Kristian Strømgaard
Professor
Medicinal Chemistry Research
Jagtvej 162, 2100 København Ø, 30, Building: 240
- Published
Uncompetitive antagonism of AMPA receptors : Mechanistic insights from studies of polyamine toxin derivatives. / Andersen, Trine F; Tikhonov, Denis B; Bølcho, Ulrik; Bolshakov, Konstantin; Nelson, Jared K; Pluteanu, Florentina; Mellor, Ian R; Egebjerg, Jan; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 49, No. 18, 07.09.2006, p. 5414-5423.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist. / Andersen, Trine F; Vogensen, Stine B; Jensen, Lars S; Knapp, Kolja M; Strømgaard, Kristian.
In: Bioorganic & Medicinal Chemistry, Vol. 13, No. 17, 01.09.2005, p. 5104-5112.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Contrasting actions of philanthotoxin-343 and philanthotoxin-(12) on human muscle nicotinic acetylcholine receptors. / Brier, Tim J; Mellor, Ian R; Tikhonov, Denis B; Neagoe, Ioana; Shao, Zuoyi; Brierley, Matt J; Strømgaard, Kristian; Jaroszewski, Jerzy W; Krogsgaard-Larsen, Povl; Usherwood, Peter N R.
In: Molecular Pharmacology, Vol. 64, No. 4, 10.2003, p. 954-964.Research output: Contribution to journal › Journal article › Research › peer-review
Terpene trilactones from Ginkgo biloba are antagonists of cortical glycine and GABA(A) receptors. / Ivic, Lidija; Sands, Tristan T J; Fishkin, Nathan; Nakanishi, Koji; Kriegstein, Arnold R; Strømgaard, Kristian.
In: Journal of Biological Chemistry, Vol. 278, No. 49, 05.12.2003, p. 49279-49285.Research output: Contribution to journal › Journal article › Research › peer-review
Ginkgolides : selective acetylations, translactonization, and biological evaluation. / Jaracz, Stanislav; Strømgaard, Kristian; Nakanishi, Koji.
In: Journal of Organic Chemistry, Vol. 67, No. 13, 28.06.2002, p. 4623-4626.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Ginkgolides and glycine receptors : a structure-activity relationship study. / Jaracz, Stanislav; Nakanishi, Koji; Jensen, Anders A.; Strømgaard, Kristian.
In: Chemistry: A European Journal, Vol. 10, No. 6, 2004, p. 1507-18.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Stoffer fra Tempeltæet (Ginkgo biloba) som redskaber for studier af hjernens funktion. / Jensen, Anders A.; Strømgaard, Kristian.
In: Dansk Kemi 83, Vol. 87, No. 1, 2006, p. 16-18.Research output: Contribution to journal › Journal article › Communication
- Published
Probing the pharmacophore of ginkgolides as glycine receptor antagonists. / Jensen, Anders Asbjørn; Begum, Nasreen; Vogensen, Stine Byskov; Knapp, Kolja Michael; Gundertofte, Klaus; Dzyuba, Sergei V.; Ishii, Hideki; Nakanishi, Koji; Kristiansen, Uffe; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 50, No. 7, 2007, p. 1610-1617.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design, synthesis, and pharmacological characterization of polyamine toxin derivatives : potent ligands for the pore-forming region of AMPA receptors. / Jensen, Lars S; Bølcho, Ulrik; Egebjerg, Jan; Strømgaard, Kristian.
In: ChemMedChem, Vol. 1, No. 4, 04.2006, p. 419-428.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Expressed protein ligation of ionotropic glutamate receptors. / Jensen, Mette Stougård; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Biopolymers, Vol. 88, No. 4, 2007, p. 602.Research output: Contribution to journal › Conference abstract in journal › Research
- Published
Solid-phase synthesis of polyamine toxin analogues : potent and selective antagonists of Ca2+-permeable AMPA receptors. / Kromann, Hasse; Krikstolaityte, Sonata; Andersen, Anne J; Andersen, Kim; Krogsgaard-Larsen, Povl; Jaroszewski, Jerzy W; Egebjerg, Jan; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 45, No. 26, 19.12.2002, p. 5745-5754.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Modification of the philanthotoxin-343 polyamine moiety results in different structure-activity profiles at muscle nicotinic ACh, NMDA and AMPA receptors. / Mellor, I R; Brier, T J; Pluteanu, F; Strømgaard, K; Saghyan, A; Eldursi, N; Brierley, M J; Andersen, K; Jaroszewski, J W; Krogsgaard-Larsen, P; Usherwood, P N R.
