Darryl S Pickering
Associate Professor
Molecular and Cellular Pharmacology
Jagtvej 160, 2100 København Ø, 22, Building: C213
- 2013
- Published
UCCB01-125, a dimeric inhibitor of PSD-95, reduces inflammatory pain without disrupting cognitive or motor performance: Comparison with the NMDA receptor antagonist MK-801. / Andreasen, Jesper T.; Bach, Anders; Gynther, Mikko; Nasser, Arafat; Mogensen, Jesper; Strømgaard, Kristian; Pickering, Darryl S.
In: Neuropharmacology, Vol. 67, 04.2013, p. 193-200.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Does increasing the ratio of AMPA-to-NMDA receptor mediated neurotransmission engender antidepressant action? Studies in the mouse forced swim and tail suspension tests. / Andreasen T., Jesper; Gynther, Mikko Otto Oskari; Rygaard, Allan; Bøgelund, Trine; Nielsen, Simon Dalsgaard; Clausen, Rasmus Prætorius; Mogensen, Jesper; Pickering, Darryl S.
In: Neuroscience Letters, Vol. 546, 2013, p. 6-10.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Chemo-enzymatic synthesis of new 2,4-syn-functionalized (S)-glutamate analogues and structure-activity relationship studies at ionotropic glutamate receptors and excitatory amino acid transporters. / Assaf, Z.; Larsen, Anja Probst; Venskutonyte, Raminta; Han, Liwei; Abrahamsen, Bjarke; Nielsen, Birgitte; Gajhede, Michael; Kastrup, Jette Sandholm; Jensen, Anders A.; Pickering, Darryl S; Frydenvang, Karla ; Gefflaut, T; Bunch, Lennart.
In: Journal of Medicinal Chemistry, Vol. 56, No. 4, 2013, p. 1614-1628.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Studies on an (S)-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor antagonist IKM-159 : asymmetric synthesis, neuroactivity, and structural characterization. / Juknaite, Lina; Sugamata, Yutaro; Tokiwa, Kazuya; Ishikawa, Yuichi; Takamizawa, Satoshi; Eng, Andrew; Sakai, Ryuichi; Pickering, Darryl S; Frydenvang, Karla; Swanson, Geoffrey T; Kastrup, Jette Sandholm Jensen; Oikawa, Masato.
In: Journal of Medicinal Chemistry, Vol. 56, No. 6, 2013, p. 2283-2293.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structural analysis of the positive AMPA receptor modulators CX516 and Me-CX516 in complex with the GluA2 ligand-binding domain. / Krintel, Christian; Harpsøe, Kasper; Zachariassen, Linda G; Peters, Dan; Frydenvang, Karla; Pickering, Darryl S; Gajhede, Michael; Kastrup, Jette S.
In: Acta crystallographica. Section D, Biological crystallography, Vol. 69, No. Pt 9, 09.2013, p. 1645-52.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Crystal structure and pharmacological characterization of a novel N-methyl-D-aspartate (NMDA) receptor antagonist at the GluN1 glycine binding site. / Kvist, Trine; Steffensen, Thomas Bielefeldt; Greenwood, Jeremy R; Mehrzad Tabrizi, Fatemeh; Hansen, Kasper Bø; Gajhede, Michael; Pickering, Darryl S; Traynelis, Stephen F; Kastrup, Jette Sandholm; Bräuner-Osborne, Hans.
In: The Journal of Biological Chemistry, Vol. 288, 2013, p. 33124-35.Research output: Contribution to journal › Journal article › Research › peer-review
- 2014
- Published
Analogues of 3-Hydroxyisoxazole-Containing Glutamate Receptor Ligands Based on the 3-Hydroxypyrazole-Moiety: Design, Synthesis and Pharmacological Characterization. / Jørgensen, Lars; Nielsen, Birgitte; Pickering, Darryl S; Kristensen, Anders Skov; Frydenvang, Karla Andrea; Madsen, Ulf; Clausen, Rasmus Prætorius.
