Kristian Strømgaard
Professor
Medicinal Chemistry Research
Jagtvej 162, 2100 København Ø, 30, Building: 240
- 2012
- Published
General synthesis of β-alanine-containing spider polyamine toxins and discovery of nephila polyamine toxins 1 and 8 as highly potent inhibitors of ionotropic glutamate receptors. / Lucas, Simon; Poulsen, Mette H; Nørager, Niels G; Barslund, Anne F; Bach, Tinna B; Kristensen, Anders S; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 55, No. 22, 26.11.2012, p. 10297-10301.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
An expanded view of the protein folding landscape of PDZ domains. / Hultqvist, Greta; Pedersen, Søren W; Chi, Celestine N.; Strømgaard, Kristian; Gianni, Stefano; Jemth, Per.
In: Biochemical and Biophysical Research Communications, Vol. 421, No. 3, 11.05.2012, p. 550-553.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A heteromeric snake toxin and the molecular details of pain perception. / Strømgaard, Kristian; Kristensen, Anders Skov.
In: Angewandte Chemie International Edition, Vol. 51, No. 17, 23.04.2012, p. 4009-4011.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A high-affinity, dimeric inhibitor of PSD-95 bivalently interacts with PDZ1-2 and protects against ischemic brain damage. / Bach, Anders*; Clausen, Bettina H; Møller, Magda; Vestergaard, Bente; Chi, Celestine N; Round, Adam; Sørensen, Pernille Louise; Nissen, Klaus Bertram; Kastrup, Jette Sandholm; Gajhede, Michael; Jemth, Per; Kristensen, Anders Skov; Lundström, Patrik; Lambertsen, Kate Lykke; Strømgaard, Kristian* (*Corresponding).
In: Proceedings of the National Academy of Sciences of the United States of America, Vol. 109, No. 9, 28.02.2012, p. 3317-3322.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Side-chain interactions form late and cooperatively in the binding reaction between disordered peptides and PDZ domains. / Haq, S Raza; Chi, Celestine N; Bach, Anders; Dogan, Jakob; Engström, Åke; Hultqvist, Greta; Karlsson, O. Andreas; Lundström, Patrik; Montemiglio, Linda Celeste; Strømgaard, Kristian; Gianni, Stefano; Jemth, Per.
In: Journal of the American Chemical Society, Vol. 134, No. 1, 01.2012, p. 599-605.Research output: Contribution to journal › Journal article › Research › peer-review
- Submitted
High-affinity, dimeric inhibitors of PSD-95 as efficient neuroprotectants against ischemic brain damage and for treatment of pain. / Bach, Anders (Inventor); Strømgaard, Kristian (Inventor).
Patent No.: WO2012/156308 (Granted: EP2707014B1; US9139615B2).Research output: Patent
- Published
Interaction of antidepressants with the serotonin and norepinephrine transporters : mutational studies of the S1 substrate binding pocket. / Sørensen, Lena; Andersen, Jacob; Thomsen, Mette; Hansen, Stinna M.R.; Zhao, Xiaobei; Sandelin, Albin Gustav; Strømgaard, Kristian; Kristensen, Anders S.
In: The Journal of Biological Chemistry, Vol. 287, No. 52, 2012, p. 43694-43707.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Interaction of antidepressants with the serotonin and norepinephrine transporters : mutational studies of the S1 substrate binding pocket. / Sørensen, Lena; Andersen, Jacob; Thomsen, Mette; Hansen, Stinna M.R.; Zhao, Xiaobei; Sandelin, Albin Gustav; Strømgaard, Kristian; Kristensen, Anders Skov.
In: Journal of Biological Chemistry, Vol. 287, 2012, p. 43694-43707.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Ligand binding by PDZ domains. / Chi, Celestine N.; Bach, Anders; Strømgaard, Kristian; Gianni, Stefano; Jemth, Per.
In: BioFactors, Vol. 38, No. 5, 2012, p. 338-348 (Review).Research output: Contribution to journal › Journal article › Research › peer-review
- 2011
- Published
Small molecules from spiders used as chemical probes. / Olsen, Christian Adam; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Angewandte Chemie International Edition, Vol. 50, No. 48, 25.11.2011, p. 11296-11311.Research output: Contribution to journal › Review › Research › peer-review
- Published
SLC6 Neurotransmitter Transporters: Structure, Function, and Regulation. / Kristensen, Anders S; Andersen, Jacob; Jørgensen, Trine N; Sørensen, Lena; Eriksen, Jacob; Løland, Claus Juul; Strømgaard, Kristian; Gether, Ulrik.
