Jesper Langgaard Kristensen

Jesper Langgaard Kristensen

Professor with special responsibilities


  1. Published

    Stereoselective synthesis of highly substituted bicyclic γ-lactones using homoaldol addition of 1-(1-cycloalkenyl)methyl carbamates. / Özlügedik, M.; Kristensen, Jesper Langgaard; Reuber, J.; Fröhlich, R.; Hoppe, D.

    In: Synthesis, No. 14, 01.10.2004, p. 2303-2316.

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Nonracemic, chiral homoenolate reagents derived from (cycloalk-1-enyl)methyl carbamates and evaluation of their configurational stabilities. / Özlügedik, M.; Kristensen, Jesper Langgaard; Wibbeling, B.; Fröhlich, R.; Hoppe, D.

    In: European Journal of Organic Chemistry, No. 3, 01.01.2002, p. 414-427.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Palladium-catalyzed asymmetric allylic alkylation of a-aryl ketones. / Trost, B.M.; Schroeder, G.M.; Kristensen, Jesper Langgaard.

    In: Angewandte Chemie International Edition, Vol. 41, No. 18, 16.09.2002, p. 3492-3495.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    A Prodrug Approach Involving In Situ Depot Formation to Achieve Localized and Sustained Action of Diclofenac After Joint Injection. / Thing, Mette; Agårdh, Li; Larsen, Susan; Rasmussen, Rune; Pallesen, Jakob; Mertz, Nina; Kristensen, Jesper Langgaard; Hansen, Martin; Ostergaard, Jesper; Larsen, Claus Selch.

    In: Journal of Pharmaceutical Sciences, Vol. 103, No. 12, 2014, p. 4021–4029.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Synthesis and binding studies of 2-arylapomorphines. / Søndergaard, Kåre; Kristensen, Jesper Langgaard; Palner, Mikael; Gillings, Nic; Knudsen, Gitte Moos; Roth, Bryan; Begtrup, M.

    In: Organic & Biomolecular Chemistry, Vol. 3, No. 22, 21.11.2005, p. 4077-4081.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Synthesis of (R)-(-)-2-fluoronorapomorphine - A precursor for the synthesis of (R)-(-)-2-fluoro-N-[C]propylnorapomorphine for evaluation as a dopamine D agonist ligand for PET investigations. / Søndergaard, Kåre; Kristensen, Jesper Langgaard; Gillings, Nic; Begtrup, M.

    In: European Journal of Organic Chemistry, No. 20, 14.10.2005, p. 4428-4433.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Accepted/In press

    Convenient Entry to 18 F-Labeled Amines through the Staudinger Reduction. / Stéen, E. Johanna L.; Shalgunov, Vladimir; Denk, Christoph; Mikula, Hannes; Kjær, Andreas; Kristensen, Jesper L.; Herth, Matthias M.

    In: European Journal of Organic Chemistry, 01.01.2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Improved radiosynthesis and preliminary in vivo evaluation of the 11 C-labeled tetrazine [ 11 C]AE-1 for pretargeted PET imaging. / Stéen, E. Johanna L.; Jørgensen, Jesper T.; Petersen, Ida N.; Nørregaard, Kamilla; Lehel, Szabolcs; Shalgunov, Vladimir; Birke, Alexander; Edem, Patricia E.; L'Estrade, Elina T.; Hansen, Hanne D.; Villadsen, Jonas; Erlandsson, Maria; Ohlsson, Tomas; Yazdani, Abdolreza; Valliant, John F.; Kristensen, Jesper L.; Barz, Matthias; Knudsen, Gitte M.; Kjær, Andreas; Herth, Matthias M.

    In: Bioorganic and Medicinal Chemistry Letters, 01.01.2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Development of a simple proton nuclear magnetic resonance-based procedure to estimate the approximate distribution coefficient at physiological pH (logD7.4) : Evaluation and comparison to existing practices. / Stéen, E Johanna L; Nyberg, Nils; Lehel, Szabolcs; Andersen, Valdemar L; Di Pilato, Pantaleo; Knudsen, Gitte M; Kristensen, Jesper L; Herth, Matthias M.

    In: Bioorganic & Medicinal Chemistry Letters, Vol. 27, No. 2, 15.01.2017, p. 319-322.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Trans-cyclooctene-functionalized PeptoBrushes with improved reaction kinetics of the tetrazine ligation for pretargeted nuclear imaging : [Meeting Abstract]. / Steen, Johanna; Norregard, Kamilla; Johann, Kerstin; Jorgensen, Jesper; Svatunek, Dennis; Birke, Alexander; Edem, Patricia; Rossin, Raffaella; Seidl, Christine; Schmid, Friederike; Robillard, Marc; Mikula, Hannes; Kristensen, Jesper; Barz, Matthias; Kjaer, Andreas; Herth, Matthias.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 62, No. Supl. 1/SI, 05.2019, p. S109-S110.

    Research output: Contribution to journalConference abstract in journalResearch

  11. Published

    Towards the Dual Click F-18-labeling of Antibodies. / Steen, Johanna; Denk, Christoph; Norregaard, Kamilla; Jorgensen, Jesper; Rossin, Raffaella; Svatunek, Dennis; Edem, Patricia; Robillard, Marc; Kjaer, Andreas; Kristensen, Jesper; Mikula, Hannes; Herth, Matthias.

    2018.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  12. Published

    Pretargeted PET imaging using a dual click F-18-labeling strategy : [Meeting Abstract]. / Steen, Johanna; Denk, Christoph; Jorgensen, Jesper; Norregard, Kamilla; Rossin, Raffaella; Wilkovitsch, Martin; Svatunek, Dennis; Edem, Patricia; Kuntner, Claudia; Wanek, Thomas; Robillard, Marc; Kristensen, Jesper; Kjaer, Andreas; Mikula, Hannes; Herth, Matthias.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 62, No. Supl. 1/SI, O-08, 05.2019, p. S22-S23.

    Research output: Contribution to journalConference abstract in journalResearch

  13. Published
  14. Published

    Convenient access to F-18-labeled amines through the Staudinger reduction. / Shalgunov, Vladimir; Steen, Johanna; Denk, Christoph; Mikula, Hannes; Kjaer, Andreas; Kristensen, Jesper; Herth, Matthias.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 62, No. Supl. 1/SI, P-050, 05.2019, p. S205-S206.

    Research output: Contribution to journalConference abstract in journalResearch

  15. Published

    Snegleprotein øger forståelsen af vigtige receptorer i hjernen. / Shahsavar, Azadeh; Nielsen, Elsebeth Ø.; Kristensen, Jesper Langgaard; Gajhede, Michael; Balle, Thomas; Kastrup, Jette Sandholm Jensen.