In: Neurochemical Research, Vol. 39, No. 10, 2014, p. 1895-1905.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
L-Asp is a useful tool in the purification of the ionotropic glutamate receptor A2 ligand-binding domain. / Krintel, Christian; Frydenvang, Karla; Ceravalls de Rabassa, Anna; Kaern, Anne Mette; Gajhede, Michael; Pickering, Darryl S; Kastrup, Jette S.
In: F E B S Journal, 27.03.2014, p. 2422–2430.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design, synthesis and in vitro pharmacology of GluK1 and GluK3 antagonists. Studies towards the design of subtype-selective antagonists through 2-carboxyethyl-phenylalanines with substituents interacting with non-conserved residues in the GluK binding sites. / Sköld, Niklas; Nielsen, Birgitte; Olsen, Jakob; Han, Liwei; Olsen, Lars; Madsen, Ulf; Kristensen, Jesper Langgaard; Pickering, Darryl S; Johansen, Tommy N.
In: Bioorganic & Medicinal Chemistry, Vol. 22, No. 19, 02.08.2014, p. 5368-5377.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Molecular recognition of two 2,4-syn-functionalized (S)-glutamate analogues by the kainate receptor GluK3 ligand-binding domain. / Venskutonyte, Raminta; Larsen, Anja Probst; Frydenvang, Karla Andrea; Gajhede, Michael; Gefflaut, Thierry; Pickering, Darryl S; Bunch, Lennart; Kastrup, Jette Sandholm Jensen.
In: ChemMedChem, Vol. 9, No. 10, 2014, p. 2254-2259.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Forster Resonance Energy Transfer (FRET) Analysis of Dual CFP/YFP Labeled AMPA Receptors Reveals Structural Rearrangement within the C-Terminal Domain during Receptor Activation. / Zachariassen, Linda Grønborg; Katchan, Mila; Plested, Andrew; Pickering, Darryl S; Kristensen, Anders Skov.
2014.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- 2015
- Published
Differential role of AMPA receptors in mouse tests of antidepressant and anxiolytic action. / Andreasen, Jesper T; Fitzpatrick, Ciaran M; Larsen, Maria; Skovgaard, Lars; Nielsen, Simon D; Clausen, Rasmus P; Troelsen, Karin; Pickering, Darryl S.
In: Brain Research, Vol. 1601, 19.03.2015, p. 117-26.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Binding Mode of an α-Amino Acid-Linked Quinoxaline-2,3-dione Analogue at Glutamate Receptor Subtype GluK1. / Demmer, Charles S; Møller, Charlotte; Brown, Patricia M G E; Han, Liwei; Pickering, Darryl S; Nielsen, Birgitte; Bowie, Derek; Frydenvang, Karla; Kastrup, Jette S; Bunch, Lennart.
In: A C S Chemical Neuroscience, Vol. 6, 09.04.2015, p. 845-854.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Solid-Phase Peptide Synthesis of Human alfa-Calcitonin Gene-Related Peptide and Two Fluorescent Analogs. / Fuente-Moreno, Marina; Oddo, Alberto; Sheykhzade, Majid; Pickering, Darryl S; Hansen, Paul Robert.
Proceedings of the 24th American Peptide Symposium . 2015.Research output: Chapter in Book/Report/Conference proceeding › Article in proceedings › Research › peer-review
- Published
Blood-brain barrier permeability and brain uptake mechanism of kainic Acid and dihydrokainic Acid. / Gynther, Mikko; Petsalo, Aleksanteri; Hansen, Steen Honoré; Bunch, Lennart; Pickering, Darryl S.
