Department of Drug Design and Pharmacology

Darryl S Pickering

Associate Professor

Molecular and Cellular Pharmacology
Jagtvej 160, 2100 København Ø, 22, Building: C213
- picker@sund.ku.dk
- https://drug.ku.dk/
Phone: +45 35 33 43 42

ORCID: 0000-0001-8687-6094

All
Research

Publication year:

All

41 - 50 out of 52Page size: 10

Sort by: 1st author

Published
In vitro and in vivo effects of a novel dimeric inhibitor of PSD‐95 on excitotoxicity and functional recovery after experimental traumatic brain injury
Sommer, J. B., Bach, Anders, Rytter, Hana Malá, Strømgaard, Kristian, Mogensen, Jesper & Pickering, Darryl S, 20 Jan 2017, In : European Journal of Neuroscience. 45, 2, p. 238-248 11 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Effects of dimeric PSD-95 inhibition on excitotoxic cell death and outcome after controlled cortical impact in rats: PSD-95 inhibition in experimental TBI
Sommer, J. B., Bach, Anders, Rytter, Hana Malá, Gynther, M., Bjerre, A., Gram, M. G., Marschner, L., Strømgaard, Kristian, Mogensen, Jesper & Pickering, Darryl S, 2017, In : Neurochemical Research. 42, 12, p. 3401-3413 13 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors
Szymanska, E., Frydenvang, Karla Andrea, Pickering, Darryl S, Krintel, C., Nielsen, Birgitte, Kooshki, A., Dorvil, Linda Grønborg, Olsen, L., Kastrup, Jette Sandholm Jensen & Johansen, Tommy Nørskov, 2016, In : Journal of Medicinal Chemistry. 59, 1, p. 448-461 14 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Pharmacological characterization and binding modes of novel racemic and optically active phenylalanine-based antagonists of AMPA receptors
Szymańska, E., Nielsen, Birgitte, Johansen, Tommy Nørskov, Cuñado Moral, A. M., Pickering, Darryl S, Szczepańska, K., Mickowska, A. & Kieć-Kononowicz, K., 2017, In : European Journal of Medicinal Chemistry. 138, p. 874-883 10 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Aryl- and heteroaryl-substituted phenylalanines as AMPA receptor ligands
Szymańska, E., Chałupnik, P., Johansen, Tommy Nørskov, Nielsen, Birgitte, Cuñado Moral, A. M., Pickering, Darryl S & Kieć-Kononowicz, K., 1 Dec 2017, In : Chemical Biology & Drug Design. 90, p. 1271-1281 11 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands
Szymańska, E., Chałupnik, P., Szczepańska, K., Moral, A. M. C., Pickering, Darryl S, Nielsen, Birgitte, Johansen, Tommy Nørskov & Kieć-Kononowicz, K., 2016, In : Bioorganic & Medicinal Chemistry Letters. 26, 22, p. 5568-5572 5 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
γ-Glutamyl-dipeptides: Easy tools to rapidly probe the stereoelectronic properties of ionotropic glutamate receptor binding pocket
Tamborini, L., Nicosia, V., Conti, P., Dall'Oglio, F., De Micheli, C., Nielsen, Birgitte, Jensen, Anders A., Pickering, Darryl S & Pinto, A., 1 Dec 2016, In : Tetrahedron. 72, 51, p. 8586-8492 7 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Molecular recognition of two 2,4-syn-functionalized (S)-glutamate analogues by the kainate receptor GluK3 ligand-binding domain
Venskutonyte, R., Larsen, A. P., Frydenvang, Karla Andrea, Gajhede, Michael, Gefflaut, T., Pickering, Darryl S, Bunch, Lennart & Kastrup, Jette Sandholm Jensen, 2014, In : ChemMedChem. 9, 10, p. 2254-2259 6 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Tweaking subtype-selectivity and agonist efficacy at (S)-2-amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propionic acid (AMPA) receptors in a small series of BnTetAMPA analogues
Wang, S., Larsen, Y., Navarrete, C. V., Jensen, Anders A., Nielsen, Birgitte, Al-Musaed, A., Frydenvang, Karla Andrea, Kastrup, Jette Sandholm Jensen, Pickering, Darryl S & Clausen, Rasmus Prætorius, 2016, In : Journal of Medicinal Chemistry. 59, 5, p. 2244-2254 11 p.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
The Presence of Calcitonin Gene-Related Peptide and Its Receptors in Rat, Pig and Human Brain: Species Differences in Calcitonin Gene-Related Peptide Pharmacology
Warfvinge, K., Edvinsson, Lars, Pickering, Darryl S & Sheykhzade, Majid, 1 Dec 2019, In : Pharmacology. 104, p. 332-341 10 p.
Research output: Contribution to journal › Journal article › Research › peer-review

Previous 1 2 3 4 5 6 Next

ID: 1299533

Darryl S Pickering

Molecular and Cellular Pharmacology

In vitro and in vivo effects of a novel dimeric inhibitor of PSD‐95 on excitotoxicity and functional recovery after experimental traumatic brain injury

Effects of dimeric PSD-95 inhibition on excitotoxic cell death and outcome after controlled cortical impact in rats: PSD-95 inhibition in experimental TBI

Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors

Pharmacological characterization and binding modes of novel racemic and optically active phenylalanine-based antagonists of AMPA receptors

Aryl- and heteroaryl-substituted phenylalanines as AMPA receptor ligands

Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands

γ-Glutamyl-dipeptides: Easy tools to rapidly probe the stereoelectronic properties of ionotropic glutamate receptor binding pocket

Molecular recognition of two 2,4-syn-functionalized (S)-glutamate analogues by the kainate receptor GluK3 ligand-binding domain

Tweaking subtype-selectivity and agonist efficacy at (S)-2-amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propionic acid (AMPA) receptors in a small series of BnTetAMPA analogues

The Presence of Calcitonin Gene-Related Peptide and Its Receptors in Rat, Pig and Human Brain: Species Differences in Calcitonin Gene-Related Peptide Pharmacology

Most downloads

Investigation of the presence and antinociceptive function of muscarinic acetylcholine receptors in the African naked mole-rat (Heterocephalus glaber)