    In: Lægemiddelforskning, Vol. 2012, 2012, p. 48-50.

    Research output: Contribution to journalJournal articleCommunication

  16. Published

    Crystal Structure of Lymnaea stagnalis AChBP Complexed with the Potent nAChR Antagonist DHßE Suggests a Unique Mode of Antagonism. / Shahsavar, Azadeh; Kastrup, Jette S; Nielsen, Elsebet Ø.; Kristensen, Jesper L; Gajhede, Michael; Balle, Thomas.

    In: P L o S One, Vol. 7, No. 8, 2012, p. e40757.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Radiolabelling and PET brain imaging of the a1-adrenoceptor antagonist Lu AE43936. / Risgaard, Rune; Ettrup, Anders Janusz; Balle, Thomas; Dyssegaard, Agnete; Hansen, Hanne Demant; Lehel, Szabolcs; Madsen, Jacob; Pedersen, Henrik; Püschl, Ask; Badolo, Lassina; Bang-Andersen, Benny; Knudsen, Gitte Moos; Kristensen, Jesper Langgaard.

    In: Nuclear Medicine & Biology, Vol. 40, No. 1, 2013, p. 135-140.

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Synthesis and SAR study of a novel series of dopamine receptor agonists. / Risgaard, R.; Jensen, M.; Jørgensen, M.; Bang-Andersen, B.; Christoffersen, C.T.; Jensen, Klaus Gervig; Kristensen, Jesper Langgaard; Püschl, A.

    In: Bioorganic and Medicinal Chemistry, Vol. 22, No. 1, 01.01.2014, p. 381-392.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Synthesis and biological evaluation of 4-(aminomethyl)-1-hydroxypyrazole analogues of muscimol as ¿-aminobutyric acidA receptor agonists. / Petersen, Jette Gellert; Bergmann, Rikke; Møller, Henriette A.; Jørgensen, Charlotte Grube; Nielsen, Birgitte; Kehler, Jan; Frydenvang, Karla ; Kristensen, Jesper; Balle, Thomas; Jensen, Anders A.; Kristiansen, Uffe; Frølund, Bente.

    In: Journal of Medicinal Chemistry, Vol. 56, No. 3, 2013, p. 993-1006.

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Convergent [18]F-labeling and evaluation of N-benzyl-phenethylamines as 5-HT2A receptor PET ligands. / Petersen, Ida Nymann; Villadsen, Jonas; Hansen, Hanne Demant; Jensen, Anders A; Lehel, Szabolcs; Gillings, Nic; Herth, Matthias M; Knudsen, Gitte M; Kristensen, Jesper L.

    In: Bioorganic & Medicinal Chemistry, Vol. 24, 2016, p. 5353-5356.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Nucleophilic 18F-Labeling of Spirocyclic Iodonium Ylide or Boronic Pinacol Ester Precursors - Advantages and Disadvantages. / Petersen, Ida Nymann; Kristensen, Jesper Langgaard; Herth, Matthias Manfred.

    In: European Journal of Organic Chemistry, Vol. 2017, No. 3, 18.01.2017, p. 453-458.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Identification of a new metabolite of GHB : gamma-hydroxybutyric acid glucuronide. / Petersen, Ida Nymann; Tortzen, Christian; Kristensen, Jesper Langgaard; Pedersen, Daniel Sejer; Breindahl, Torben.

    In: Journal of Analytical Toxicology, Vol. 37, No. 5, 06.2013, p. 291-7.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Tying up Nicotine: New Selective Competitive Antagonist of the Neuronal Nicotinic Acetylcholine Receptors. / Petersen, Ida Nymann; Crestey, François; Jensen, Anders A; Indurthi, Dinesh C; Pedersen, Henrik; Andreasen, Jesper T; Balle, Thomas; Kristensen, Jesper L.

    In: A C S Medicinal Chemistry Letters, Vol. 6, No. 4, 09.04.2015, p. 472-475.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Synthesis and stability study of a new major metabolite of gamma-hydroxybutyric acid. / Petersen, Ida Nymann; Kristensen, Jesper Langgaard; Tortzen, Christian; Breindahl, Torben; Pedersen, Daniel Sejer.

    In: Beilstein Journal of Organic Chemistry, Vol. 9, 2013, p. 641-646.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Total synthesis of ascididemin via anionic cascade ring closure. / Petersen, Ida Nymann; Crestey, François; Kristensen, Jesper Langgaard.

    In: Chemical Communications, Vol. 48, No. 72, 2012, p. 9092-9094.

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Synthesis of Pyridoacridines through Anionic Cascade Ring Closure. / Petersen, I.N.; Kristensen, Jesper Langgaard.

    In: Synthesis, Vol. 46, 01.01.2014, p. 1469-1474.

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    18F-Labelling of electron rich iodonium ylides : application to the radiosynthesis of potential 5-HT2A receptor PET ligands. / Petersen, I N; Villadsen, J; Hansen, H D; Madsen, J; Jensen, A A; Gillings, N; Lehel, Szabolcs; Herth, M M; Knudsen, G M; Kristensen, J L.

    In: Organic & Biomolecular Chemistry, Vol. 15, 04.2017, p. 4351-4358.

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Aminolysis of resin-bound N-nosylaziridine-2-carboxylic acids. / Olsen, Christian A; Christensen, Caspar; Nielsen, Birgitte; Farah, Mohamed M; Mohamed, Farah M; Witt, Matthias; Clausen, Rasmus P; Kristensen, Jesper L; Franzyk, Henrik; Jaroszewski, Jerzy W.

    In: Organic Letters, Vol. 8, No. 15, 2006, p. 3371-4.

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    Synthesis of N-alkylated amino acids using fluorous-tagged hydroxylamines. / Nielsen, Simon Dalsgaard; Smith, Garrick P; Begtrup, Mikael; Kristensen, Jesper Langgaard.

    In: Tetrahedron, Vol. 67, No. 29, 22.07.2011, p. 5261-5267.

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    Amination of aryl iodides using a fluorous-tagged ammonia equivalent. / Nielsen, Simon Dalsgaard; Smith, Garrick; Begtrup, Mikael; Kristensen, Jesper Langgaard.

    In: European Journal of Organic Chemistry, Vol. 2010, No. 19, 2010, p. 3704-3710.

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    Synthesis and application of a new fluorous-tagged ammonia equivalent. / Nielsen, Simon Dalsgaard; Smith, Garrick; Begtrup, Mikael; Kristensen, Jesper Langgaard.