In: Neurochemical Research, Vol. 40, No. 3, 03.2015, p. 542-549.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structure-Activity Relationship Study of Ionotropic Glutamate Receptor Antagonist (2S,3R)-3-(3-Carboxyphenyl)pyrrolidine-2-carboxylic Acid. / Krogsgaard-Larsen, Niels; Storgaard, Morten; Møller, Charlotte; Demmer, Charles S; Hansen, Jeanette; Han, Liwei; Monrad, Rune N; Nielsen, Birgitte; Tapken, Daniel; Pickering, Darryl S; Kastrup, Jette S; Frydenvang, Karla; Bunch, Lennart.
In: Journal of Medicinal Chemistry, Vol. 58, No. 15, 2015, p. 6131-50.Research output: Contribution to journal › Journal article › Research › peer-review
- 2016
- Published
Synthesis and Pharmacological Characterization of the Selective GluK1 Radioligand (S)-2-Amino-3-(6-[3H]-2,4-dioxo-3,4-dihydrothieno[3,2-d]pyrimidin-1(2H)-yl)propanoic acid ([3H]-NF608). / Alcaide, Anna; Marconi, Laura; Marek, Ales; Haym, Isabell; Nielsen, Birgitte; Møllerud, Stine; Jensen, Mikael; Conti, Paola; Pickering, Darryl S; Bunch, Lennart.
In: MedChemComm, Vol. 7, 2016, p. 2136-2144.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Effects of the dimeric PSD-95 inhibitor UCCB01-144 in mouse models of pain, cognition and motor function. / Andreasen, Jesper T; Nasser, Arafat; Caballero-Puntiverio, Maitane; Sahlholt, Maj; Bach, Anders; Gynther, Mikko; Strømgaard, Kristian; Pickering, Darryl S.
In: European Journal of Pharmacology, Vol. 780, 05.06.2016, p. 166-73.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Positive allosteric modulation of AMPA receptors differentially modulates the behavioural effects of citalopram in mouse models of antidepressant and anxiolytic action. / Fitzpatrick, Ciarán Martin; Larsen, Maria; Madsen, Louise; Pickering, Darryl S; Clausen, Rasmus Prætorius; Andreasen T., Jesper.
In: Behavioural Pharmacology, Vol. 27, No. 6, 26.06.2016, p. 549-555.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Systemic and Brain Pharmacokinetics of Perforin Inhibitor Prodrugs. / Gynther, Mikko; Pickering, Darryl S; Spicer, Julie; Denny, William; Huttunen, Kristiina.
In: Molecular Pharmaceutics, Vol. 13, No. 7, 2016, p. 2484-2491.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Neto2 influences on kainate receptor pharmacology and function. / Han, Liwei; Howe, James; Pickering, Darryl S.
In: Basic & Clinical Pharmacology & Toxicology, Vol. 119, 2016, p. 141-148.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Investigation of the presence and antinociceptive function of muscarinic acetylcholine receptors in the African naked mole-rat (Heterocephalus glaber). / Jørgensen, Kristine B.; Krogh-Jensen, Karen; Pickering, Darryl S; Kanui, Titus; Abelson, Klas.
In: Journal of Comparative Physiology A. Sensory, neural, and behavioral physiology, Vol. 202, No. 1, 01.01.2016, p. 7-15.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Enthalpy-Entropy Compensation in the Binding of Modulators at Ionotropic Glutamate Receptor GluA2. / Krintel, Christian; Francotte, Pierre; Pickering, Darryl S; Juknaite, Lina; Pøhlsgaaard, Jakob; Olsen, Lars; Frydenvang, Karla Andrea; Goffin, Eric; Pirotte, Bernard; Kastrup, Jette Sandholm Jensen.
In: Biophysical Journal, Vol. 110, No. 11, 2016, p. 2397-2406.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structure of a High-Affinity Kainate Receptor: GluK4 Ligand-Binding Domain Crystallized with Kainate. / Kristensen, Ole; Kristensen, Lise Baadsgaard; Møllerud, Stine; Frydenvang, Karla Andrea; Pickering, Darryl S; Kastrup, Jette Sandholm Jensen.
