Jakob Staun Pallesen

Jakob Staun Pallesen

Postdoc


Publication year:
  1. 2019
  2. E-pub ahead of print

    A Comparative Assessment Study of Known Small-Molecule Keap1-Nrf2 Protein-Protein Interaction Inhibitors : Chemical Synthesis, Binding Properties, and Cellular Activity. / Tran, Kim Tai; Pallesen, Jakob S; Solbak, Sara Marie Øie; Narayanan, Dilip; Baig, Amina; Zang, Jie; Aguayo-Orozco, Alejandro; Carmona, Rosa; Garcia, Anthony; Bach, Anders.

    In: Journal of Medicinal Chemistry, 14.08.2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    N1-Substituted Quinoxaline-2,3-diones as Kainate Receptor Antagonists: X-ray Crystallography, Structure-Affinity Relationships and in vitro Pharmacology. / Pallesen, Jakob Staun; Møllerud, Stine; Frydenvang, Karla Andrea; Pickering, Darryl S; Bornholt, Jan; Nielsen, Birgitte; Pasini, Diletta; Han, Liwei; Marconi, Laura; Kastrup, Jette Sandholm Jensen; Johansen, Tommy Nørskov.

    In: A C S Chemical Neuroscience, Vol. 10, 20.03.2019, p. 1841-1853.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. 2018
  5. Published

    Non-covalent Small-Molecule Kelch-like ECH-Associated Protein 1-Nuclear Factor Erythroid 2-Related Factor 2 (Keap1-Nrf2) Inhibitors and Their Potential for Targeting Central Nervous System Diseases. / Pallesen, Jakob S; Tran, Kim T; Bach, Anders.

    In: Journal of Medicinal Chemistry, Vol. 61, No. 18, 11.05.2018, p. 8088-8103.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. 2017
  7. Published

    Pharmacology and crystal structure of novel 2,3-quinoxalinediones at kainate receptors. / Møllerud, Stine; Pallesen, Jakob Staun; Pasini, Diletta; Marconi, Laura; Han, Liwei; Bornholt, Jan; Johansen, Tommy Nørskov; Kastrup, Jette Sandholm ; Pickering, Darryl S; Frydenvang, Karla Andrea.

    In: Journal of Neurochemistry, Vol. 142, No. S1, MTU07-13, 08.2017, p. 124.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

ID: 137258903