Department of Drug Design and Pharmacology

Darryl S Pickering

Associate Professor

Molecular and Cellular Pharmacology
Jagtvej 160, 2100 København Ø, 22, Building: C213
- picker@sund.ku.dk
- https://drug.ku.dk/
Phone: +45 35 33 43 42

ORCID: 0000-0001-8687-6094

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Published
Lessons from crystal structures of kainate receptors
Frantsen, Stine Møllerud, Frydenvang, Karla Andrea, Pickering, Darryl S & Kastrup, Jette Sandholm Jensen, 1 Jan 2017, In : Neuropharmacology. 112, Part A, p. 16-28 13 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
N-(7-(1H-imidazol-1-yl)-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl)benzamide - a new kainate receptor selective antagonist and analgesic: Synthesis, X-ray crystallography, structure-affinity relationships, in vitro and in vivo pharmacology
Frantsen, Stine Møllerud, Hansen, Rie Bager, Pallesen, J. S., Temperini, Piero, Pasini, D., Bornholdt, J., Nielsen, Birgitte, Mamedova, Esmira, Chalupnik, P., Paternain, A. V., Lerma, J., Diaz del Castillo, Marta, Andreasen T., Jesper, Frydenvang, Karla Andrea, Kastrup, Jette Sandholm Jensen, Johansen, Tommy Nørskov & Pickering, Darryl S, 2019, In : ACS Chemical Neuroscience. 10, p. 4685-4695 11 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
A pharmacological profile of the high-affinity GluK5 kainate receptor
Frantsen, Stine Møllerud, Kastrup, Jette Sandholm Jensen & Pickering, Darryl S, 2016, In : European Journal of Pharmacology. 788, p. 315-320 6 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Structure and affinity of two bicyclic glutamate analogues at AMPA and kainate receptors
Frantsen, Stine Møllerud, Pinto, A., Marconi, L., Frydenvang, Karla Andrea, Thorsen, Thor Seneca, Laulumaa, S. K., Venskutonyte, R., Winther, Nikolaj Sebastian, Cunado Moral, A. M., Tamborini, L., Conti, P., Pickering, Darryl S & Kastrup, Jette Sandholm Jensen, 2017, In : A C S Chemical Neuroscience. 8, 9, p. 2056-2064 9 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Pharmacology and crystal structure of novel 2,3-quinoxalinediones at kainate receptors
Frantsen, Stine Møllerud, Pallesen, J. S., Pasini, D., Marconi, L., Han, L., Bornholt, J., Johansen, Tommy Nørskov, Kastrup, Jette Sandholm Jensen, Pickering, Darryl S & Frydenvang, Karla Andrea, Aug 2017, In : Journal of Neurochemistry. 142, S1, p. 124 1 p., MTU07-13.
Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
Published
Ionotropic glutamate-like receptor d2 binds D-serine and glycine.
Naur, P., Hansen, K. B., Kristensen, Anders Skov, Dravid, S. M., Pickering, Darryl S, Olsen, L., Vestergaard, Bente, Egebjerg, J., Gajhede, Michael, Traynelis, S. F. & Kastrup, Jette Sandholm Jensen, 2007, In : Proceedings of the National Academy of Science of the United States of America. 104, 35, p. 14116-14121
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Pharmacological properties of homomeric and heteromeric GluR1o and GluR3o receptors
Nielsen, B. S., Banke, T. G., Schousboe, Arne & Pickering, Darryl S, 1998, In : European Journal of Pharmacology. 360, 2-3, p. 227-38 11 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Exploring the GluR2 ligand-binding core in complex with the bicyclical AMPA analogue (S)-4-AHCP
Nielsen, B. B., Pickering, Darryl S, Greenwood, J. R., Brehm, L., Gajhede, Michael, Schousboe, Arne & Kastrup, Jette Sandholm Jensen, 2005, In : FEBS Journal. 272, 7, p. 1639-48 9 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
The antagonistic effect of antipsychotic drugs on a HEK293 cell line stably expressing human alpha(1A1)-adrenoceptors
Nourian, Z., Mulvany, M. J., Nielsen, K. B., Pickering, Darryl S & Kristensen, T., 2008, In : European Journal of Pharmacology. 596, 1-3, p. 32-40
Research output: Contribution to journal › Journal article › Research › peer-review
Published
N1-Substituted Quinoxaline-2,3-diones as Kainate Receptor Antagonists: X-ray Crystallography, Structure-Affinity Relationships and in vitro Pharmacology
Pallesen, J. S., Frantsen, Stine Møllerud, Frydenvang, Karla Andrea, Pickering, Darryl S, Bornholt, J., Nielsen, Birgitte, Pasini, D., Han, L., Marconi, L., Kastrup, Jette Sandholm Jensen & Johansen, Tommy Nørskov, 20 Mar 2019, In : A C S Chemical Neuroscience. 10, p. 1841-1853 13 p.
Research output: Contribution to journal › Journal article › Research › peer-review

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ID: 1299533

Darryl S Pickering

Molecular and Cellular Pharmacology

Lessons from crystal structures of kainate receptors

N-(7-(1H-imidazol-1-yl)-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl)benzamide - a new kainate receptor selective antagonist and analgesic: Synthesis, X-ray crystallography, structure-affinity relationships, in vitro and in vivo pharmacology

A pharmacological profile of the high-affinity GluK5 kainate receptor

Structure and affinity of two bicyclic glutamate analogues at AMPA and kainate receptors

Pharmacology and crystal structure of novel 2,3-quinoxalinediones at kainate receptors

Ionotropic glutamate-like receptor d2 binds D-serine and glycine.

Pharmacological properties of homomeric and heteromeric GluR1o and GluR3o receptors

Exploring the GluR2 ligand-binding core in complex with the bicyclical AMPA analogue (S)-4-AHCP

The antagonistic effect of antipsychotic drugs on a HEK293 cell line stably expressing human alpha(1A1)-adrenoceptors

N1-Substituted Quinoxaline-2,3-diones as Kainate Receptor Antagonists: X-ray Crystallography, Structure-Affinity Relationships and in vitro Pharmacology

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