In: Structure, Vol. 24, No. 9, 2016, p. 1582-1589.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A pharmacological profile of the high-affinity GluK5 kainate receptor. / Møllerud, Stine; Kastrup, Jette Sandholm Jensen; Pickering, Darryl S.
In: European Journal of Pharmacology, Vol. 788, 2016, p. 315-320.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Effects of sertraline, duloxetine, vortioxetine, and idazoxan in the rat affective bias test. / Refsgaard, Louise Konradsen; Haubro, Kia; Pickering, Darryl S; Stuart, Sarah; Robinson, Emma; Andreasen T., Jesper.
In: Psychopharmacology, Vol. 233, No. 21, 14.10.2016, p. 3763-3770.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Modelling Affective Pain in Mice: Effects of Inflammatory Hypersensitivity on Place Escape/Avoidance Behaviour, Anxiety and Hedonic State. / Refsgaard, Louise Konradsen; Hoffmann-Petersen, Julie; Sahlholt, Maj; Pickering, Darryl S; Andreasen T., Jesper.
In: Journal of Neuroscience Methods, Vol. 262, 2016, p. 85-92.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors. / Szymanska, Ewa; Frydenvang, Karla Andrea; Pickering, Darryl S; Krintel, Christian; Nielsen, Birgitte; Kooshki, Ayesheh; Zachariassen, Linda Grønborg; Olsen, Lars; Kastrup, Jette Sandholm Jensen; Johansen, Tommy Nørskov.
In: Journal of Medicinal Chemistry, Vol. 59, No. 1, 2016, p. 448-461.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands. / Szymańska, Ewa; Chałupnik, Paulina; Szczepańska, Katarzyna; Moral, Ana Maria Cuñado; Pickering, Darryl S; Nielsen, Birgitte; Johansen, Tommy Nørskov; Kieć-Kononowicz, Kieć-Kononowicz.
In: Bioorganic & Medicinal Chemistry Letters, Vol. 26, No. 22, 2016, p. 5568-5572.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
γ-Glutamyl-dipeptides: Easy tools to rapidly probe the stereoelectronic properties of ionotropic glutamate receptor binding pocket. / Tamborini, Lucia; Nicosia, Veronica; Conti, Paola; Dall'Oglio, Federica; De Micheli, Carlo; Nielsen, Birgitte; Jensen, Anders A.; Pickering, Darryl S; Pinto, Andrea.
In: Tetrahedron, Vol. 72, No. 51, 01.12.2016, p. 8586-8492.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Tweaking subtype-selectivity and agonist efficacy at (S)-2-amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propionic acid (AMPA) receptors in a small series of BnTetAMPA analogues. / Wang, Shuang-Yan; Larsen, Younes; Navarrete, Cristina V.; Jensen, Anders A.; Nielsen, Birgitte; Al-Musaed, Ali; Frydenvang, Karla; Kastrup, Jette Sandholm; Pickering, Darryl S; Clausen, Rasmus Prætorius.
In: Journal of Medicinal Chemistry, Vol. 59, No. 5, 2016, p. 2244-2254.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structural rearrangement of the intracellular domains during AMPA receptor activation. / Zachariassen, Linda Grønborg; Katchan, Ljudmila; Jensen, Anna Guldvang; Pickering, Darryl S; Plested, Andrew; Kristensen, Anders Skov.
In: Proceedings of the National Academy of Sciences USA (PNAS), Vol. 113, No. 27, 2016, p. E3950-E3959.Research output: Contribution to journal › Journal article › Research › peer-review
- 2017
- Published
Revisiting the Quinoxalinedione scaffold in the Construction of New Ligands for the Ionotropic Glutamate Receptors. / Demmer, Charles Sylvain; Rombach, David; Liu, Na; Nielsen, Birgitte; Pickering, Darryl S; Bunch, Lennart.
