Jesper Langgaard Kristensen
Professor with special responsibilities
Medicinal Chemistry Research
Jagtvej 162, 2100 København Ø, 30, Building: 342
- 2013
- Published
Design, synthesis and biological evaluation of Erythrina alkaloid analogues as neuronal nicotinic acetylcholine receptor antagonists. / Crestey, François; Jensen, Anders A.; Borch, Morten; Andreasen T., Jesper; Andersen, Jacob; Balle, Thomas; Kristensen, Jesper Langgaard.
In: Journal of Medicinal Chemistry, Vol. 56, No. 23, 2013, p. 9673-9682.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of a 11C-labeled tetrazine for rapid tetrazine–trans-cyclooctene ligation. / Herth, Matthias Manfred; Andersen, Valdemar L. ; Lehel, Szabolcs; Madsen, Jacob; Knudsen, Gitte Moos; Kristensen, Jesper Langgaard.
In: Chemical Communications, Vol. 49, 2013, p. 3805-3807.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Medicindepot dannes efter injektion i leddet. / Larsen, Susan Weng; Thing, Mette Agergaard; Østergaard, Jesper; Kristensen, Jesper Langgaard; Hansen, Martin; Larsen, Claus Selch.
In: Lægemiddelforskning, Vol. 2013, 2013, p. 38-40.Research output: Contribution to journal › Journal article › Research
- Published
Palladium-mediated conversion of para-aminoarylboronic esters into para-aminoaryl- 11C-methanes. / Andersen, Valdemar Lykke; Herth, Matthias Manfred; Lehel, Szabolcs; Knudsen, Gitte Moos; Kristensen, Jesper Langgaard.
In: Tetrahedron Letters, Vol. 54, No. 3, 2013, p. 213-216.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Radiolabelling and PET brain imaging of the a1-adrenoceptor antagonist Lu AE43936. / Risgaard, Rune; Ettrup, Anders Janusz; Balle, Thomas; Dyssegaard, Agnete; Hansen, Hanne Demant; Lehel, Szabolcs; Madsen, Jacob; Pedersen, Henrik; Püschl, Ask; Badolo, Lassina; Bang-Andersen, Benny; Knudsen, Gitte Moos; Kristensen, Jesper Langgaard.
In: Nuclear Medicine & Biology, Vol. 40, No. 1, 2013, p. 135-140.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structure-activity relationships of constrained phenylethylamine ligands for the serotonin 5-ht2 receptors. / Isberg, Vignir; Paine, James; Leth-Petersen, Sebastian; Kristensen, Jesper Langgaard; Gloriam, David E.
In: P L o S One, Vol. 8, No. 11, e78515, 2013.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and biological evaluation of 4-(aminomethyl)-1-hydroxypyrazole analogues of muscimol as ¿-aminobutyric acidA receptor agonists. / Petersen, Jette Gellert; Bergmann, Rikke; Møller, Henriette A.; Jørgensen, Charlotte Grube; Nielsen, Birgitte; Kehler, Jan; Frydenvang, Karla ; Kristensen, Jesper; Balle, Thomas; Jensen, Anders A.; Kristiansen, Uffe; Frølund, Bente.
In: Journal of Medicinal Chemistry, Vol. 56, No. 3, 2013, p. 993-1006.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and stability study of a new major metabolite of gamma-hydroxybutyric acid. / Petersen, Ida Nymann; Kristensen, Jesper Langgaard; Tortzen, Christian; Breindahl, Torben; Pedersen, Daniel Sejer.
In: Beilstein Journal of Organic Chemistry, Vol. 9, 2013, p. 641-646.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Preclinical Safety Assessment of the 5-HT(2A) Receptor Agonist PET Radioligand [ (11)C]Cimbi-36. / Ettrup, Anders; Holm, Søren; Hansen, Martin; Wasim, Muhammad; Santini, Martin Andreas; Palner, Mikael; Madsen, Jacob; Svarer, Claus; Kristensen, Jesper Langgaard; Knudsen, Gitte Moos.
In: Molecular Imaging and Biology, Vol. 15, No. 4, 10.01.2013, p. 376-83.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of C-11-labeled oxindole derivatives for in vivo PET imaging of the 5-HT7 receptor. / Herth, Matthias Manfred; Hansen, Hanne; Andersen, Valdemar L.; Volk, Balazs; Ettrup, Anders; Antoni, Ferenc; Lehel, Szabolcs; Dyssegaard, Agnete; Kristensen, Jesper L.; Knudsen, Gitte M.
2013. S82-S82.Research output: Contribution to conference › Conference abstract for conference › Research
- Published
Synthesis and evaluation of [C-11]CIMBI-712 and [C-11]CIMBI-772. / Andersen, Valdemar Lykke; Herth, Matthias Manfred; Hansen, Hanne Demant; Kristensen, Jesper Langgaard; Knudsen, Karen Birgitte Moos.
2013. S101-S101.Research output: Contribution to conference › Conference abstract for conference › Research
- Published
PRODRUGS OF NON- STEROID ANTI - INFLAMMATORY AGENTS (NSAIDS). / Larsen, Claus Selch (Inventor); Larsen, Susan Weng (Inventor); Thing, Mette Agergaard (Inventor); Kristensen, Jesper Langgaard (Inventor); JENSEN, HENRIK (Inventor); OESTERGAARD, JESPER (Inventor).
IPC No.: C07D 487/ 04 A I. Patent No.: WO2013064153.Research output: Patent
- Published
Identification of a new metabolite of GHB : gamma-hydroxybutyric acid glucuronide. / Petersen, Ida Nymann; Tortzen, Christian; Kristensen, Jesper Langgaard; Pedersen, Daniel Sejer; Breindahl, Torben.
In: Journal of Analytical Toxicology, Vol. 37, No. 5, 06.2013, p. 291-7.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Posttranslational Modifications of the Histone 3 Tail and Their Impact on the Activity of Histone Lysine Demethylases In Vitro. / Lohse, Brian; Helgstrand, Charlotte; Andersson, Jan Legaard; Leurs, Ulrike; Cloos, Paul Andreas Compare; Kristensen, Jesper Langgaard; Clausen, Rasmus Prætorius.
In: P L o S One, Vol. 8, No. 7, 02.07.2013, p. e67653.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1305029
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A strategic approach to [6,6]-bicyclic lactones: application towards the CD fragment of DHβE
Research output: Contribution to journal › Journal article › Research › peer-review
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103
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Structure-activity relationships of constrained phenylethylamine ligands for the serotonin 5-ht2 receptors
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
79
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Substrate- and Cofactor-independent Inhibition of Histone Demethylase KDM4C
Research output: Contribution to journal › Journal article › Research › peer-review
Published