In: Pharmacological Reviews, Vol. 63, No. 3, 01.09.2011, p. 585-640.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A fluorescence polarization based screening assay for identification of small molecule inhibitors of the PICK1 PDZ domain. / Thorsen, Thor S; Madsen, Kenneth L; Dyhring, Tino; Bach, Anders; Peters, Dan; Strømgaard, Kristian; Rønn, Lars Christian B; Gether, Ulrik.
In: Combinatorial Chemistry & High Throughput Screening, Vol. 14, No. 7, 01.08.2011, p. 590-600.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Molecular determinants for selective recognition of antidepressants in the human serotonin and norepinephrine transporters. / Andersen, Jacob; Stuhr-Hansen, Nicolai; Zachariassen, Linda; Toubro, Søren; Hansen, Stinna Maria R; Eildal, Jonas Nii Nortey; Bond, Andrew D; Bøgesø, Klaus P; Bang-Andersen, Benny; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Proceedings of the National Academy of Sciences of the United States of America, Vol. 108, No. 29, 19.07.2011, p. 12137-12142.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Cell-permeable and plasma-stable peptidomimetic inhibitors of the postsynaptic density-95/N-methyl-D-aspartate receptor interaction. / Bach, Anders*; Eildal, Jonas Nii Nortey*; Stuhr-Hansen, Nicolai; Deeskamp, Rasmus; Gottschalk, Marie; Pedersen, Søren Wittrup; Kristensen, Anders Skov; Strømgaard, Kristian (*Shared 1st authors).
In: Journal of Medicinal Chemistry, Vol. 54, No. 5, 10.03.2011, p. 1333-1346.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Expedient synthesis of 1,3-substituted benzene peptidomimetics. / Bach, Anders; Strømgaard, Kristian.
In: Synthesis, Vol. 2011, No. 5, 08.02.2011, p. 807-815.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Biophysical characterization of the complex between human papillomavirus E6 protein and synapse-associated protein 97. / Chi, Celestine Ngang; Bach, Anders; Engström, Åke; Strømgaard, Kristian; Lundström, Patrik; Ferguson, Neil; Jemth, Per.
In: Journal of Biological Chemistry, Vol. 286, No. 5, 04.02.2011, p. 3597-3606.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Improving the stability of alpha-conotoxin AuIB through N-to-C cyclization : The effect of linker length on stability and activity at nicotinic acetylcholine receptors. / Armishaw, Christopher J; Jensen, Anders A; Balle, Lena D; Scott, Krystle C M; Sørensen, Lena; Strømgaard, Kristian.
In: Antioxidants & Redox Signaling, Vol. 14, No. 1, 2011, p. 65-76.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Solid-phase synthesis and biological evaluation of Joro spider toxin-4 from Nephila clavata. / Barslund, Anne Fuglsang; Poulsen, Mette Homann; Bach, Tinna Brøbech; Lucas, Simon; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Journal of Natural Products, Vol. 74, No. 3, 2011, p. 483-486.Research output: Contribution to journal › Journal article › Research › peer-review
- 2010
- Published
Antidepressive lægemidler : nu i 3D. / Andersen, Jacob; Sørensen, Lena; Strømgaard, Kristian; Kristensen, Anders Skov.
In: Lægemiddelforskning, Vol. 2010, 12.2010, p. 25-27.Research output: Contribution to journal › Journal article › Communication
- Published
Modified peptides as potent inhibitors of the PSD-95/NMDA receptor interaction. / Bach, Anders (Inventor); Strømgaard, Kristian (Inventor).
Patent No.: WO2010/004003 (Granted: EP2320927B1; US9241967B2).Research output: Patent
- Published
Assessment of structurally diverse philanthotoxin analogues for inhibitory activity on ionotropic glutamate receptor subtypes : Discovery of nanomolar, nonselective, and use-dependent antagonists. / Frølund, Sidsel; Bella, Angelo; Kristensen, Anders Skov; Ziegler, Hanne Lindvig; Witt, Matthias; Olsen, Christian Adam; Strømgaard, Kristian; Franzyk, Henrik; Jaroszewski, Jerzy W.
