Darryl S Pickering

Darryl S Pickering

Associate Professor


  1. Published

    Design, synthesis, and pharmacology of a highly subtype-selective GluR1/2 agonist, (RS)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)propionic acid (Cl-HIBO). / Bjerrum, Esben J; Kristensen, Anders S; Pickering, Darryl S; Greenwood, Jeremy R; Nielsen, Birgitte; Liljefors, Tommy; Schousboe, Arne; Bräuner-Osborne, Hans; Madsen, Ulf; Pickering, Darryl.

    In: Journal of Medicinal Chemistry, Vol. 46, No. 11, 2003, p. 2246-9.

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Action of bicyclic isoxazole GABA analogues on GABA transporters and its relation to anticonvulsant activity. / Bolvig, T; Larsson, O M; Pickering, D S; Nelson, N; Falch, E; Krogsgaard-Larsen, P; Schousboe, A; Pickering, Darryl.

    In: European Journal of Pharmacology, Vol. 375, No. 1-3, 1999, p. 367-74.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Characterization of the 1H-cyclopentapyrimidine-2,4(1H,3H)-dione derivative (S)-CPW399 as a novel, potent, and subtype-selective AMPA receptor full agonist with partial desensitization properties. / Campiani, G; Morelli, E; Nacci, V; Fattorusso, C; Ramunno, A; Novellino, E; Greenwood, J; Liljefors, T; Griffiths, R; Sinclair, C; Reavy, H; Kristensen, A S; Pickering, D S; Schousboe, A; Cagnotto, A; Fumagalli, E; Mennini, T; Pickering, Darryl.

    In: Journal of Medicinal Chemistry, Vol. 44, No. 26, 2001, p. 4501-4.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Agonist discrimination between AMPA receptor subtypes. / Coquelle, T; Christensen, J K; Banke, T G; Madsen, U; Schousboe, A; Pickering, Darryl.

    In: NeuroReport, Vol. 11, No. 12, 2000, p. 2643-8.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Molecular determinants of desensitization and assembly of the chimeric GABA(A) receptor subunits (alpha1/gamma2) and (gamma2/alpha1) in combinations with beta2 and gamma2. / Elster, L; Kristiansen, U; Pickering, D S; Olsen, R W; Schousboe, A.

    In: Neurochemistry International, Vol. 38, No. 7, 2001, p. 581-92.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Tyr702 is an important determinant of agonist binding and domain closure of the ligand-binding core of GluR2. / Frandsen, Anne; Pickering, Darryl S.; Vestergaard, Bente; Kasper, Christina; Nielsen, Bettina Bryde; Greenwood, Jeremy R; Campiani, Giuseppe; Fattorusso, Caterina; Gajhede, Michael; Schousboe, Arne; Kastrup, Jette Sandholm.

    In: Molecular Pharmacology, Vol. 67, No. 3, 2005, p. 703-13.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    D-aspartate and NMDA, but not L-aspartate, block AMPA receptors in rat hippocampal neurons. / Gong, Xiang-Qun; Frandsen, Anne; Lu, Wei-Yang; Wan, Yudi; Zabek, Rebecca L; Pickering, Darryl; Bai, Donglin.

    In: British Journal of Pharmacology, Vol. 145, No. 4, 2005, p. 449-59.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    3-hydroxypyridazine 1-oxides as carboxylate bioisosteres : a new series of subtype-selective AMPA receptor agonists. / Greenwood, Jeremy R; Mewett, Ken N; Allan, Robin D; Martín, Belén Ortiz; Pickering, Darryl.

    In: Neuropharmacology, Vol. 51, No. 1, 07.2006, p. 52-9.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Role of desensitization and subunit expression for kainate receptor-mediated neurotoxicity in murine neocortical cultures. / Jensen, J B; Schousboe, A; Pickering, D S; Pickering, Darryl.

    In: Journal of Neuroscience Research, Vol. 55, No. 2, 1999, p. 208-17.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Depolarization-induced release of [(3)H]D-aspartate from GABAergic neurons caused by reversal of glutamate transporters. / Jensen, J B; Pickering, D S; Schousboe, A; Pickering, Darryl.

    In: International Journal of Developmental Neuroscience, Vol. 18, No. 2-3, 2000, p. 309-15.

    Research output: Contribution to journalJournal articleResearchpeer-review

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