In: A C S Chemical Neuroscience, Vol. 8, No. 11, 01.12.2017, p. 2477-2495.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Augmentation of Anticancer Drug Efficacy in Murine Hepatocellular Carcinoma Cells by a Peripherally Acting Competitive N-Methyl-d-aspartate (NMDA) Receptor Antagonist. / Gynther, Mikko; Proietti Silvestri, Ilaria; Hansen, Jacob C; Hansen, Kasper B; Malm, Tarja; Ishchenko, Yevheniia; Larsen, Younes; Han, Liwei; Kayser, Silke; Auriola, Seppo; Petsalo, Aleksanteri; Nielsen, Birgitte; Pickering, Darryl S; Bunch, Lennart.
In: Journal of Medicinal Chemistry, Vol. 60, No. 23, 14.12.2017, p. 9885-9904.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design and Synthesis of a Series of L-trans-4-Substituted Prolines as Selective Antagonists for the Ionotropic Glutamate Receptors Including Functional and X-ray Crystallographic Studies of New Subtype Selective Kainic Acid Receptor Subtype 1 (GluK1) Antagonist (2S,4R)-4-(2-Carboxyphenoxy)pyrrolidine-2-carboxylic Acid. / Krogsgaard-Larsen, Niels; Delgar, Claudia; Koch, Karina; Brown, Patricia M G E; Møller, Charlotte; Han, Liwei; Huynh, Tri Hien Viet; Hansen, Stinne Wessel; Nielsen, Birgitte; Bowie, Derek; Pickering, Darryl S; Kastrup, Jette Sandholm Jensen; Frydenvang, Karla Andrea; Bunch, Lennart.
In: Journal of Medicinal Chemistry, Vol. 60, No. 1, 2017, p. 441-457.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Lessons from crystal structures of kainate receptors. / Møllerud, Stine; Frydenvang, Karla Andrea; Pickering, Darryl S; Kastrup, Jette Sandholm Jensen.
In: Neuropharmacology, Vol. 112, No. Part A, 01.01.2017, p. 16-28.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Pharmacology and crystal structure of novel 2,3-quinoxalinediones at kainate receptors. / Møllerud, Stine; Pallesen, Jakob Staun; Pasini, Diletta; Marconi, Laura; Han, Liwei; Bornholt, Jan; Johansen, Tommy Nørskov; Kastrup, Jette Sandholm ; Pickering, Darryl S; Frydenvang, Karla Andrea.
In: Journal of Neurochemistry, Vol. 142, No. S1, MTU07-13, 08.2017, p. 124.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Structure and affinity of two bicyclic glutamate analogues at AMPA and kainate receptors. / Møllerud, Stine; Pinto, Andrea; Marconi, Laura; Frydenvang, Karla Andrea; Thorsen, Thor Seneca; Laulumaa, Saara Kaisa; Venskutonyte, Raminta; Winther, Nikolaj; Cunado Moral, Ana Maria; Tamborini, Lucia; Conti, Paola; Pickering, Darryl S; Kastrup, Jette Sandholm Jensen.
In: A C S Chemical Neuroscience, Vol. 8, No. 9, 2017, p. 2056-2064.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Investigation of antidepressant-like and anxiolytic-like actions and cognitive and motor side effects of four N-methyl-D-aspartate receptor antagonists in mice. / Refsgaard, Louise Konradsen; Pickering, Darryl S; Andreasen T., Jesper.
In: Behavioural Pharmacology, Vol. 28, No. 1, 01.02.2017, p. 37-47.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Binding and functional pharmacological characteristics of gepant-type antagonists in rat brain and mesenteric arteries. / Sheykhzade, Majid; Amandi, Nilofar; Pla, Monica Vidal; Abdolalizadeh, Bahareh; Sams, Anette; Warfvinge, Karin; Edvinsson, Lars; Pickering, Darryl S.