    In: Chemistry: A European Journal, Vol. 16, No. 15, 2010, p. 4557-4566.

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Synthesis and characterisation of substrate-based peptides as inhibitors of histone demethylase KDM4C. / Nielsen, Simon D; Leurs, Ulrike; Bergner, Magnus; Barris, Silvia Amor; Devkota, Kanchan; Meyer, Kamilla; Iaria, Daniella; McCaughan, Jack; Lohse, Brian; Kristensen, Jesper L; Clausen, Rasmus Prætorius.

    In: Protein and Peptide Letters, Vol. 23, No. 9, 13.06.2016, p. 772 - 776.

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Characterization of the hepatic cytochrome P450 enzymes involved in the metabolism of 25I-NBOMe and 25I-NBOH. / Nielsen, Line Marie; Holm, Niels Bjerre; Leth-Petersen, Sebastian; Kristensen, Jesper Langgaard; Olsen, Lars; Linnet, Kristian.

    In: Drug Testing and Analysis, Vol. 9, No. 5, 2017, p. 671–679.

    Research output: Contribution to journalJournal articleResearchpeer-review

  34. Published

    Novel 4-(piperidin-4-yl)-1-hydroxypyrazoles as gamma-aminobutyric acidA receptor ligands : synthesis, pharmacology, and structure-activity relationships. / Møller, Henriette A; Sander, Tommy; Kristensen, Jesper Langgaard; Nielsen, Birgitte; Krall, Jacob; Bergmann, Marianne Lerbæk; Christiansen, Bolette; Balle, Thomas; Jensen, Anders Asbjørn; Frølund, Bente Flensborg.

    In: Journal of Medicinal Chemistry, Vol. 53, No. 8, 2010, p. 3417-3421.

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. Published

    Long-Acting Diclofenac Ester Prodrugs for Joint Injection : Kinetics, Mechanism of Degradation, and In Vitro Release From Prodrug Suspension. / Mertz, Nina; Larsen, Susan Weng; Kristensen, Jesper; Østergaard, Jesper; Larsen, Claus.

    In: Journal of Pharmaceutical Sciences, Vol. 105, No. 10, 27.07.2016, p. 3079–3087.

    Research output: Contribution to journalJournal articleResearchpeer-review

  36. Published

    Synthesis of substituted 2-cyanoarylboronic esters. / Lysén, Morten; Hansen, Henriette M; Begtrup, Mikael; Kristensen, Jesper L.

    In: Journal of Organic Chemistry, Vol. 71, No. 6, 17.03.2006, p. 2518-20.

    Research output: Contribution to journalJournal articleResearchpeer-review

  37. Published

    Synthesis of tertiary benzamides via Pd-catalyzed coupling of arylboronic esters and carbamoyl chlorides. / Lysén, M.; Kelleher, Susan; Begtrup, M.; Kristensen, Jesper Langgaard.

    In: Journal of Organic Chemistry, Vol. 70, No. 13, 24.06.2005, p. 5342-5343.

    Research output: Contribution to journalJournal articleResearchpeer-review

  38. Published

    Convergent synthesis of 6-substituted phenanthridines via anionic ring closure. / Lysén, M.; Kristensen, Jesper Langgaard; Vedsø, P.; Begtrup, M.

    In: Organic Letters, Vol. 4, No. 2, 01.01.2002, p. 257-259.

    Research output: Contribution to journalJournal articleResearchpeer-review

  39. Published

    Synthesis, cross-coupling, and anionic cyclization of ortho-substituted naphthaleneboronic esters. / Lysén, M.; Madden, M.; Kristensen, Jesper Langgaard; Vedsø, P.; Zöllner, C.; Begtrup, M.

    In: Synthesis, No. 20, 17.10.2006, p. 3478-3484.

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    Posttranslational Modifications of the Histone 3 Tail and Their Impact on the Activity of Histone Lysine Demethylases In Vitro. / Lohse, Brian; Helgstrand, Charlotte; Andersson, Jan Legaard; Leurs, Ulrike; Cloos, Paul Andreas Compare; Kristensen, Jesper Langgaard; Clausen, Rasmus Prætorius.

    In: P L o S One, Vol. 8, No. 7, 02.07.2013, p. e67653.

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    Targeting histone lysine demethylases by truncating the histone 3 tail to obtain selective substrate-based inhibitors. / Lohse, Brian; Nielsen, Anders L; Kristensen, Jan B L; Helgstrand, Charlotte; Cloos, Paul Andreas Compare; Olsen, Lars; Gajhede, Michael; Clausen, Rasmus Prætorius; Kristensen, Jesper Langgaard.

    In: Angewandte Chemie International Edition, Vol. 50, No. 39, 19.09.2011, p. 9100-9103.

    Research output: Contribution to journalJournal articleResearchpeer-review

  42. Published

    Inhibitors of histone demethylases. / Lohse, Brian; Kristensen, Jesper L; Kristensen, Line H; Agger, Karl; Helin, Kristian; Gajhede, Michael; Clausen, Rasmus P.

    In: Bioorganic & Medicinal Chemistry, Vol. 19, No. 12, 01.02.2011, p. 3625-3636.

    Research output: Contribution to journalReviewResearchpeer-review

  43. Published

    Inhibitor scaffold for the histone lysine demethylase KDM4C (JMJD2C). / Leurs, Ulrike; Clausen, Rasmus P; Kristensen, Jesper L; Lohse, Brian.

    In: Bioorganic & Medicinal Chemistry Letters, Vol. 22, No. 18, 15.09.2012, p. 5811-3.

    Research output: Contribution to journalJournal articleResearchpeer-review

  44. Published

    Dissecting the Binding Mode of Low Affinity Phage Display Peptide Ligands to Protein Targets by Hydrogen/Deuterium Exchange Coupled to Mass Spectrometry. / Leurs, Ulrike; Lohse, Brian; Ming, Shonoi A; Cole, Philip A; Clausen, Rasmus P; Kristensen, Jesper L; Rand, Kasper D.

    In: Analytical Chemistry, Vol. 86, No. 23, 17.10.2014, p. 11734-11741.

    Research output: Contribution to journalJournal articleResearchpeer-review

  45. Published

    Substrate- and Cofactor-independent Inhibition of Histone Demethylase KDM4C. / Leurs, Ulrike; Lohse, Brian; Rand, Kasper Dyrberg; Ming, Shonoi; Riise, Erik Skjold; Cole, Philip A.; Kristensen, Jesper Langgaard; Clausen, Rasmus Prætorius.