In: Journal of Medicinal Chemistry, Vol. 53, No. 20, 2010, p. 7441-7451.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Chemical biology. / Strømgaard, Kristian.
Textbook of drug design and discovery. ed. / Povl Krogsgaard-Larsen; Kristian Strømgaard; Ulf Madsen. 4. ed. Boca Raton : CRC Press, 2010. p. 59-74.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Education
- Published
Deciphering the kinetic binding mechanism of dimeric ligands using a potent plasma-stable dimeric inhibitor of postsynaptic density protein-95 as an example. / Chi, Celestine N; Bach, Anders; Gottschalk, Marie; Kristensen, Anders Skov; Strømgaard, Kristian; Jemth, Per.
In: Journal of Biological Chemistry, Vol. 285, No. 36, 2010, p. 28252-28260.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Identification of a small-molecule inhibitor of the PICK1 PDZ domain that inhibits hippocampal LTP and LTD. / Thorsen, Thor S; Madsen, Kenneth L; Rebola, Nelson; Rathje, Mette; Anggono, Victor; Bach, Anders; Moreira, Irina S; Stuhr-Hansen, Nicolai; Dyhring, Tino; Peters, Dan; Beuming, Thijs; Huganir, Richard; Weinstein, Harel; Mulle, Christophe; Strømgaard, Kristian; Rønn, Lars Christian B; Gether, Ulrik.
In: Proceedings of the National Academy of Science of the United States of America, Vol. 107, No. 1, 2010, p. 413-8.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Mutational mapping and modeling of the binding site for (S)-citalopram in the human serotonin transporter. / Andersen, Jacob; Olsen, Lars; Hansen, Kasper Bø; Taboureau, Olivier; Jørgensen, Flemming Steen; Jørgensen, Anne Marie; Bang-Andersen, Benny; Egebjerg, Jan; Strømgaard, Kristian; Kristensen, Anders Skov.
In: Journal of Biological Chemistry, Vol. 285, No. 3, 2010, p. 2051-2063.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structure and absolute configuration of ginkgolide B characterized by IR- and VCD spectroscopy. / Andersen, Niels Højmark; Christensen, Niels Johan; Lassen, Peter Rygaard; Freedman, Teresa B.N.; Nafie, Laurence A.; Strømgaard, Kristian; Hemmingsen, Lars Bo Stegeager.
In: Chirality, Vol. 22, No. 2, 2010, p. 217-223.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structure-activity relationships of a small-molecule inhibitor of the PDZ domain of PICK1. / Bach, Anders; Stuhr-Hansen, Nicolai; Thorsen, Thor S; Bork, Nicolai; Moreira, Irina S; Frydenvang, Karla; Padrah, Shahrokh; Christensen, S Brøgger; Madsen, Kenneth L; Weinstein, Harel; Gether, Ulrik; Strømgaard, Kristian.
In: Organic & Biomolecular Chemistry, Vol. 8, No. 19, 2010, p. 4281-4288.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Textbook of drug design and discovery. / Krogsgaard-Larsen, Povl; Strømgaard, Kristian; Madsen, Ulf.
4 ed. Boca Raton : CRC Press, 2010. 460 p.Research output: Book/Report › Book
- 2009
- Published
A sequential binding mechanism in a PDZ domain. / Chi, Celestine N; Bach, Anders; Engström, Åke; Wang, Huiqun; Strømgaard, Kristian; Gianni, Stefano; Jemth, Per.
In: Biochemistry, Vol. 48, No. 30, 2009, p. 7089-7097.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design and synthesis of highly potent and plasma-stable dimeric inhibitors of the PSD-95-NMDA receptor interaction. / Bach, Anders; Chi, Celestine N; Pang, Gar Fai; Olsen, Lars; Kristensen, Anders Skov; Jemth, Per; Strømgaard, Kristian.
In: Angewandte Chemie - International Edition, Vol. 48, No. 51, 2009, p. 9685-9689.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Detecting protein-protein interactions in living cells : development of a bioluminescence resonance energy transfer assay to evaluate the PSD-95/NMDA receptor interaction. / Gottschalk, Marie; Bach, Anders; Hansen, Jakob Lerche; Krogsgaard-Larsen, Povl; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Neurochemical Research, Vol. 34, No. 10, 2009, p. 1729-1737.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Location of the antidepressant binding site in the serotonin transporter : importance of SER-438 in recognition of citalopram and tricyclic antidepressants. / Andersen, Jacob; Taboureau, Olivier; Hansen, Kasper Bø; Olsen, Lars; Egebjerg, Jan; Strømgaard, Kristian; Kristensen, Anders Skov.
