 2005, p. 3926-36.

    Research output: Research - peer-reviewJournal article

  4. Published

    Synthesis of novel N1-substituted bicyclic pyrazole amino acids and evaluation of their interaction with glutamate receptors. / Conti, Paola; Grazioso, Giovanni; di Ventimiglia, Samuele Joppolo; Pinto, Andrea; Roda, Gabriella; Madsen, Ulf; Bräuner-Osborne, Hans; Nielsen, Birgitte; Costagli, Chiara; Galli, Alessandro.

    In: Chemistry & Biodiversity, Vol. 2, No. 6, 06.2005, p. 748-57.

    Research output: Research - peer-reviewJournal article

  5. Published

    Synthesis, binding affinity at glutamic acid receptors, neuroprotective effects, and molecular modeling investigation of novel dihydroisoxazole amino acids. / Conti, Paola; De Amici, Marco; Grazioso, Giovanni; Roda, Gabriella; Pinto, Andrea; Hansen, Kasper Bø; Nielsen, Birgitte; Madsen, Ulf; Bräuner-Osborne, Hans; Egebjerg, Jan; Vestri, Valentina; Pellegrini-Giampietro, Domenico E; Sibille, Pauline; Acher, Francine C; De Micheli, Carlo.

    In: Journal of Medicinal Chemistry, Vol. 48, No. 20, 06.10.2005, p. 6315-25.

    Research output: Research - peer-reviewJournal article

  6. Published

    Tetrazolyl isoxazole amino acids as ionotropic glutamate receptor antagonists: synthesis, modelling and molecular pharmacology. / Frølund, Bente; Greenwood, Jeremy R; Holm, Mai Marie; Egebjerg, Jan; Madsen, Ulf; Nielsen, Birgitte; Bräuner-Osborne, Hans; Stensbøl, Tine B; Krogsgaard-Larsen, Povl.

    In: Bioorganic & Medicinal Chemistry, Vol. 13, No. 18, 15.09.2005, p. 5391-8.

    Research output: Research - peer-reviewJournal article

  7. Published

    Tweaking agonist efficacy at N-methyl-D-aspartate receptors by site-directed mutagenesis. / Hansen, Kasper B; Clausen, Rasmus P; Bjerrum, Esben J; Bechmann, Christian; Greenwood, Jeremy R; Christensen, Caspar; Kristensen, Jesper L; Egebjerg, Jan; Bräuner-Osborne, Hans.

    In: Molecular Pharmacology, Vol. 68, No. 6, 12.2005, p. 1510-23.

    Research output: Research - peer-reviewJournal article

  8. Published
  9. Published

    Rigid nonproteinogenic cyclic amino acids as ligands for glutamate receptors: trans-tris(homoglutamic) acids. / Meyer, Udo; Bisel, Philippe; Bräuner-Osborne, Hans; Madsen, Ulf; Höfner, Georg; Wanner, Klaus Th; Frahm, August Wilhelm.

    In: Chirality, Vol. 17, No. 2, 02.2005, p. 99-107.

    Research output: Research - peer-reviewJournal article

  10. Published

    Deorphanization of GPRC6A: a promiscuous L-alpha-amino acid receptor with preference for basic amino acids. / Wellendorph, Petrine; Hansen, Kasper B; Balsgaard, Anders; Greenwood, Jeremy R; Egebjerg, Jan; Bräuner-Osborne, Hans.

    In: Molecular Pharmacology, Vol. 67, No. 3, 03.2005, p. 589-97.

    Research output: Research - peer-reviewJournal article

  11. Published

    Novel cyclic gamma-hydroxybutyrate (GHB) analogs with high affinity and stereoselectivity of binding to GHB sites in rat brain. / Wellendorph, Petrine; Høg, Signe; Greenwood, Jeremy R; de Lichtenberg, Anne; Nielsen, Birgitte; Frølund, Bente; Brehm, Lotte; Clausen, Rasmus P; Bräuner-Osborne, Hans.

    In: Journal of Pharmacology and Experimental Therapeutics, Vol. 315, No. 1, 10.2005, p. 346-51.

    Research output: Research - peer-reviewJournal article

ID: 1302910