Jesper Langgaard Kristensen

Jesper Langgaard Kristensen

Professor with special responsibilities


  1. 2019
  2. E-pub ahead of print

    Enantioselective Total Synthesis of (+)-Dihydro-β-erythroidine. / Clementson, Sebastian; Jessing, Mikkel; Pedersen, Henrik; Vital, Paulo; Kristensen, Jesper L.

    In: Journal of the American Chemical Society, 28.05.2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Convenient access to F-18-labeled amines through the Staudinger reduction. / Shalgunov, Vladimir; Steen, Johanna; Denk, Christoph; Mikula, Hannes; Kjaer, Andreas; Kristensen, Jesper; Herth, Matthias.

    2019. S205-S206.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  4. Published

    Pretargeted PET imaging using a dual click F-18-labeling strategy. / Steen, Johanna; Denk, Christoph; Jorgensen, Jesper; Norregard, Kamilla; Rossin, Raffaella; Wilkovitsch, Martin; Svatunek, Dennis; Edem, Patricia; Kuntner, Claudia; Wanek, Thomas; Robillard, Marc; Kristensen, Jesper; Kjaer, Andreas; Mikula, Hannes; Herth, Matthias.

    2019. S22-S23.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  5. Published

    Trans-cyclooctene-functionalized PeptoBrushes with improved reaction kinetics of the tetrazine ligation for pretargeted nuclear imaging. / Steen, Johanna; Norregard, Kamilla; Johann, Kerstin; Jorgensen, Jesper; Svatunek, Dennis; Birke, Alexander; Edem, Patricia; Rossin, Raffaella; Seidl, Christine; Schmid, Friederike; Robillard, Marc; Mikula, Hannes; Kristensen, Jesper; Barz, Matthias; Kjaer, Andreas; Herth, Matthias.

    2019. S109-S110.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  6. Accepted/In press

    Convenient Entry to 18 F-Labeled Amines through the Staudinger Reduction. / Stéen, E. Johanna L.; Shalgunov, Vladimir; Denk, Christoph; Mikula, Hannes; Kjær, Andreas; Kristensen, Jesper L.; Herth, Matthias M.

    In: European Journal of Organic Chemistry, 01.01.2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Improved radiosynthesis and preliminary in vivo evaluation of the 11 C-labeled tetrazine [ 11 C]AE-1 for pretargeted PET imaging. / Stéen, E. Johanna L.; Jørgensen, Jesper T.; Petersen, Ida N.; Nørregaard, Kamilla; Lehel, Szabolcs; Shalgunov, Vladimir; Birke, Alexander; Edem, Patricia E.; L'Estrade, Elina T.; Hansen, Hanne D.; Villadsen, Jonas; Erlandsson, Maria; Ohlsson, Tomas; Yazdani, Abdolreza; Valliant, John F.; Kristensen, Jesper L.; Barz, Matthias; Knudsen, Gitte M.; Kjær, Andreas; Herth, Matthias M.

    In: Bioorganic and Medicinal Chemistry Letters, 01.01.2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Human biodistribution and radiation dosimetry of the 5-HT2A receptor agonist Cimbi-36 labeled with carbon-11 in two positions. / Johansen, Annette; Holm, Søren; Dall, Bente; Keller, Sune; Kristensen, Jesper L; Knudsen, Gitte M; Hansen, Hanne D.

    In: EJNMMI Research, Vol. 9, 71, 2019, p. 1-10.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. 2018
  10. Published

    Towards the Dual Click F-18-labeling of Antibodies. / Steen, Johanna; Denk, Christoph; Norregaard, Kamilla; Jorgensen, Jesper; Rossin, Raffaella; Svatunek, Dennis; Edem, Patricia; Robillard, Marc; Kjaer, Andreas; Kristensen, Jesper; Mikula, Hannes; Herth, Matthias.

    2018.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  11. Published

    The importance of small polar radiometabolites in molecular neuroimaging : A PET study with [11C]Cimbi-36 labeled in two positions. / Johansen, Annette; Hansen, Hanne D; Svarer, Claus; Lehel, Szabolcs; Leth-Petersen, Sebastian; Kristensen, Jesper L; Gillings, Nic; Knudsen, Gitte M.

    In: Journal of Cerebral Blood Flow and Metabolism, Vol. 38, No. 4, 04.2018, p. 659-668.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Dual Nicotinic Acetylcholine Receptor α4β2 Antagonists/α7 Agonists: Synthesis, Docking Studies, and Pharmacological Evaluation of Tetrahydroisoquinolines and Tetrahydroisoquinolinium Salts. / Crestey, François; Jensen, Anders A.; Soerensen, Christian; Magnus, Charlotte Busk; Andreasen T., Jesper; Peters, Günther Herbert Johannes; Kristensen, Jesper Langgaard.

    In: Journal of Medicinal Chemistry, Vol. 61, 2018, p. 1719-1729.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. 2017
  14. Published

    Synthesis, radiofluorination, and preliminary evaluation of the potential 5-HT2A receptor agonists [18 F]Cimbi-92 and [18 F]Cimbi-150. / Edgar, Fraser Graeme; Hansen, Hanne D; Leth-Petersen, Sebastian; Ettrup, Anders; Kristensen, Jesper L; Knudsen, Gitte M; Herth, Matthias M.

    In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 60, No. 12, 10.2017, p. 586-591.