In: Journal of Biological Chemistry, Vol. 284, No. 15, 2009, p. 10276-10284.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Rational design of a-conotoxin analogues targeting a7 nicotinic acetylcholine receptors : Improved antagonistic activity by incorporation of proline derivatives. / Armishaw, Christopher; Jensen, Anders Asbjørn; Balle, Thomas; Clark, Richard J; Harpsøe, Kasper; Skonberg, Christian; Liljefors, Tommy; Strømgaard, Kristian.
In: Journal of Biological Chemistry, Vol. 284, No. 14, 2009, p. 9498-9512.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Recent advances in the understanding of the interaction of antidepressant drugs with serotonin and norepinephrine transporters. / Andersen, Jacob; Kristensen, Anders Skov; Bang-Andersen, Benny; Strømgaard, Kristian.
In: Chemical Communications, No. 25, 2009, p. 3677-3692.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Skræddersyede proteiner : uden naturens begrænsninger. / Strømgaard, Kristian; Jensen, Mette Stougård; Kristensen, Anders Skov.
In: Lægemiddelforskning, 2009, p. 10-12.Research output: Contribution to journal › Journal article › Communication
- Published
Synthesis and biological activity of argiotoxin 636 and analogues : selective antagonists for ionotropic glutamate receptors. / Nelson, Jared Keith; Frølund, Sidsel Ullerup; Tikhonov, Dennis B; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Angewandte Chemie - International Edition, Vol. 48, No. 17, 2009, p. 3087-3091.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and biological activity of novel a-conotoxin analogues incorporating substituted proline derivatives. / Armishaw, Christopher; Jensen, Anders Asbjørn; Skonberg, Christian; Liljefors, Tommy; Strømgaard, Kristian.
Peptides for youth: The proceedings of the 20th American peptide symposium. ed. / Susan Del Valle; Emanuel Escher; William D Lubell. Vol. 611 Springer, 2009. p. 179-180 (Advances in Experimental Medicine and Biology, Vol. 611).Research output: Chapter in Book/Report/Conference proceeding › Article in proceedings › Research › peer-review
- 2008
- Published
Electrophysiological characterization of analogues of philanthotoxin-343 on ionotropic glutamate receptors. / Frølund, Sidsel Ullerup; Ziegler, Hanne Lindvig; Franzyk, Henrik; Strømgaard, Kristian; Kristensen, Anders Skov; Jaroszewski, Jerzy Witold.
2008. Poster session presented at Fællesmøde for de danske farmakologiske selskaber 2008, Odense, Denmark.Research output: Contribution to conference › Poster › Research
- Published
From the selective serotonin transporter inhibitor citalopram to the selective norepinephrine transporter inhibitor talopram : Synthesis and structure-activity relationship studies. / Eildal, Jonas Nii Nortey; Andersen, Jacob; Kristensen, Anders Skov; Jørgensen, Anne Marie; Bang-Andersen, Benny; Jørgensen, Morten; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 51, No. 10, 2008, p. 3045-3048.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Giftstoffer fra hvepse og edderkopper i forskning og lægemiddeludvikling. / Strømgaard, Kristian.
In: Carlsbergfondet. Aarsskrift, 2008, p. 42-47.Research output: Contribution to journal › Journal article › Communication
- Published
Modified peptides as potent inhibitors of the postsynaptic density-95/N-methyl-D-aspartate receptor interaction. / Bach, Anders; Chi, Celestine N.; Olsen, Thomas B.; Pedersen, Søren Wittrup; Røder, Martin U.; Pang, Gar Fai; Clausen, Rasmus Prætorius; Jemth, Per; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 51, No. 20, 2008, p. 6450-6459.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Protein-protein interaktion : et nyt mål for udvikling af lægemidler. / Bach, Anders; Gottschalk, Marie; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Lægemiddelforskning, 2008, p. 10-12.Research output: Contribution to journal › Journal article › Communication
- 2007
- Published
Expressed protein ligation of ionotropic glutamate receptors. / Jensen, Mette Stougård; Kristensen, Anders Skov; Strømgaard, Kristian.
