Bente Frølund

Bente Frølund

Professor with special responsibilities


  1. 2019
  2. E-pub ahead of print

    Developing new 4-PIOL and 4-PHP analogues for photo-inactivation of γ-aminobutyric acid type A receptors. / Mortensen, Martin; Krall, Jakob; Kongstad, Kenneth T; Brygger, Benjamin M; Lenzi, Ombretta; Francotte, Pierre; Sørensen, Troels E; Nielsen, Birgitte; Jensen, Anders A; Smart, Trevor G; Frølund, Bente.

    In: ACS Chemical Neuroscience, 07.10.2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Five-membered N-heterocyclic Scaffolds as Novel Amino Bioisosteres at gamma-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters. / Giraudo, Alessandro; Krall, Jacob; Bavo, Francesco; Nielsen, Birgitte; Kongstad, Kenneth Thermann; Rolando, Barbara; De Blasio, Rosella; Gloriam, David E; Löffler, Rebekka; Thiesen, Louise; Harpsøe, Kasper; Frydenvang, Karla; Boschi, Donatella; Wellendorph, Petrine; Lolli, Marco L; Jensen, Anders A.; Frølund, Bente.

    In: Journal of Medicinal Chemistry, Vol. 62, No. 12, 27.06.2019, p. 5797-5809.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. E-pub ahead of print

    Structural and molecular aspects of betaine-GABA transporter 1 (BGT1) and its relation to brain function. / Kickinger, Stefanie; Hellsberg, Eva; Frølund, Bente; Schousboe, Arne; Ecker, Gerhard F; Wellendorph, Petrine.

    In: Neuropharmacology, 18.05.2019.

    Research output: Contribution to journalReviewResearchpeer-review

  5. Published

    Synthesis and Pharmacological Evaluation of [C-11]4-Methoxy-N-[2-(thiophen-2-yl) imidazo[1,2-a] pyridin-3-yl]benzamide as a Brain Penetrant PET Ligand Selective for the delta-Subunit-Containing gamma-Aminobutyric Acid Type A Receptors. / L'Estrade, Elina T.; Hansen, Hanne D.; Falk-Petersen, Christina; Haugaard, Anne; Griem-Krey, Nane; Jung, Sascha; Lueddens, Hartmut; Schirmeister, Tanja; Erlandsson, Maria; Ohlsson, Tomas; Knudsen, Gitte M.; Herth, Matthias M.; Wellendorph, Petrine; Frolund, Bente.

    In: ACS Omega, Vol. 4, No. 5, 05.2019, p. 8846-8851.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Lack of evidence for synaptic high-affinity γ-hydroxybutyric acid (GHB) transport in rat brain synaptosomes and 11 Na+ -dependent SLC neurotransmitter transporters. / Thiesen, Louise; Frølund, Bente; Wellendorph, Petrine.

    In: Journal of Neurochemistry, Vol. 149, No. 2, 04.2019, p. 195-210.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Discovery of 2-(Imidazo[1,2-b]pyridazin-2-yl)acetic Acid as a New Class of Ligands Selective for the γ-Hydroxybutyric Acid (GHB) High-Affinity Binding Sites. / Krall, Jacob; Bavo, Francesco; Falk-Petersen, Christina B; Jensen, Claus Hatt; Nielsen, Julie Olsson; Tian, Yongsong; Anglani, Valeria; Kongstad, Kenneth Thermann; Piilgaard, Louise; Nielsen, Birgitte; Gloriam, David E; Kehler, Jan; Jensen, Anders A.; Harpsøe, Kasper; Wellendorph, Petrine; Frølund, Bente.

    In: Journal of Medicinal Chemistry, Vol. 62, No. 5, 14.03.2019, p. 2798-2813.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Designing Poly-agonists for Treatment of Metabolic Diseases : Challenges and Opportunities. / Petersen, Jonas; Strømgaard, Kristian; Frølund, Bente; Clemmensen, Christoffer.

    In: Drugs, Vol. 79, No. 11, 2019, p. 1187-1197.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. 2018
  10. Published

    4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric gamma-aminobutyric acid receptor binding site. / Alessandro, Giraudo; Krall, Jacob; Nielsen, Birgitte; Sørensen, Troels Ersted; Kongstad, Kenneth Thermann; Barbara, Rolando; Donatella, Boschi; Frølund, Bente; Lolli, Marco L.

    In: European Journal of Medicinal Chemistry, Vol. 158, 05.10.2018, p. 311-321.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Synthesis, pharmacological activity and molecular modeling studies of a series of 2-amino-1,4,5,6-tetrahydropyrimidine-5-carboxylic acid analogues as betaine/GABA transporter 1 (BGT1) substrate-inhibitors. / Kickinger, Stefanie; Al-Khawaja, Anas; Haugaard, Anne Staehr; Loeffler, Rebekka; Damgaard, Maria; Eckert, Gerhard; Frolund, Bente; Wellendorph, Petrine.

    2018. Abstract from 256th National Meeting and Exposition of the American-Chemical-Society (ACS) - Nanoscience, Nanotechnology and Beyond, United States.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  12. Published

    Structure-Function Evaluation of Imidazopyridine Derivatives Selective for δ-Subunit-Containing γ-Aminobutyric Acid Type A (GABAA) Receptors. / Yakoub, Kirsten; Jung, Sascha; Sattler, Christian; Damerow, Helen; Weber, Judith; Kretzschmann, Annika; Cankaya, Aylin S; Piel, Markus; Rösch, Frank; Haugaard, Anne S; Frølund, Bente; Schirmeister, Tanja; Lüddens, Hartmut.

    In: Journal of Medicinal Chemistry, Vol. 61, No. 5, 08.03.2018, p. 1951-1968.

    Research output: Contribution to journalJournal articleResearchpeer-review

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