Kristian Strømgaard
Professor
Medicinal Chemistry Research
Jagtvej 162, 2100 København Ø, 30, Building: 240
- Published
Design and synthesis of peptide YY analogues with c-terminal backbone amide-to-ester modifications. / Albertsen, Louise; Andersen, J.J.; Paulsson, J.F.; Thomsen, J.K.; Norrild, Jens Chr.; Strømgaard, K.
In: A C S Medicinal Chemistry Letters, Vol. 4, No. 12, 12.12.2013, p. 1228-1232.Research output: Contribution to journal › Journal article › Research › peer-review
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A parallel semisynthetic approach for structure-activity relationship studies of peptide YY. / Albertsen, Louise; Østergaard, Søren; Paulsson, Johan F; Norrild, Jens Chr.; Strømgaard, Kristian.
In: ChemMedChem, Vol. 8, No. 9, 09.2013, p. 1505-13.Research output: Contribution to journal › Journal article › Research › peer-review
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Recombinant production of peptide C-terminal α-amides using an engineered intein. / Albertsen, Louise; Shaw, Allan C; Norrild, Jens Chr.; Strømgaard, Kristian.
In: Bioconjugate Chemistry, Vol. 24, No. 11, 20.11.2013, p. 1883-94.Research output: Contribution to journal › Journal article › Research › peer-review
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Mutational mapping and modeling of the binding site for (S)-citalopram in the human serotonin transporter. / Andersen, Jacob; Olsen, Lars; Hansen, Kasper Bø; Taboureau, Olivier; Jørgensen, Flemming Steen; Jørgensen, Anne Marie; Bang-Andersen, Benny; Egebjerg, Jan; Strømgaard, Kristian; Kristensen, Anders Skov.
In: Journal of Biological Chemistry, Vol. 285, No. 3, 2010, p. 2051-2063.Research output: Contribution to journal › Journal article › Research › peer-review
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Molecular basis for selective serotonin reuptake inhibition by the antidepressant agent fluoxetine (prozac). / Andersen, Jacob; Stuhr-Hansen, Nicolai; Zachariassen, Linda Grønborg; Koldsø, Heidi; Schiøtt, Birgit; Strømgaard, Kristian; Kristensen, Anders S.
In: Molecular Pharmacology, Vol. 85, No. 5, 05.2014, p. 703-14.Research output: Contribution to journal › Journal article › Research › peer-review
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Antidepressive lægemidler : nu i 3D. / Andersen, Jacob; Sørensen, Lena; Strømgaard, Kristian; Kristensen, Anders Skov.
In: Lægemiddelforskning, Vol. 2010, 12.2010, p. 25-27.Research output: Contribution to journal › Journal article › Communication
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Binding site residues control inhibitor selectivity in the human norepinephrine transporter but not in the human dopamine transporter. / Andersen, Jacob; Ringsted, Kristoffer B; Bang-Andersen, Benny; Strømgaard, Kristian; Kristensen, Anders S.
In: Scientific Reports, Vol. 5, 15650, 2015, p. 1-12.Research output: Contribution to journal › Journal article › Research › peer-review
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Location of the antidepressant binding site in the serotonin transporter : importance of SER-438 in recognition of citalopram and tricyclic antidepressants. / Andersen, Jacob; Taboureau, Olivier; Hansen, Kasper Bø; Olsen, Lars; Egebjerg, Jan; Strømgaard, Kristian; Kristensen, Anders Skov.
In: Journal of Biological Chemistry, Vol. 284, No. 15, 2009, p. 10276-10284.Research output: Contribution to journal › Journal article › Research › peer-review
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Molecular determinants for selective recognition of antidepressants in the human serotonin and norepinephrine transporters. / Andersen, Jacob; Stuhr-Hansen, Nicolai; Zachariassen, Linda; Toubro, Søren; Hansen, Stinna Maria R; Eildal, Jonas Nii Nortey; Bond, Andrew D; Bøgesø, Klaus P; Bang-Andersen, Benny; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Proceedings of the National Academy of Sciences of the United States of America, Vol. 108, No. 29, 19.07.2011, p. 12137-12142.Research output: Contribution to journal › Journal article › Research › peer-review
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Recent advances in the understanding of the interaction of antidepressant drugs with serotonin and norepinephrine transporters. / Andersen, Jacob; Kristensen, Anders Skov; Bang-Andersen, Benny; Strømgaard, Kristian.
In: Chemical Communications, No. 25, 2009, p. 3677-3692.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1302559
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PDZ domain-mediated interactions of G protein-coupled receptors with postsynaptic density protein 95: quantitative characterization of interactions
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