In: Biopolymers, Vol. 88, No. 4, 2007, p. 602.Research output: Contribution to journal › Conference abstract in journal › Research
- Published
Probing the pharmacophore of ginkgolides as glycine receptor antagonists. / Jensen, Anders Asbjørn; Begum, Nasreen; Vogensen, Stine Byskov; Knapp, Kolja Michael; Gundertofte, Klaus; Dzyuba, Sergei V.; Ishii, Hideki; Nakanishi, Koji; Kristiansen, Uffe; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 50, No. 7, 2007, p. 1610-1617.Research output: Contribution to journal › Journal article › Research › peer-review
- 2006
- Published
Uncompetitive antagonism of AMPA receptors : Mechanistic insights from studies of polyamine toxin derivatives. / Andersen, Trine F; Tikhonov, Denis B; Bølcho, Ulrik; Bolshakov, Konstantin; Nelson, Jared K; Pluteanu, Florentina; Mellor, Ian R; Egebjerg, Jan; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 49, No. 18, 07.09.2006, p. 5414-5423.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design, synthesis, and pharmacological characterization of polyamine toxin derivatives : potent ligands for the pore-forming region of AMPA receptors. / Jensen, Lars S; Bølcho, Ulrik; Egebjerg, Jan; Strømgaard, Kristian.
In: ChemMedChem, Vol. 1, No. 4, 04.2006, p. 419-428.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Protolytic properties of polyamine wasp toxin analogues studied by 13C NMR spectroscopy. / Strømgaard, Kristian; Piazzi, Lorna; Olsen, Christian A; Franzyk, Henrik; Jaroszewski, Jerzy W.
In: Magnetic Resonance in Chemistry, Vol. 44, No. 11, 2006, p. 1013-22.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Stoffer fra Tempeltæet (Ginkgo biloba) som redskaber for studier af hjernens funktion. / Jensen, Anders A.; Strømgaard, Kristian.
In: Dansk Kemi 83, Vol. 87, No. 1, 2006, p. 16-18.Research output: Contribution to journal › Journal article › Communication
- Published
Unaturlige aminosyrer skaber ny viden om proteiner. / Rannes, Julie; Andersen, Jacob; Jensen, Anders A.; Christensen, Leif; Strømgaard, Kristian.
In: Lægemiddelforskning, 2006, p. 28-29.Research output: Contribution to journal › Journal article › Communication
- 2005
- Published
Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist. / Andersen, Trine F; Vogensen, Stine B; Jensen, Lars S; Knapp, Kolja M; Strømgaard, Kristian.
In: Bioorganic & Medicinal Chemistry, Vol. 13, No. 17, 01.09.2005, p. 5104-5112.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Polyamine toxins : development of selective ligands for ionotropic receptors. / Strømgaard, Kristian; Jensen, Lars S; Vogensen, Stine B.
In: Toxicon, Vol. 45, No. 3, 01.03.2005, p. 249-254.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Natural products as tools for studies of ligand-gated ion channels. / Strømgaard, Kristian.
In: Chemical Record, Vol. 5, No. 4, 2005, p. 229-239.Research output: Contribution to journal › Journal article › Research › peer-review
- 2004
- Published
Preparation of a tritiated ginkgolide. / Strømgaard, Kristian; Suehiro, Makiko; Nakanishi, Koji.
In: Bioorganic & Medicinal Chemistry Letters, Vol. 14, No. 22, 15.11.2004, p. 5673-5675.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
AMPA receptor ligands : synthetic and pharmacological studies of polyamines and polyamine toxins. / Strømgaard, Kristian; Mellor, Ian.
In: Medicinal Research Reviews, Vol. 24, No. 5, 09.2004, p. 589-620.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Chemistry and biology of terpene trilactones from Ginkgo biloba. / Strømgaard, Kristian; Nakanishi, Koji.
In: Angewandte Chemie International Edition, Vol. 43, No. 13, 19.03.2004, p. 1640-1658.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Ginkgolides and glycine receptors : a structure-activity relationship study. / Jaracz, Stanislav; Nakanishi, Koji; Jensen, Anders A.; Strømgaard, Kristian.
In: Chemistry: A European Journal, Vol. 10, No. 6, 2004, p. 1507-18.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Site-specific incorporation of unnatural amino acids into proteins. / Strømgaard, Anne; Jensen, Anders A.; Strømgaard, Kristian.