In: Neuropharmacology, Vol. 44, No. 1, 01.2003, p. 70-80.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Unaturlige aminosyrer skaber ny viden om proteiner. / Rannes, Julie; Andersen, Jacob; Jensen, Anders A.; Christensen, Leif; Strømgaard, Kristian.
In: Lægemiddelforskning, 2006, p. 28-29.Research output: Contribution to journal › Journal article › Communication
- Published
Site-specific incorporation of unnatural amino acids into proteins. / Strømgaard, Anne; Jensen, Anders A.; Strømgaard, Kristian.
In: ChemBioChem, Vol. 5, No. 7, 2004, p. 909-16.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Protolytic properties of polyamine wasp toxin analogues studied by 13C NMR spectroscopy. / Strømgaard, Kristian; Piazzi, Lorna; Olsen, Christian A; Franzyk, Henrik; Jaroszewski, Jerzy W.
In: Magnetic Resonance in Chemistry, Vol. 44, No. 11, 2006, p. 1013-22.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Solid-phase synthesis and pharmacological evaluation of analogues of PhTX-12-A potent and selective nicotinic acetylcholine receptor antagonist. / Strømgaard, Kristian; Mellor, Ian R; Andersen, Kim; Neagoe, Ioana; Pluteanu, Florentina; Usherwood, Peter N R; Krogsgaard-Larsen, Povl; Jaroszewski, Jerzy W.
In: Bioorganic & Medicinal Chemistry Letters, Vol. 12, No. 8, 22.04.2002, p. 1159-1162.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
AMPA receptor ligands : synthetic and pharmacological studies of polyamines and polyamine toxins. / Strømgaard, Kristian; Mellor, Ian.
In: Medicinal Research Reviews, Vol. 24, No. 5, 09.2004, p. 589-620.Research output: Contribution to journal › Journal article › Research › peer-review
Ginkgolide derivatives for photolabeling studies : preparation and pharmacological evaluation. / Strømgaard, Kristian; Saito, D Roland; Shindou, Hideo; Ishii, Satoshi; Shimizu, Takao; Nakanishi, Koji.
In: Journal of Medicinal Chemistry, Vol. 45, No. 18, 29.08.2002, p. 4038-4046.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Polyamine toxins : development of selective ligands for ionotropic receptors. / Strømgaard, Kristian; Jensen, Lars S; Vogensen, Stine B.
In: Toxicon, Vol. 45, No. 3, 01.03.2005, p. 249-254.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Chemistry and biology of terpene trilactones from Ginkgo biloba. / Strømgaard, Kristian; Nakanishi, Koji.
In: Angewandte Chemie International Edition, Vol. 43, No. 13, 19.03.2004, p. 1640-1658.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Preparation of a tritiated ginkgolide. / Strømgaard, Kristian; Suehiro, Makiko; Nakanishi, Koji.
In: Bioorganic & Medicinal Chemistry Letters, Vol. 14, No. 22, 15.11.2004, p. 5673-5675.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of polyamines and polyamine toxins. An improved alkylation procedure. / Strømgaard, Kristian; Andersen, TF.
In: Tetrahedron Letters, Vol. 45, 2004, p. 7929-7933.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Natural products as tools for studies of ligand-gated ion channels. / Strømgaard, Kristian.
In: Chemical Record, Vol. 5, No. 4, 2005, p. 229-239.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Preparation of 7-substituted ginkgolide derivatives : potent platelet activating factor (PAF) receptor antagonists. / Vogensen, Stine Byskov; Strømgaard, Kristian; Shindou, Hideo; Jaracz, Stanislav; Suehiro, Makiko; Ishii, Satoshi; Shimizu, Takao; Nakanishi, Koji.
In: Journal of Medicinal Chemistry, Vol. 46, No. 4, 13.02.2003, p. 601-608.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1302559
Most downloads
-
2910
downloads
PDZ domain-mediated interactions of G protein-coupled receptors with postsynaptic density protein 95: quantitative characterization of interactions
Research output: Contribution to journal › Journal article › Research › peer-review
Published