    In: A C S Chemical Biology, Vol. 9, No. 9, 11.07.2014, p. 2131-2138.

    Research output: Contribution to journalJournal articleResearchpeer-review

  46. Published

    Metabolic fate of hallucinogenic NBOMes. / Leth-Petersen, Sebastian; Gabel-Jensen, Charlotte; Gillings, Nic; Lehel, Szabolzs; Hansen, Hanne D; Knudsen, Gitte M; Kristensen, Jesper L.

    In: Chemical Research in Toxicology, Vol. 29, No. 1, 2016, p. 96–100.

    Research output: Contribution to journalJournal articleResearchpeer-review

  47. Published

    5-HT2A/5-HT2C receptor pharmacology and intrinsic clearance of N-benzylphenethylamines modified at the primary site of metabolism. / Leth-Petersen, Sebastian; Petersen, Ida Nymann; Jensen, Anders A; Bundgaard, Christoffer; Bæk, Mathias; Kehler, Jan; Kristensen, Jesper L.

    In: A C S Chemical Neuroscience, 26.08.2016, p. 1-6.

    Research output: Contribution to journalJournal articleResearchpeer-review

  48. Published

    Correlating the Metabolic Stability of Psychedelic 5-HT2A Agonists with Anecdotal Reports of Human Oral Bioavailability. / Leth-Petersen, Sebastian; Bundgaard, Christoffer; Hansen, Martin; Carnerup, Martin A; Kehler, Jan; Kristensen, Jesper Langgaard.

    In: Neurochemical Research, Vol. 39, No. 10, 12.02.2014, p. 2018-2023.

    Research output: Contribution to journalJournal articleResearchpeer-review

  49. Published

    Medicindepot dannes efter injektion i leddet. / Larsen, Susan Weng; Thing, Mette Agergaard; Østergaard, Jesper; Kristensen, Jesper Langgaard; Hansen, Martin; Larsen, Claus Selch.

    In: Lægemiddelforskning, Vol. 2013, 2013, p. 38-40.

    Research output: Contribution to journalJournal articleResearch

  50. Published

    IMIDAZOLE DERIVATIVES AS PRODRUGS OF DICLOFENAC. / Larsen, Claus Selch (Inventor); Larsen, Susan Weng (Inventor); Thing, Mette Agergaard (Inventor); Kristensen, Jesper Langgaard (Inventor); JENSEN, HENRIK (Inventor); ØSTERGAARD, JESPER (Inventor).

    IPC No.: A61P 29/ 00 A I. Patent No.: WO2016066612.

    Research output: PatentResearch

  51. Published

    PRODRUGS OF NON- STEROID ANTI - INFLAMMATORY AGENTS (NSAIDS). / Larsen, Claus Selch (Inventor); Larsen, Susan Weng (Inventor); Thing, Mette Agergaard (Inventor); Kristensen, Jesper Langgaard (Inventor); JENSEN, HENRIK (Inventor); OESTERGAARD, JESPER (Inventor).

    IPC No.: C07D 487/ 04 A I. Patent No.: WO2013064153.

    Research output: PatentResearch

  52. Published

    PRODRUGS OF NAPROXEN AND DICLOFENAC. / Larsen, Claus Selch (Inventor); Larsen, Susan Weng (Inventor); Thing, Mette Agergaard (Inventor); Kristensen, Jesper Langgaard (Inventor); JENSEN, HENRIK (Inventor); ØSTERGAARD, JESPER (Inventor).

    IPC No.: A61K 45/ 06 A I. Patent No.: US2016074523.

    Research output: PatentResearch

  53. Published

    Computational Methods to Predict the Regioselectivity of Electrophilic Aromatic Substitution Reactions of Heteroaromatic Systems. / Kruszyk, Monika; Jessing, Mikkel; Kristensen, Jesper L; Jorgensen, Morten.

    In: Journal of Organic Chemistry, Vol. 81, No. 12, 13.05.2016, p. 5128–5134.

    Research output: Contribution to journalJournal articleResearchpeer-review

  54. Published

    Synthesis of ortho substituted arylboronic esters by in situ trapping of unstable lithio intermediates : 2-(5,5-Dimethyl-1,3,2-dioxaborinan-2-YL)Benzoic acid ethyl ester: [Benzoic acid, 2-(5,5-dimethyl-1,3,2-dioxaborinan-2-yl)-, ethyl ester]. / Kristensen, Jesper Langgaard; Lysén, Morten; Vedsø, Per; Begtrup, Mikael.

    In: Organic Syntheses, Vol. 81, 01.01.2005, p. 134-139.

    Research output: Contribution to journalJournal articleResearchpeer-review

  55. Published

    Synthesis of RHPS4 via an anionic ring closing cascade. / Kristensen, Jesper Langgaard.

    In: Tetrahedron Letters, Vol. 49, No. 15, 2008, p. 2351-2354.

    Research output: Contribution to journalJournal articleResearchpeer-review

  56. Published

    Synthesis of Ortho Substituted Arylboronic Esters by in Situ Trapping of Unstable Lithio Intermediates. / Kristensen, Jesper Langgaard; Lysén, M.; Vedsø, Per; Begtrup, M.

    In: Organic Letters, Vol. 3, No. 10, 17.05.2001, p. 1435-1437.

    Research output: Contribution to journalLetterResearchpeer-review

  57. Published

    Synthesis of novel azaxanthones derived from N-hydroxyazoles. / Kristensen, Jesper Langgaard; Vedsø, P.; Begtrup, M.

    In: Tetrahedron, Vol. 58, No. 12, 18.03.2002, p. 2397-2404.

    Research output: Contribution to journalJournal articleResearchpeer-review

  58. Published

    Ny bioisoster kan skabe nye lægemidler. / Kristensen, Jesper Langgaard; Clausen, Rasmus Prætorius.

    In: Lægemiddelforskning, Vol. 2004, 2004, p. 16-17.

    Research output: Contribution to journalJournal articleCommunication

  59. Published

    Preparation of 5-acyl- and 5-aryl-substituted 1-(benzyloxy)pyrazoles via directed ortho-lithiation/transmetalation and palladium catalyzed cross- coupling. / Kristensen, Jesper Langgaard; Begtrup, M.; Vedsø, P.

    In: Synthesis, No. 11, 01.11.1998, p. 1604-1608.

    Research output: Contribution to journalJournal articleResearchpeer-review

  60. Published

    Exploring the neuroleptic substituent in octoclothepin : potential ligands for positron emission tomography with subnanomolar affinity for alpha1-adrenoceptors. / Kristensen, Jesper Langgaard; Pu¨schl, Ask; Jensen, Martin; Risgaard, Rune; Christoffersen, Claus T; Bang-Andersen, Benny; Balle, Thomas.