In: ChemBioChem, Vol. 5, No. 7, 2004, p. 909-16.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of polyamines and polyamine toxins. An improved alkylation procedure. / Strømgaard, Kristian; Andersen, TF.
In: Tetrahedron Letters, Vol. 45, 2004, p. 7929-7933.Research output: Contribution to journal › Journal article › Research › peer-review
- 2003
Terpene trilactones from Ginkgo biloba are antagonists of cortical glycine and GABA(A) receptors. / Ivic, Lidija; Sands, Tristan T J; Fishkin, Nathan; Nakanishi, Koji; Kriegstein, Arnold R; Strømgaard, Kristian.
In: Journal of Biological Chemistry, Vol. 278, No. 49, 05.12.2003, p. 49279-49285.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Contrasting actions of philanthotoxin-343 and philanthotoxin-(12) on human muscle nicotinic acetylcholine receptors. / Brier, Tim J; Mellor, Ian R; Tikhonov, Denis B; Neagoe, Ioana; Shao, Zuoyi; Brierley, Matt J; Strømgaard, Kristian; Jaroszewski, Jerzy W; Krogsgaard-Larsen, Povl; Usherwood, Peter N R.
In: Molecular Pharmacology, Vol. 64, No. 4, 10.2003, p. 954-964.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Preparation of 7-substituted ginkgolide derivatives : potent platelet activating factor (PAF) receptor antagonists. / Vogensen, Stine Byskov; Strømgaard, Kristian; Shindou, Hideo; Jaracz, Stanislav; Suehiro, Makiko; Ishii, Satoshi; Shimizu, Takao; Nakanishi, Koji.
In: Journal of Medicinal Chemistry, Vol. 46, No. 4, 13.02.2003, p. 601-608.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Modification of the philanthotoxin-343 polyamine moiety results in different structure-activity profiles at muscle nicotinic ACh, NMDA and AMPA receptors. / Mellor, I R; Brier, T J; Pluteanu, F; Strømgaard, K; Saghyan, A; Eldursi, N; Brierley, M J; Andersen, K; Jaroszewski, J W; Krogsgaard-Larsen, P; Usherwood, P N R.
In: Neuropharmacology, Vol. 44, No. 1, 01.2003, p. 70-80.Research output: Contribution to journal › Journal article › Research › peer-review
- 2002
- Published
Solid-phase synthesis of polyamine toxin analogues : potent and selective antagonists of Ca2+-permeable AMPA receptors. / Kromann, Hasse; Krikstolaityte, Sonata; Andersen, Anne J; Andersen, Kim; Krogsgaard-Larsen, Povl; Jaroszewski, Jerzy W; Egebjerg, Jan; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 45, No. 26, 19.12.2002, p. 5745-5754.Research output: Contribution to journal › Journal article › Research › peer-review
Ginkgolide derivatives for photolabeling studies : preparation and pharmacological evaluation. / Strømgaard, Kristian; Saito, D Roland; Shindou, Hideo; Ishii, Satoshi; Shimizu, Takao; Nakanishi, Koji.
In: Journal of Medicinal Chemistry, Vol. 45, No. 18, 29.08.2002, p. 4038-4046.Research output: Contribution to journal › Journal article › Research › peer-review
Ginkgolides : selective acetylations, translactonization, and biological evaluation. / Jaracz, Stanislav; Strømgaard, Kristian; Nakanishi, Koji.
In: Journal of Organic Chemistry, Vol. 67, No. 13, 28.06.2002, p. 4623-4626.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Solid-phase synthesis and pharmacological evaluation of analogues of PhTX-12-A potent and selective nicotinic acetylcholine receptor antagonist. / Strømgaard, Kristian; Mellor, Ian R; Andersen, Kim; Neagoe, Ioana; Pluteanu, Florentina; Usherwood, Peter N R; Krogsgaard-Larsen, Povl; Jaroszewski, Jerzy W.
In: Bioorganic & Medicinal Chemistry Letters, Vol. 12, No. 8, 22.04.2002, p. 1159-1162.Research output: Contribution to journal › Journal article › Research › peer-review
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PDZ domain-mediated interactions of G protein-coupled receptors with postsynaptic density protein 95: quantitative characterization of interactions
Research output: Contribution to journal › Journal article › Research › peer-review
Published