In: Vascular Pharmacology, Vol. 90, 10.02.2017, p. 36-43.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
In vitro and in vivo effects of a novel dimeric inhibitor of PSD‐95 on excitotoxicity and functional recovery after experimental traumatic brain injury. / Sommer, Jens Bak; Bach, Anders; Rytter, Hana Malá; Strømgaard, Kristian; Mogensen, Jesper; Pickering, Darryl S.
In: European Journal of Neuroscience, Vol. 45, No. 2, 20.01.2017, p. 238-248.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Effects of dimeric PSD-95 inhibition on excitotoxic cell death and outcome after controlled cortical impact in rats : PSD-95 inhibition in experimental TBI. / Sommer, Jens Bak; Bach, Anders; Rytter, Hana Malá; Gynther, Mikko; Bjerre, Ann-Sofie; Gram, Marie Gajhede; Marschner, Linda; Strømgaard, Kristian; Mogensen, Jesper; Pickering, Darryl S.
In: Neurochemical Research, Vol. 42, No. 12, 2017, p. 3401-3413.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Effects of the dimeric PSD-95 inhibitor UCCB01-144 on functional recovery after fimbria-fornix transection in rats. / Sommer, Jens Bak; Bach, Anders; Malá, Hana ; Strømgaard, Kristian; Mogensen, Jesper; Pickering, Darryl S.
In: Pharmacology, Biochemistry and Behavior, Vol. 161, 10.2017, p. 62-67.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Aryl- and heteroaryl-substituted phenylalanines as AMPA receptor ligands. / Szymańska, Ewa; Chałupnik, Paulina; Johansen, Tommy Nørskov; Nielsen, Birgitte; Cuñado Moral, Ana Maria; Pickering, Darryl S; Kieć-Kononowicz, Katarzyna.
In: Chemical Biology & Drug Design, Vol. 90, 01.12.2017, p. 1271-1281.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Pharmacological characterization and binding modes of novel racemic and optically active phenylalanine-based antagonists of AMPA receptors. / Szymańska, Ewa; Nielsen, Birgitte; Johansen, Tommy Nørskov; Cuñado Moral, Anna Maria; Pickering, Darryl S; Szczepańska, Katarzyna; Mickowska, Anna; Kieć-Kononowicz, Katarzyna.
In: European Journal of Medicinal Chemistry, Vol. 138, 2017, p. 874-883.Research output: Contribution to journal › Journal article › Research › peer-review
- 2018
- Published
(S)-2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements, Structural and Biological Investigation. / Brogi, Simone; Brindisi, Marghertia; Butini, Stefania; Kshirsagar, Giridhar; Maramai, Samuele; Chemi, Giulia; Gemma, Sandra; Campiani, Giuseppe; Novellino, Ettore; Fiorenzani, Paolo; Pinassi, Jessica; Aloisi, Anna Maria; Gynther, Mikko; Venskutonyte, Raminta; Han, Liwei; Frydenvang, Karla Andrea; Kastrup, Jette Sandholm Jensen; Pickering, Darryl S.
In: Journal of Medicinal Chemistry, Vol. 61, No. 5, 08.03.2018, p. 2124-2130.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Vascular and molecular pharmacology of the metabolically stable CGRP analogue, SAX. / Sheykhzade, Majid; Abdolalizadeh, Bahareh; Koole, Cassandra; Pickering, Darryl S; Dreisig, Karin; Johansson, Sara Ellinor; Abboud, Balsam Kadri; Dreier, Rasmus; Berg, Jais Oliver; Jeppesen, Jørgen Lykke; Sexton, Patrick; Edvinsson, Lars; Wootten, Denise; Sams, Anette.
In: European Journal of Pharmacology, Vol. 829, 2018, p. 85-92.Research output: Contribution to journal › Journal article › Research › peer-review
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Investigation of the presence and antinociceptive function of muscarinic acetylcholine receptors in the African naked mole-rat (Heterocephalus glaber)
Research output: Contribution to journal › Journal article › Research › peer-review
Published