Employees – University of Copenhagen

Anders A. Jensen

Anders A. Jensen

Associate Professor


  1. 2019
  2. Published

    Use of the 4-Hydroxy-Triazole Moiety as a Bioisosteric Tool for the Development of Ionotropic Glutamate Receptor Ligands. / Sainas, Stefano; Temperini, Piero; Farnsworth, Jill C; Yi, Feng; Møllerud, Stine; Jensen, Anders A.; Nielsen, Birgitte; Kastrup, Jette Sandholm Jensen; Hansen, Kasper B; Boschi, Donatella; Pickering, Darryl S; Clausen, Rasmus Prætorius; Lolli, Marco.

    In: Journal of Medicinal Chemistry, Vol. 62, 09.05.2019, p. 4467-4482.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Discovery of 2-(Imidazo[1,2-b]pyridazin-2-yl)acetic Acid as a New Class of Ligands Selective for the γ-Hydroxybutyric Acid (GHB) High-Affinity Binding Sites. / Krall, Jacob; Bavo, Francesco; Falk-Petersen, Christina B; Jensen, Claus Hatt; Nielsen, Julie Olsson; Tian, Yongsong; Anglani, Valeria; Kongstad, Kenneth Thermann; Piilgaard, Louise; Nielsen, Birgitte; Gloriam, David E; Kehler, Jan; Jensen, Anders; Harpsøe, Kasper; Wellendorph, Petrine; Frølund, Bente.

    In: Journal of Medicinal Chemistry, Vol. 62, No. 5, 14.03.2019, p. 2798-2813.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Accepted/In press

    Design and Synthesis of 2,3-trans-Proline Analogs as Ligands for the Ionotropic Glutamate Receptors and the Excitatory Amino Acid Transporters. / Poulie, Christian Bernard Matthijs; Alcaide Lopez, Anna; Krell-Jørgensen, Mikkel Poul; Larsen, Younes; Astier, Eloi; Bjørn-Yoshimoto, Walden; Yi, Feng; Syrenne, Jed T; Storgaard, Morten; Nielsen, Birgitte; Frydenvang, Karla Andrea; Jensen, Anders A.; Hansen, Kasper B; Pickering, Darryl S; Bunch, Lennart.

    In: A C S Chemical Neuroscience, 2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. 2018
  6. Published

    Conformational transitions of the serotonin 5-HT3 receptor. / Polovinkin, Lucie; Hassaine, Ghérici; Perot, Jonathan; Neumann, Emmanuelle; Jensen, Anders A; Lefebvre, Solène N; Corringer, Pierre-Jean; Neyton, Jacques; Chipot, Christophe; Dehez, Francois; Schoehn, Guy; Nury, Hugues.

    In: Nature, Vol. 563, No. 7730, 11.2018, p. 275-279.

    Research output: Contribution to journalLetterResearchpeer-review

  7. Published

    Probing the molecular basis for affinity/potency- and efficacy-based subtype-selectivity exhibited by benzodiazepine-site modulators at GABAA receptors. / Söderhielm, Pella Cecilia; Balle, Thomas; Bak-Nyhus, Søren; Zhang, Michael; Hansen, Karoline M.; Ahring, Philip K.; Jensen, Anders A.

    In: Biochemical Pharmacology, Vol. 158, 08.2018, p. 339-358.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    5-HT2C Receptor Structures Reveal the Structural Basis of GPCR Polypharmacology. / Peng, Yao; McCorvy, John D.; Harpsøe, Kasper; Lansu, Katherine; Yuan, Shuguang; Popov, Petr; Qu, Lu; Pu, Mengchen; Che, Tao; Nikolajsen, Louise F.; Huang, Xi-ping; Wu, Yiran; Shen, Ling; Bjørn-Yoshimoto, Walden E.; Ding, Kang; Wacker, Daniel; Han, Gye Won; Cheng, Jianjun; Katritch, Vsevolod; Jensen, Anders A.; Hanson, Michael A.; Zhao, Suwen; Gloriam, David E.; Roth, Bryan L.; Stevens, Raymond C.; Liu, Zhi-jie.

    In: Cell, Vol. 172, No. 4, P719-730.E14, 2018, p. 719-730.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Chemoenzymatic synthesis and pharmacological characterization of functionalized aspartate analogues as novel excitatory amino acid transporter inhibitors. / Fu, Haigen; Zhang, J.; Tepper, P.G.; Bunch, Lennart; Jensen, Anders A.; Poelarends, G.J.

    In: Journal of Medicinal Chemistry, Vol. 61, No. 17, 2018, p. 7741-7753 .

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Delineation of the functional properties and the mechanism of action of AA29504, an allosteric agonist and positive allosteric modulator of GABAA receptors. / Olander, Emma Rie; Madjroh, Nawid; Bunch, Lennart; Söderhielm, Pella Cecilia; Jensen, Anders A.

    In: Biochemical Pharmacology, Vol. 150, 2018, p. 305-319.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Dual Nicotinic Acetylcholine Receptor α4β2 Antagonists/α7 Agonists: Synthesis, Docking Studies, and Pharmacological Evaluation of Tetrahydroisoquinolines and Tetrahydroisoquinolinium Salts. / Crestey, François; Jensen, Anders A.; Soerensen, Christian; Magnus, Charlotte Busk; Andreasen T., Jesper; Peters, Günther Herbert Johannes; Kristensen, Jesper Langgaard.

    In: Journal of Medicinal Chemistry, Vol. 61, 2018, p. 1719-1729.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Functional Properties and Mechanism of Action of PPTQ, an Allosteric Agonist and Low Nanomolar Positive Allosteric Modulator at GABAA Receptors. / Madjroh, Nawid; Olander, Emma Rie; Bundgaard, Christoffer; Söderhielm, Pella Cecilia; Jensen, Anders A.

    In: Biochemical Pharmacology, Vol. 147, 2018, p. 153-169.

    Research output: Contribution to journalJournal articleResearchpeer-review

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