    In: Journal of Medicinal Chemistry, Vol. 53, No. 19, 2010, p. 7021-7034.

    Research output: Contribution to journalJournal articleResearchpeer-review

  61. Published

    Histonhaler : et nyt mål inden for kræftbehandling. / Kristensen, Jesper Langgaard; Lohse, Brian; Clausen, Rasmus Prætorius.

    In: Lægemiddelforskning, Vol. 2010, 12.2010, p. 7-9.

    Research output: Contribution to journalJournal articleCommunication

  62. Published

    Synthesis of pentacyclic 13-azadibenzo[a,de]anthracenes via anionic cascade ring closure. / Kristensen, Jesper Langgaard; Vedsø, P.; Begtrup, M.

    In: Journal of Organic Chemistry, Vol. 68, No. 10, 16.05.2003, p. 4091-4092.

    Research output: Contribution to journalJournal articleResearchpeer-review

  63. Published

    Textbook of Drug Design and Discovery : In vivo imaging in drug discovery. / Kristensen, Jesper Langgaard; Herth, Matthias Manfred.

    Textbook of Drug Design and Discovery. Fifth edition. ed. CRC Press, 2017.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  64. Published

    Enzyme kinetic studies of histone demethylases KDM4C and KDM6A : Towards understanding selectivity of inhibitors targeting oncogenic histone demethylases. / Kristensen, Jan B L; Nielsen, Anders L; Jørgensen, Lars; Kristensen, Line Hyltoft; Helgstrand, Charlotte; Juknaite, Lina; Kristensen, Jesper Langgaard; Kastrup, Jette Sandholm; Clausen, Rasmus Prætorius; Olsen, Lars; Gajhede, Michael.

    In: F E B S Letters, Vol. 585, No. 12, 23.06.2011, p. 1951-1956.

    Research output: Contribution to journalJournal articleResearchpeer-review

  65. Published

    Conformationally Constrained Peptidomimetics as Inhibitors of the Protein Arginine Methyl Transferases. / Knuhtsen, Astrid; Legrand, Baptiste; Van der Poorten, Olivier; Amblard, Muriel; Martinez, Jean; Ballet, Steven; Kristensen, Jesper L; Pedersen, Daniel Sejer.

    In: Chemistry: A European Journal, Vol. 22, No. 39, 12.08.2016, p. 14022–14028.

    Research output: Contribution to journalJournal articleResearchpeer-review

  66. Published

    The importance of small polar radiometabolites in molecular neuroimaging : A PET study with [11C]Cimbi-36 labeled in two positions. / Johansen, Annette; Hansen, Hanne D; Svarer, Claus; Lehel, Szabolcs; Leth-Petersen, Sebastian; Kristensen, Jesper L; Gillings, Nic; Knudsen, Gitte M.

    In: Journal of Cerebral Blood Flow and Metabolism, Vol. 38, No. 4, 04.2018, p. 659-668.

    Research output: Contribution to journalJournal articleResearchpeer-review

  67. Published

    Human biodistribution and radiation dosimetry of the 5-HT2A receptor agonist Cimbi-36 labeled with carbon-11 in two positions. / Johansen, Annette; Holm, Søren; Dall, Bente; Keller, Sune; Kristensen, Jesper L; Knudsen, Gitte M; Hansen, Hanne D.

    In: EJNMMI Research, Vol. 9, 71, 2019, p. 1-10.

    Research output: Contribution to journalJournal articleResearchpeer-review

  68. Published

    A strategic approach to [6,6]-bicyclic lactones : application towards the CD fragment of DHβE. / Jepsen, Tue Heesgaard; Glibstrup, Emil; Crestey, Francois Louis Jean; Jensen, Anders A.; Kristensen, Jesper Langgaard.

    In: Beilstein Journal of Organic Chemistry, Vol. 13, 2017, p. 988-994.

    Research output: Contribution to journalJournal articleResearchpeer-review

  69. Published

    In situ generation of the Ohira-Bestmann Reagent from stable sulfonyl azide : scalable synthesis of alkynes from aldehydes. / Jepsen, Tue Heesgaard; Kristensen, Jesper Langgaard.

    In: Journal of Organic Chemistry, Vol. 79, No. 19, 12.09.2014, p. 9423-9426.

    Research output: Contribution to journalJournal articleResearchpeer-review

  70. Published

    Synthesis and pharmacological evaluation of DHβE analogs as neuronal nicotinic acetylcholine receptor antagonists. / Jepsen, Tue H.; Jensen, Anders A.; Lund, Mads Henrik; Glibstrup, Emil; Kristensen, Jesper Langgaard.

    In: A C S Medicinal Chemistry Letters, Vol. 5, No. 7, 2014, p. 766-770.

    Research output: Contribution to journalJournal articleResearchpeer-review

  71. Published

    Detailed characterization of the in vitro pharmacological and pharmacokinetic properties of N-(2-hydroxybenzyl)-2,5-dimethoxy-4-cyanophenylethylamine (25CN-NBOH), a highly selective and brain-penetrant 5-HT2A receptor agonist. / Jensen, Anders A; McCorvy, John D; Petersen, Sebastian Leth; Bundgaard, Christoffer; Liebscher, Gudrun; Kenakin, Terry P; Bräuner-Osborne, Hans; Kehler, Jan; Kristensen, Jesper L.

    In: Journal of Pharmacology and Experimental Therapeutics, Vol. 361, No. 3, 2017, p. 441-453.

    Research output: Contribution to journalJournal articleResearchpeer-review

  72. Published

    Structure-activity relationships of constrained phenylethylamine ligands for the serotonin 5-ht2 receptors. / Isberg, Vignir; Paine, James; Leth-Petersen, Sebastian; Kristensen, Jesper Langgaard; Gloriam, David E.

    In: P L o S One, Vol. 8, No. 11, e78515, 2013.

    Research output: Contribution to journalJournal articleResearchpeer-review

  73. Published

    Correction : Structure-activity relationships of constrained phenylethylamine ligands for the serotonin 5-HT2 receptors (PLoS ONE). / Isberg, Vignir; Paine, James; Leth-Petersen, Sebastian; Kristensen, Jesper L.; Gloriam, David E.

    In: PLOS ONE, Vol. 9, No. 1, 17.01.2014.

