Darryl S Pickering
Associate Professor
Molecular and Cellular Pharmacology
Jagtvej 160, 2100 København Ø, 22, Building: C213
- 2007
- Published
Pharmacological characterisation of biarylisopropylalsulphonamide AMPA-R potentiators. / Pickering, Darryl S; Sanz, Contreraz; Harpsøe, Kasper; Clausen, Rasmus Prætorius; Sauerberg, P.; Liljefors, Tommy; Madsen, Ulf; Kaae, B.H.
In: Journal of Neurochemistry, Vol. 102 (suppl. 1), No. 41, 2007.Research output: Contribution to journal › Conference abstract in journal › Research
- Published
Structural proof of a dimeric positive modulator bridging two identical AMPA receptor-binding sites. / Kaae, Birgitte Høiriis; Harpsøe, Kasper; Kastrup, Jette Sandholm Jensen; Sanz, Alberto Contreras; Pickering, Darryl Scott; Metzler, Bjørn; Clausen, Rasmus Prætorius; Gajhede, Michael; Sauerberg, Per; Liljefors, Tommy; Madsen, Ulf.
In: Chemistry & Biology, Vol. 14, No. 11, 2007, p. 1294-303.Research output: Contribution to journal › Journal article › Research › peer-review
- 2006
- Published
3-hydroxypyridazine 1-oxides as carboxylate bioisosteres : a new series of subtype-selective AMPA receptor agonists. / Greenwood, Jeremy R; Mewett, Ken N; Allan, Robin D; Martín, Belén Ortiz; Pickering, Darryl.
In: Neuropharmacology, Vol. 51, No. 1, 07.2006, p. 52-9.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The structure of a mixed GluR2 ligand-binding core dimer in complex with (S)-glutamate and the antagonist (S)-NS1209. / Kasper, Christina; Pickering, Darryl S; Mirza, Osman; Olsen, Lars; Kristensen, Anders S; Greenwood, Jeremy R; Liljefors, Tommy; Schousboe, Arne; Wätjen, Frank; Gajhede, Michael; Sigurskjold, Bent W; Kastrup, Jette S.
In: Journal of Molecular Biology, Vol. 357, No. 4, 2006, p. 1184-201.Research output: Contribution to journal › Journal article › Research › peer-review
- 2005
- Published
Convergent synthesis and pharmacology of substituted tetrazolyl-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid analogues. / Vogensen, SB; Clausen, Rasmus Prætorius; Greenwood, JR; Johansen, Tommy Nørskov; Pickering, DS; Nielsen, Birgitte; Ebert, Barke; Krogsgaard-Larsen, P.
In: Journal of Medicinal Chemistry, Vol. 48, No. 9, 05.05.2005, p. 3438-3442.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
4-Alkylated homoibotenic acid (HIBO) analogues: versatile pharmacological agents with diverse selectivity profiles towards metabotropic and ionotropic glutamate receptor subtypes. / Madsen, Ulf; Pickering, Darryl S; Nielsen, Birgitte; Bräuner-Osborne, Hans.
In: Neuropharmacology, Vol. 49 Suppl 1, 2005, p. 114-9.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
D-aspartate and NMDA, but not L-aspartate, block AMPA receptors in rat hippocampal neurons. / Gong, Xiang-Qun; Frandsen, Anne; Lu, Wei-Yang; Wan, Yudi; Zabek, Rebecca L; Pickering, Darryl; Bai, Donglin.
In: British Journal of Pharmacology, Vol. 145, No. 4, 2005, p. 449-59.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Exploring the GluR2 ligand-binding core in complex with the bicyclical AMPA analogue (S)-4-AHCP. / Nielsen, Bettina B; Pickering, Darryl S; Greenwood, Jeremy R; Brehm, Lotte; Gajhede, Michael; Schousboe, Arne; Kastrup, Jette S.
In: FEBS Journal, Vol. 272, No. 7, 2005, p. 1639-48.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Tyr702 is an important determinant of agonist binding and domain closure of the ligand-binding core of GluR2. / Frandsen, Anne; Pickering, Darryl S.; Vestergaard, Bente; Kasper, Christina; Nielsen, Bettina Bryde; Greenwood, Jeremy R; Campiani, Giuseppe; Fattorusso, Caterina; Gajhede, Michael; Schousboe, Arne; Kastrup, Jette Sandholm.
In: Molecular Pharmacology, Vol. 67, No. 3, 2005, p. 703-13.Research output: Contribution to journal › Journal article › Research › peer-review
- 2004
- Published
A stereochemical anomaly: the cyclised (R)-AMPA analogue (R)-3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid [(R)-5-HPCA] resembles (S)-AMPA at glutamate receptors. / Vogensen, SB; Greenwood, JR; Varming, Annemarie R.; Brehm, L; Pickering, DS; Nielsen, Birgitte; Liljefors, T; Clausen, Rasmus Prætorius; Johansen, Tommy Nørskov; Krogsgaard-Larsen, P.
In: Organic & Biomolecular Chemistry, Vol. 2, No. 2, 2004, p. 206-213.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1299533
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Investigation of the presence and antinociceptive function of muscarinic acetylcholine receptors in the African naked mole-rat (Heterocephalus glaber)
Research output: Contribution to journal › Journal article › Research › peer-review
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