Albert Jelke Kooistra

Albert Jelke Kooistra

Assistant professor


  1. 2019
  2. Covalent Inhibition of the Histamine H3 Receptor

    Wágner, G., Mocking, T. A. M., Kooistra, Albert Jelke, Slynko, I., Ábrányi-Balogh, P., Keserű, G. M., Wijtmans, M., Vischer, H. F., de Esch, I. J. P. & Leurs, R., 11 Dec 2019, In : Molecules (Print Archive Edition). 24, 19 p., 4541.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Community assessment to advance computational prediction of cancer drug combinations in a pharmacogenomic screen

    AstraZeneca-Sanger Drug Combination DREAM Consortium, A. D. C. D. C., 1 Dec 2019, In : Nature Communications. 10, 1, 17 p., 2674.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. The Landscape of Atypical and Eukaryotic Protein Kinases

    Kanev, G. K., de Graaf, C., de Esch, I. J. P., Leurs, R., Würdinger, T., Westerman, B. A. & Kooistra, Albert Jelke, Nov 2019, In : Trends in Pharmacological Sciences. 40, 11, p. 818-832 15 p.

    Research output: Contribution to journalReviewResearchpeer-review

  5. Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors (Part 2)

    de Heuvel, E., Singh, A. K., Boronat, P., Kooistra, Albert Jelke, van der Meer, T., Sadek, P., Blaazer, A. R., Shaner, N. C., Bindels, D. S., Caljon, G., Maes, L., Sterk, G. J., Siderius, M., Oberholzer, M., de Esch, I. J. P., Brown, D. G. & Leurs, R., 15 Sep 2019, In : Bioorganic & Medicinal Chemistry. 27, 18, p. 4013-4029 17 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Route to Prolonged Residence Time at the Histamine H1 Receptor: Growing from Desloratadine to Rupatadine

    Bosma, R., Wang, Z., Kooistra, Albert Jelke, Bushby, N., Kuhne, S., van den Bor, J., Waring, M. J., de Graaf, C., de Esch, I. J., Vischer, H. F., Sheppard, R. J., Wijtmans, M. & Leurs, R., 25 Jul 2019, In : Journal of Medicinal Chemistry. 62, 14, p. 6630-6644 15 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Aminergic GPCR-Ligand Interactions: A Chemical and Structural Map of Receptor Mutation Data

    Vass, M., Podlewska, S., De Esch, I. J. P., Bojarski, A. J., Leurs, R., Kooistra, Albert Jelke & De Graaf, C., 2019, In : Journal of Medicinal Chemistry. 62, 8, p. 3784-3839 56 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. 2018
  9. Development of novel fluorescent histamine H1-receptor antagonists to study ligand-binding kinetics in living cells

    Stoddart, L. A., Vernall, A. J., Bouzo-Lorenzo, M., Bosma, R., Kooistra, Albert Jelke, De Graaf, C., Vischer, H. F., Leurs, R., Briddon, S. J., Kellam, B. & Hill, S. J., 1 Dec 2018, In : Scientific Reports. 8, 1, 1572.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Structural insights into serotonin receptor ligands polypharmacology

    Podlewska, S., Kafel, R., Lacivita, E., Satała, G., Kooistra, Albert Jelke, Vass, M., de Graaf, C., Leopoldo, M., Bojarski, A. J. & Mordalski, Stefan Mateusz, 10 May 2018, In : European Journal of Medicinal Chemistry. 151, p. 797-814 18 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Chemical Diversity in the G Protein-Coupled Receptor Superfamily

    Vass, M., Kooistra, Albert Jelke, Yang, D., Stevens, R. C., Wang, M. W. & de Graaf, C., 1 May 2018, In : Trends in Pharmacological Sciences. 39, 5, p. 494-512 19 p.

    Research output: Contribution to journalReviewResearchpeer-review

  12. Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology

    Hauwert, N. J., Mocking, T. A. M., Da Costa Pereira, D., Kooistra, Albert Jelke, Wijnen, L. M., Vreeker, G. C. M., Verweij, E. W. E., De Boer, A. H., Smit, M. J., De Graaf, C., Vischer, H. F., De Esch, I. J. P., Wijtmans, M. & Leurs, R., 28 Mar 2018, In : Journal of the American Chemical Society. 140, 12, p. 4232-4243 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

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