    Research output: Contribution to journalComment/debateResearchpeer-review

  74. Published

    Development of C-11-labeled oxindole derivatives for in vivo PET imaging of the 5-HT7 receptor. / Herth, Matthias Manfred; Hansen, Hanne; Andersen, Valdemar L.; Volk, Balazs; Ettrup, Anders; Antoni, Ferenc; Lehel, Szabolcs; Dyssegaard, Agnete; Kristensen, Jesper L.; Knudsen, Gitte M.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 56, 05.2013, p. S82-S82.

    Research output: Contribution to journalJournal articleResearchpeer-review

  75. Published

    Accelerating preclinical PET-screening: reductive amination with [11C]methoxybenzaldehydes. / Herth, Matthias Manfred; Leth-Petersen, Sebastian; Lehel, Szabolcs; Hansen, Martin; Gillings, Nic; Madsen, Jacob; Kristensen, Jesper Langgaard.

    In: R S C Advances, Vol. 41, 2014, p. 21347-21350.

    Research output: Contribution to journalJournal articleResearchpeer-review

  76. Published

    Development of a 11C-labeled tetrazine for rapid tetrazine–trans-cyclooctene ligation. / Herth, Matthias Manfred; Andersen, Valdemar L. ; Lehel, Szabolcs; Madsen, Jacob; Knudsen, Gitte Moos; Kristensen, Jesper Langgaard.

    In: Chemical Communications, Vol. 49, 2013, p. 3805-3807.

    Research output: Contribution to journalJournal articleResearchpeer-review

  77. Published

    Synthesis and In Vitro Evaluation of Oxindole Derivatives as Potential Radioligands for 5-HT7 Receptor Imaging with PET. / Herth, Matthias Manfred; Volk, Balázs; Pallagi, Katalin; Koefoed Bech, Lasse; A. Antoni, Ferenc; Knudsen, Gitte Moos; Kristensen, Jesper Langgaard.

    In: ACS Chemical Neuroscience, Vol. 3, No. 12, 31.08.2012, p. 1002-1007.

    Research output: Contribution to journalJournal articleResearchpeer-review

  78. Published

    Development of New PET Radiotracers for In Vivo 5-HT7 Brain Imaging. / Herth, Matthias Manfred; Hansen, Hanne; Lehel, Szabolcs; Ettrup, Anders; Paine, James; Madsen, Jacob; Gillings, Nic; Kristensen, Jesper; Knudsen, Gitte.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 54, 2011, p. S277-S277.

    Research output: Contribution to journalJournal articleResearchpeer-review

  79. Published

    Synthesis and evaluation of [11C]Cimbi-806 as a potential PET ligand for 5-HT7 receptor imaging. / Herth, Matthias Manfred; Hansen, Hanne Demant; Ettrup, Anders Janusz; Dyssegaard, Agnete; Lehel, Szabolcs; Kristensen, Jesper Langgaard; Knudsen, Gitte Moos.

    In: Bioorganic and Medicinal Chemistry, Vol. 20, No. 14, 2012, p. 4574-4581.

    Research output: Contribution to journalJournal articleResearchpeer-review

  80. Published

    Evaluation of 3-Ethyl-3-(phenylpiperazinylbutyl)oxindoles as PET Ligands for the Serotonin 5-HT7 Receptor : Synthesis, Pharmacology, Radiolabeling, and in Vivo Brain Imaging in Pigs. / Herth, Matthias M; Andersen, Valdemar L; Hansen, Hanne D; Stroth, Nikolas; Volk, Balázs; Lehel, Szabolcs; Dyssegaard, Agnete; Ettrup, Anders; Svenningsson, Per; Knudsen, Gitte M; Kristensen, Jesper Langgaard.

    In: Journal of Medicinal Chemistry, Vol. 58, No. 8, 13.04.2015, p. 3631–3636.

    Research output: Contribution to journalJournal articleResearchpeer-review

  81. Published

    Synthesis and evaluation of 18F-labeled 5-HT2A receptor agonists as PET ligands. / Herth, Matthias M; Petersen, Ida Nymann; Hansen, Hanne Demant; Hansen, Martin; Ettrup, Anders; Jensen, Anders A; Lehel, Szabolcs; Dyssegaard, Agnete; Gillings, Nic; Knudsen, Gitte M; Kristensen, Jesper L.

    In: Nuclear Medicine and Biology, Vol. 43, No. 8, 19.04.2016, p. 455-462.

    Research output: Contribution to journalJournal articleResearchpeer-review

  82. Published

    Synthesis and pharmacological evaluation of N-benzyl substituted 4-bromo-2,5-dimethoxyphenethylamines as 5-HT2A/2C partial agonists. / Hansen, Martin; Jacobsen, Stine Engesgaard; Plunkett, Shane; Liebscher, Gudrun Eckhard; McCorvy, John D; Bräuner-Osborne, Hans; Kristensen, Jesper Langgaard.

    In: Bioorganic & Medicinal Chemistry, Vol. 23, No. 14, 2015, p. 3933-3937.

    Research output: Contribution to journalJournal articleResearchpeer-review

  83. Published

    Synthesis and structure-activity relationships of N-benzyl phenethylamines as 5-HT2A/2C agonists. / Hansen, Martin; Phonekeo, Karina; Paine, James S; Leth-Petersen, Sebastian; Begtrup, Mikael; Bräuner-Osborne, Hans; Kristensen, Jesper Langgaard.

    In: A C S Chemical Neuroscience, Vol. 5, No. 3, 07.01.2014, p. 243-249.

    Research output: Contribution to journalJournal articleResearchpeer-review

  84. Published

    Tweaking agonist efficacy at N-methyl-D-aspartate receptors by site-directed mutagenesis. / Hansen, Kasper B; Clausen, Rasmus P; Bjerrum, Esben J; Bechmann, Christian; Greenwood, Jeremy R; Christensen, Caspar; Kristensen, Jesper L; Egebjerg, Jan; Bräuner-Osborne, Hans.

    In: Molecular Pharmacology, Vol. 68, No. 6, 12.2005, p. 1510-23.

    Research output: Contribution to journalJournal articleResearchpeer-review

  85. Published

    Synthesis of azaphenanthridines via anionic ring closure. / Hansen, Henriette Møller; Lysén, M.; Begtrup, M.; Kristensen, Jesper Langgaard.

    In: Tetrahedron, Vol. 61, No. 42, 17.10.2005, p. 9955-9960.

    Research output: Contribution to journalJournal articleResearchpeer-review

  86. Published

    In vivo PET imaging of cerebral 5-HT7 receptors with novel radioligands. / Hansen, Hanne D.; Herth, Matthias Manfred; Ettrup, Anders; Szabolcs, Lehel; Dyssegaard, Agnete; Kristensen, Jesper; Knudsen, Gitte M.

