Darryl S Pickering - Research outputs - Employees

Department of Drug Design and Pharmacology

Darryl S Pickering

Darryl S Pickering

Associate Professor

Molecular and Cellular Pharmacology
Jagtvej 160, 2100 København Ø, 22, Building: C213
- picker@sund.ku.dk
- https://drug.ku.dk/
Phone: +45 35 33 43 42

ORCID: 0000-0001-8687-6094

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Published
N-(7-(1H-imidazol-1-yl)-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl)benzamide - a new kainate receptor selective antagonist and analgesic : Synthesis, X-ray crystallography, structure-affinity relationships, in vitro and in vivo pharmacology. / Møllerud, Stine ; Hansen, Rie B; Pallesen, Jakob S; Temperini, Piero; Pasini, Diletta; Bornholdt, Jan; Nielsen, Birgitte ; Mamedova, Esmira; Chalupnik, Paulina; Paternain, Ana V; Lerma, Juan; Del Castillo, Marta Diaz ; Andreasen, Jesper T ; Frydenvang, Karla ; Kastrup, Jette Sandholm ; Johansen, Tommy N ; Pickering, Darryl S.
In: ACS Chemical Neuroscience, Vol. 10, 2019, p. 4685-4695.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
N1-Substituted Quinoxaline-2,3-diones as Kainate Receptor Antagonists: X-ray Crystallography, Structure-Affinity Relationships and in vitro Pharmacology. / Pallesen, Jakob Staun; Møllerud, Stine ; Frydenvang, Karla Andrea ; Pickering, Darryl S; Bornholt, Jan; Nielsen, Birgitte; Pasini, Diletta; Han, Liwei; Marconi, Laura; Kastrup, Jette Sandholm Jensen ; Johansen, Tommy Nørskov.
In: A C S Chemical Neuroscience, Vol. 10, 20.03.2019, p. 1841-1853.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Design and Synthesis of 2,3-trans-Proline Analogs as Ligands for the Ionotropic Glutamate Receptors and the Excitatory Amino Acid Transporters. / Poulie, Christian Bernard Matthijs; Alcaide Lopez, Anna; Krell-Jørgensen, Mikkel Poul; Larsen, Younes; Astier, Eloi; Bjørn-Yoshimoto, Walden E.; Yi, Feng; Syrenne, Jed T; Storgaard, Morten; Nielsen, Birgitte ; Frydenvang, Karla Andrea ; Jensen, Anders A.; Hansen, Kasper B; Pickering, Darryl S ; Bunch, Lennart.
In: A C S Chemical Neuroscience, Vol. 10, No. 6, 19.06.2019, p. 2989-3007.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
Use of the 4-Hydroxy-Triazole Moiety as a Bioisosteric Tool for the Development of Ionotropic Glutamate Receptor Ligands. / Sainas, Stefano; Temperini, Piero; Farnsworth, Jill C; Yi, Feng; Møllerud, Stine ; Jensen, Anders A.; Nielsen, Birgitte ; Kastrup, Jette Sandholm Jensen; Hansen, Kasper B; Boschi, Donatella; Pickering, Darryl S ; Clausen, Rasmus Prætorius; Lolli, Marco.
In: Journal of Medicinal Chemistry, Vol. 62, 09.05.2019, p. 4467-4482.
Research output: Contribution to journal › Journal article › Research › peer-review
Published
The Presence of Calcitonin Gene-Related Peptide and Its Receptors in Rat, Pig and Human Brain : Species Differences in Calcitonin Gene-Related Peptide Pharmacology. / Warfvinge, Karin; Edvinsson, Lars ; Pickering, Darryl S ; Sheykhzade, Majid.
In: Pharmacology, Vol. 104, 01.12.2019, p. 332-341.
Research output: Contribution to journal › Journal article › Research › peer-review

ID: 1299533