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    18F-Labelling of electron rich iodonium ylides : application to the radiosynthesis of potential 5-HT2A receptor PET ligands. / Petersen, I N; Villadsen, J; Hansen, H D; Madsen, J; Jensen, A A; Gillings, N; Lehel, Szabolcs; Herth, M M; Knudsen, G M; Kristensen, J L.

    In: Organic & Biomolecular Chemistry, Vol. 15, 04.2017, p. 4351-4358.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Ortho lithiation-in situ borylation of substituted morpholine benzamides. / Cederbalk, Anna; Lysén, Morten; Kehler, Jan; Kristensen, Jesper L.

    In: Tetrahedron, Vol. 73, No. 12, 23.03.2017, p. 1576–1582.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Nucleophilic 18F-Labeling of Spirocyclic Iodonium Ylide or Boronic Pinacol Ester Precursors - Advantages and Disadvantages. / Petersen, Ida Nymann; Kristensen, Jesper Langgaard; Herth, Matthias Manfred.

    In: European Journal of Organic Chemistry, Vol. 2017, No. 3, 18.01.2017, p. 453-458.

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Development of a simple proton nuclear magnetic resonance-based procedure to estimate the approximate distribution coefficient at physiological pH (logD7.4) : Evaluation and comparison to existing practices. / Stéen, E Johanna L; Nyberg, Nils; Lehel, Szabolcs; Andersen, Valdemar L; Di Pilato, Pantaleo; Knudsen, Gitte M; Kristensen, Jesper L; Herth, Matthias M.

    In: Bioorganic & Medicinal Chemistry Letters, Vol. 27, No. 2, 15.01.2017, p. 319-322.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    A strategic approach to [6,6]-bicyclic lactones : application towards the CD fragment of DHβE. / Jepsen, Tue Heesgaard; Glibstrup, Emil; Crestey, Francois Louis Jean; Jensen, Anders A.; Kristensen, Jesper Langgaard.

    In: Beilstein Journal of Organic Chemistry, Vol. 13, 2017, p. 988-994.

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Characterization of the hepatic cytochrome P450 enzymes involved in the metabolism of 25I-NBOMe and 25I-NBOH. / Nielsen, Line Marie; Holm, Niels Bjerre; Leth-Petersen, Sebastian; Kristensen, Jesper Langgaard; Olsen, Lars; Linnet, Kristian.

    In: Drug Testing and Analysis, Vol. 9, No. 5, 2017, p. 671–679.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Detailed characterization of the in vitro pharmacological and pharmacokinetic properties of N-(2-hydroxybenzyl)-2,5-dimethoxy-4-cyanophenylethylamine (25CN-NBOH), a highly selective and brain-penetrant 5-HT2A receptor agonist. / Jensen, Anders A; McCorvy, John D; Petersen, Sebastian Leth; Bundgaard, Christoffer; Liebscher, Gudrun; Kenakin, Terry P; Bräuner-Osborne, Hans; Kehler, Jan; Kristensen, Jesper L.

    In: Journal of Pharmacology and Experimental Therapeutics, Vol. 361, No. 3, 2017, p. 441-453.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Textbook of Drug Design and Discovery : In vivo imaging in drug discovery. / Kristensen, Jesper Langgaard; Herth, Matthias Manfred.

    Textbook of Drug Design and Discovery. Fifth edition. ed. CRC Press, 2017.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  23. 2016
  24. Published

    5-HT2A/5-HT2C receptor pharmacology and intrinsic clearance of N-benzylphenethylamines modified at the primary site of metabolism. / Leth-Petersen, Sebastian; Petersen, Ida Nymann; Jensen, Anders A; Bundgaard, Christoffer; Bæk, Mathias; Kehler, Jan; Kristensen, Jesper L.

    In: A C S Chemical Neuroscience, 26.08.2016, p. 1-6.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Conformationally Constrained Peptidomimetics as Inhibitors of the Protein Arginine Methyl Transferases. / Knuhtsen, Astrid; Legrand, Baptiste; Van der Poorten, Olivier; Amblard, Muriel; Martinez, Jean; Ballet, Steven; Kristensen, Jesper L; Pedersen, Daniel Sejer.

    In: Chemistry: A European Journal, Vol. 22, No. 39, 12.08.2016, p. 14022–14028.

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Long-Acting Diclofenac Ester Prodrugs for Joint Injection : Kinetics, Mechanism of Degradation, and In Vitro Release From Prodrug Suspension. / Mertz, Nina; Larsen, Susan Weng; Kristensen, Jesper; Østergaard, Jesper; Larsen, Claus.

    In: Journal of Pharmaceutical Sciences, Vol. 105, No. 10, 27.07.2016, p. 3079–3087.

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Synthesis and characterisation of substrate-based peptides as inhibitors of histone demethylase KDM4C. / Nielsen, Simon D; Leurs, Ulrike; Bergner, Magnus; Barris, Silvia Amor; Devkota, Kanchan; Meyer, Kamilla; Iaria, Daniella; McCaughan, Jack; Lohse, Brian; Kristensen, Jesper L; Clausen, Rasmus Prætorius.

    In: Protein and Peptide Letters, Vol. 23, No. 9, 13.06.2016, p. 772 - 776.

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Computational Methods to Predict the Regioselectivity of Electrophilic Aromatic Substitution Reactions of Heteroaromatic Systems. / Kruszyk, Monika; Jessing, Mikkel; Kristensen, Jesper L; Jorgensen, Morten.

    In: Journal of Organic Chemistry, Vol. 81, No. 12, 13.05.2016, p. 5128–5134.

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published
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