    In: Journal of Cerebral Blood Flow and Metabolism, Vol. 32, 08.2012, p. S126-S127.

    Research output: Contribution to journalJournal articleResearchpeer-review

  87. Published

    Labeling and preliminary in vivo evaluation of the 5-HT7 receptor selective agonist [(11)C]E-55888. / Hansen, Hanne D; Andersen, Valdemar L; Lehel, Szabolcs; Magnussen, Janus H; Dyssegaard, Agnete; Stroth, Nikolas; Kristensen, Jesper Langgaard; Knudsen, Gitte M; Herth, Matthias M.

    In: Bioorganic & Medicinal Chemistry Letters, Vol. 25, No. 9, 01.05.2015, p. 1901-4.

    Research output: Contribution to journalJournal articleResearchpeer-review

  88. Published

    Radiosynthesis and in vivo evaluation of novel radioligands for PET imaging of cerebral 5-HT7 receptors. / Hansen, Hanne D; Herth, Matthias M; Ettrup, Anders; Andersen, Valdemar L; Lehel, Szabolcs; Dyssegaard, Agnete; Kristensen, Jesper Langgaard; Knudsen, Gitte M.

    In: Journal of Nuclear Medicine, Vol. 55, No. 4, 24.02.2014, p. 640-646.

    Research output: Contribution to journalJournal articleResearchpeer-review

  89. Published

    An Improved Radiolabelling Strategy for the 5-HT2A Agonist, [C-11]Cimbi-36. / Gillings, Nic; Lehel, Szabolcs; Herth, Matthias; Leth-Petersen, Sebastian; Madsen, Jacob; Gabel-Jensen, Charlotte; Kristensen, Jesper L.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 58, 15.05.2015, p. S296-S296.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  90. Published

    Palladium-Catalyzed Arylation and Acylation of 1-Benzyloxy-1,2,3-triazole Through a Directed Ortho Lithiation-Transmetalation Strategy. / Felding, Jakob; Uhlmann, Peter; Kristensen, Jesper Langgaard; Vedsø, Per; Begtrup, Mikael.

    In: Synthesis, Vol. 8, 1998, p. 1181-1184.

    Research output: Contribution to journalJournal articleResearchpeer-review

  91. Published

    Synthesis of 4-substituted 1-(benzyloxy)pyrazoles via iodine-magnesium exchange of 1-(benzyloxy)-4-iodopyrazole. / Felding, Jakob; Kristensen, Jesper Langgaard; Bjerregaard, Trine; Sander, Lone; Vedsø, P.; Begtrup, M.

    In: Journal of Organic Chemistry, Vol. 64, No. 11, 28.05.1999, p. 4196-4198.

    Research output: Contribution to journalJournal articleResearchpeer-review

  92. Published

    Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT2A receptors, in mice. / Fantegrossi, William E; Gray, Bradley W; Bailey, Jessica M; Smith, Douglas A; Hansen, Martin; Kristensen, Jesper Langgaard.

    In: Psychopharmacology, Vol. 232, No. 6, 2015, p. 1039-47.

    Research output: Contribution to journalJournal articleResearchpeer-review

  93. Published

    Radiosynthesis and in vivo evaluation of a series of substituted 11C-phenethylamines as 5-HT2A agonist PET tracers. / Ettrup, Anders; Hansen, Martin; Santini, Martin A; Paine, James Stephen; Gillings, Nic; Palner, Mikael; Lehel, Szabolcs; Herth, Matthias Manfred; Madsen, Jacob; Kristensen, Jesper Langgaard; Begtrup, Mikael; Knudsen, Gitte Moos.

    In: European Journal of Nuclear Medicine and Molecular Imaging, Vol. 38, No. 4, 01.04.2011, p. 681-693.

    Research output: Contribution to journalJournal articleResearchpeer-review

  94. Published

    Preclinical Safety Assessment of the 5-HT(2A) Receptor Agonist PET Radioligand [ (11)C]Cimbi-36. / Ettrup, Anders; Holm, Søren; Hansen, Martin; Wasim, Muhammad; Santini, Martin Andreas; Palner, Mikael; Madsen, Jacob; Svarer, Claus; Kristensen, Jesper Langgaard; Knudsen, Gitte Moos.

    In: Molecular Imaging and Biology, Vol. 15, No. 4, 10.01.2013, p. 376-83.

    Research output: Contribution to journalJournal articleResearchpeer-review

  95. Published

    Serotonin 2A receptor agonist binding in the human brain with [C]Cimbi-36. / Ettrup, A.; da Cunha-Bang, S.; McMahon, Barry P.; Lehel, S.; Dyssegaard, A.; Skibsted, A.W.; Jørgensen, Louise Møller; Hansen, M.; Baandrup, A.O.; Bache, S.; Svarer, C.; Kristensen, Jesper Langgaard; Gillings, N.; Madsen, Jacob; Knudsen, G.M.

    In: Journal of Cerebral Blood Flow and Metabolism, Vol. 34, 30.04.2014, p. 1188-1196.

    Research output: Contribution to journalJournal articleResearchpeer-review

  96. Published

    Convergent synthesis of 3-arylated 1-hydroxypyrazoles via 3-metalated pyrazole-1-oxides. / Eskildsen, Jørgen; Kristensen, Jesper Langgaard; Vedsø, P.; Begtrup, M.; Kristensen, Jesper Langgaard.

    In: Journal of Organic Chemistry, Vol. 66, No. 25, 14.12.2001, p. 8654-8656.

    Research output: Contribution to journalJournal articleResearchpeer-review

  97. Published

    Synthesis, radiofluorination, and preliminary evaluation of the potential 5-HT2A receptor agonists [18 F]Cimbi-92 and [18 F]Cimbi-150. / Edgar, Fraser Graeme; Hansen, Hanne D; Leth-Petersen, Sebastian; Ettrup, Anders; Kristensen, Jesper L; Knudsen, Gitte M; Herth, Matthias M.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 60, No. 12, 10.2017, p. 586-591.

    Research output: Contribution to journalJournal articleResearchpeer-review

  98. Published

    Dual Nicotinic Acetylcholine Receptor α4β2 Antagonists/α7 Agonists: Synthesis, Docking Studies, and Pharmacological Evaluation of Tetrahydroisoquinolines and Tetrahydroisoquinolinium Salts. / Crestey, François; Jensen, Anders A.; Soerensen, Christian; Magnus, Charlotte Busk; Andreasen T., Jesper; Peters, Günther Herbert Johannes; Kristensen, Jesper Langgaard.

