Jesper Langgaard Kristensen
Professor with special responsibilities
Medicinal Chemistry Research
Jagtvej 162, 2100 København Ø, 30, Building: 342
- 2017
- Published
Synthesis, radiofluorination, and preliminary evaluation of the potential 5-HT2A receptor agonists [18 F]Cimbi-92 and [18 F]Cimbi-150. / Edgar, Fraser Graeme; Hansen, Hanne D; Leth-Petersen, Sebastian; Ettrup, Anders; Kristensen, Jesper L; Knudsen, Gitte M; Herth, Matthias M.
In: Journal of Labelled Compounds and Radiopharmaceuticals, Vol. 60, No. 12, 10.2017, p. 586-591.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
18F-Labelling of electron rich iodonium ylides : application to the radiosynthesis of potential 5-HT2A receptor PET ligands. / Petersen, I N; Villadsen, J; Hansen, H D; Madsen, J; Jensen, A A; Gillings, N; Lehel, Szabolcs; Herth, M M; Knudsen, G M; Kristensen, J L.
In: Organic & Biomolecular Chemistry, Vol. 15, 04.2017, p. 4351-4358.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Ortho lithiation-in situ borylation of substituted morpholine benzamides. / Cederbalk, Anna; Lysén, Morten; Kehler, Jan; Kristensen, Jesper L.
In: Tetrahedron, Vol. 73, No. 12, 23.03.2017, p. 1576–1582.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Nucleophilic 18F-Labeling of Spirocyclic Iodonium Ylide or Boronic Pinacol Ester Precursors - Advantages and Disadvantages. / Petersen, Ida Nymann; Kristensen, Jesper Langgaard; Herth, Matthias Manfred.
In: European Journal of Organic Chemistry, Vol. 2017, No. 3, 18.01.2017, p. 453-458.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of a simple proton nuclear magnetic resonance-based procedure to estimate the approximate distribution coefficient at physiological pH (logD7.4) : Evaluation and comparison to existing practices. / Stéen, E Johanna L; Nyberg, Nils; Lehel, Szabolcs; Andersen, Valdemar L; Di Pilato, Pantaleo; Knudsen, Gitte M; Kristensen, Jesper L; Herth, Matthias M.
In: Bioorganic & Medicinal Chemistry Letters, Vol. 27, No. 2, 15.01.2017, p. 319-322.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A strategic approach to [6,6]-bicyclic lactones : application towards the CD fragment of DHβE. / Jepsen, Tue Heesgaard; Glibstrup, Emil; Crestey, Francois Louis Jean; Jensen, Anders A.; Kristensen, Jesper Langgaard.
In: Beilstein Journal of Organic Chemistry, Vol. 13, 2017, p. 988-994.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Characterization of the hepatic cytochrome P450 enzymes involved in the metabolism of 25I-NBOMe and 25I-NBOH. / Nielsen, Line Marie; Holm, Niels Bjerre; Leth-Petersen, Sebastian; Kristensen, Jesper Langgaard; Olsen, Lars; Linnet, Kristian.
In: Drug Testing and Analysis, Vol. 9, No. 5, 2017, p. 671–679.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Detailed characterization of the in vitro pharmacological and pharmacokinetic properties of N-(2-hydroxybenzyl)-2,5-dimethoxy-4-cyanophenylethylamine (25CN-NBOH), a highly selective and brain-penetrant 5-HT2A receptor agonist. / Jensen, Anders A; McCorvy, John D; Petersen, Sebastian Leth; Bundgaard, Christoffer; Liebscher, Gudrun; Kenakin, Terry P; Bräuner-Osborne, Hans; Kehler, Jan; Kristensen, Jesper L.
In: Journal of Pharmacology and Experimental Therapeutics, Vol. 361, No. 3, 2017, p. 441-453.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Textbook of Drug Design and Discovery : In vivo imaging in drug discovery. / Kristensen, Jesper Langgaard; Herth, Matthias Manfred.
Textbook of Drug Design and Discovery. Fifth edition. ed. CRC Press, 2017.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research
ID: 1305029
Most downloads
-
123
downloads
A strategic approach to [6,6]-bicyclic lactones: application towards the CD fragment of DHβE
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
103
downloads
Structure-activity relationships of constrained phenylethylamine ligands for the serotonin 5-ht2 receptors
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
79
downloads
Substrate- and Cofactor-independent Inhibition of Histone Demethylase KDM4C
Research output: Contribution to journal › Journal article › Research › peer-review
Published