    In: Journal of Medicinal Chemistry, Vol. 61, 2018, p. 1719-1729.

    Research output: Contribution to journalJournal articleResearchpeer-review

  99. Published

    Design, synthesis and biological evaluation of Erythrina alkaloid analogues as neuronal nicotinic acetylcholine receptor antagonists. / Crestey, François; Jensen, Anders A.; Borch, Morten; Andreasen T., Jesper; Andersen, Jacob; Balle, Thomas; Kristensen, Jesper Langgaard.

    In: Journal of Medicinal Chemistry, Vol. 56, No. 23, 2013, p. 9673-9682.

    Research output: Contribution to journalJournal articleResearchpeer-review

  100. Published

    Concise synthesis of new bridged-nicotine analogues. / Crestey, François; Hooyberghs, Geert ; Kristensen, Jesper Langgaard.

    In: Tetrahedron, Vol. 68, No. 5, 04.02.2012, p. 1417-1421.

    Research output: Contribution to journalJournal articleResearchpeer-review

  101. Published

    Enantioselective Total Synthesis of (+)-Dihydro-β-erythroidine. / Clementson, Sebastian; Jessing, Mikkel; Pedersen, Henrik; Vital, Paulo; Kristensen, Jesper L.

    In: Journal of the American Chemical Society, Vol. 141, No. 22, 05.2019, p. 8783-8786.

    Research output: Contribution to journalJournal articleResearchpeer-review

  102. Published

    Nye NMDA-receptor-ligander til udforskning af hjernen. / Clausen, Rasmus Prætorius; Risgaard, Rune; Nielsen, Simon Dalsgaard; Kristensen, Jesper Langgaard; Hansen, Kasper Bø.

    In: Dansk Kemi, Vol. 91, No. 6/7, 2010, p. 21-23.

    Research output: Contribution to journalJournal articleCommunication

  103. Published

    N-Hydroxypyrazolyl glycine derivatives as selective N-methyl-D-aspartic acid receptor ligands. / Clausen, Rasmus Prætorius; Christensen, Caspar; Hansen, Kasper Bø; Greenwood, Jeremy R; Jørgensen, Lars; Micale, Nicola; Madsen, Jens Christian; Nielsen, Birgitte; Egebjerg, Jan; Bräuner-Osborne, Hans; Traynelis, Stephen F; Kristensen, Jesper Langgaard.

    In: Journal of Medicinal Chemistry, Vol. 51, No. 14, 2008, p. 4179-87.

    Research output: Contribution to journalJournal articleResearchpeer-review

  104. Published

    Ind i hjernen med nye stoffer. / Clausen, Rasmus Prætorius; Nielsen, Simon Dalsgaard; Kristensen, Jesper Langgaard; Hansen, Kasper Bø.

    In: Lægemiddelforskning, 2009, p. 34-36.

    Research output: Contribution to journalJournal articleCommunication

  105. Published

    Deprotection of 2-nitrobenzenesulfonamides using fluorous and solid phase reagents. / Christensen, C; Clausen, Rasmus Prætorius; Begtrup, M; Kristensen, Jesper Langgaard.

    In: Tetrahedron Letters, Vol. 45, No. 43, 18.10.2004, p. 7991-7993.

    Research output: Contribution to journalJournal articleResearchpeer-review

  106. Published

    Ortho lithiation-in situ borylation of substituted morpholine benzamides. / Cederbalk, Anna; Lysén, Morten; Kehler, Jan; Kristensen, Jesper L.

    In: Tetrahedron, Vol. 73, No. 12, 23.03.2017, p. 1576–1582.

    Research output: Contribution to journalJournal articleResearchpeer-review

  107. Published

    Synthesis of enantiopure 3-substituted morpholines. / Bornholdt, Jan; Felding, Jakob; Kristensen, Jesper Langgaard.

    In: Journal of Organic Chemistry, Vol. 75, No. 21, 2010, p. 7454-7457.

    Research output: Contribution to journalJournal articleResearchpeer-review

  108. Published

    Ring opening of pymisyl-protected aziridines with organocuprates. / Bornholdt, Jan; Felding, Jakob; Clausen, Rasmus Prætorius; Kristensen, Jesper Langgaard.

    In: Chemistry: A European Journal, Vol. 16, No. 41, 2010, p. 12474-12480.

    Research output: Contribution to journalJournal articleResearchpeer-review

  109. Published

    Heterocyclic pentafluorophenyl sulfonate esters as shelf stable alternatives to sulfonyl chlorides. / Bornholdt, Jan; Fjære, Karianne Wilhemsen; Felding, Jakob; Kristensen, Jesper Langgaard.

    In: Tetrahedron, Vol. 65, No. 45, 2009, p. 9280-9284.

    Research output: Contribution to journalJournal articleResearchpeer-review

  110. Published

    Palladium-mediated conversion of para-aminoarylboronic esters into para-aminoaryl- 11C-methanes. / Andersen, Valdemar Lykke; Herth, Matthias Manfred; Lehel, Szabolcs; Knudsen, Gitte Moos; Kristensen, Jesper Langgaard.

    In: Tetrahedron Letters, Vol. 54, No. 3, 2013, p. 213-216.

    Research output: Contribution to journalJournal articleResearchpeer-review

  111. Published

    Synthesis and evaluation of [C-11]CIMBI-712 and [C-11]CIMBI-772. / Andersen, Valdemar Lykke; Herth, Matthias Manfred; Hansen, Hanne Demant; Kristensen, Jesper Langgaard; Knudsen, Karen Birgitte Moos.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 56, 05.2013, p. S101-S101.

    Research output: Contribution to journalJournal articleResearchpeer-review

  112. Published

    (11)C-labeling and preliminary evaluation of pimavanserin as a 5-HT2A receptor PET-radioligand. / Andersen, Valdemar L; Hansen, Hanne D; Herth, Matthias M; Dyssegaard, Agnete; Knudsen, Gitte M; Kristensen, Jesper Langgaard.

    In: Bioorganic & Medicinal Chemistry Letters, Vol. 25, No. 5, 20.01.2015, p. 1053–1056.

    Research output: Contribution to journalJournal articleResearchpeer-review

  113. Published

    (11)C-labeling and preliminary evaluation of vortioxetine as a PET radioligand. / Andersen, Valdemar L; Hansen, Hanne D; Herth, Matthias M; Knudsen, Gitte M; Kristensen, Jesper Langgaard.

    In: Bioorganic & Medicinal Chemistry Letters, Vol. 24, No. 11, 19.04.2014, p. 2408-2411.

    Research output: Contribution to journalJournal articleResearchpeer-review

ID: 1305029