Kristian Strømgaard
Professor
Medicinal Chemistry Research
Jagtvej 162, 2100 København Ø, 30, Building: 240
- 2015
- Published
Binding of the Multimodal Antidepressant Drug Vortioxetine to the Human Serotonin Transporter. / Andersen, Jacob; Ladefoged, Lucy Kate; Wang, Danyang; Kristensen, Trine N Bjerre; Bang-Andersen, Benny; Kristensen, Anders S; Schiøtt, Birgit; Strømgaard, Kristian.
In: A C S Chemical Neuroscience, Vol. 6, No. 11, 18.11.2015, p. 1892-900.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Binding site residues control inhibitor selectivity in the human norepinephrine transporter but not in the human dopamine transporter. / Andersen, Jacob; Ringsted, Kristoffer B; Bang-Andersen, Benny; Strømgaard, Kristian; Kristensen, Anders S.
In: Scientific Reports, Vol. 5, 15650, 2015, p. 1-12.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Rigidified Clicked Dimeric Ligands for Studying the Dynamics of the PDZ1-2 Supramodule of PSD-95. / Eildal, Jonas N N; Bach, Anders; Dogan, Jakob; Ye, Fei; Zhang, Mingjie; Jemth, Per; Strømgaard, Kristian.
In: ChemBioChem, Vol. 16, 2015, p. 64–69.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design and Synthesis of High-Affinity Dimeric Inhibitors Targeting the Interactions between Gephyrin and Inhibitory Neurotransmitter Receptors. / Maric, Hans-Michael; Kasaragod, Vikram Babu; Kedström, Linda Maria Haugaard; Hausrat, Torben Johann; Kneussel, Matthias; Schindelin, Hermann; Strømgaard, Kristian.
In: Angewandte Chemie (International ed. in English), Vol. 54, No. 2, 07.01.2015, p. 490-4.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design, Synthesis, and Characterization of Fatty Acid Derivatives of a Dimeric Peptide-Based Postsynaptic Density-95 (PSD-95) Inhibitor. / Nissen, Klaus B; Andersen, Julie J; Haugaard-Kedström, Linda Maria; Bach, Anders; Strømgaard, Kristian.
In: Journal of Medicinal Chemistry, Vol. 58, 2015, p. 1575-1580.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Targeting Protein-Protein Interactions with Trimeric Ligands: High Affinity Inhibitors of the MAGUK Protein Family. / Nissen, Klaus B; Kedström, Linda Maria Haugaard; Wilbek, Theis S; Nielsen, Line S; Åberg, Emma; Kristensen, Anders S; Bach, Anders; Jemth, Per; Strømgaard, Kristian.
In: PLOS ONE, Vol. 10, No. 2, e0117668, 2015, p. 1-17.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Binding of ArgTX-636 in the NMDA receptor ion channel. / Poulsen, Mette H; Andersen, Jacob; Christensen, Rune; Hansen, Kasper Bø; Traynelis, Stephen F; Strømgaard, Kristian; Kristensen, Anders Skov.
In: Journal of Molecular Biology, Vol. 427, No. 1, 16.01.2015, p. 176-89.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Importance of the Extracellular Loop 4 in the Human Serotonin Transporter for Inhibitor Binding and Substrate Translocation. / Rannversson, Hafsteinn; Wilson, Pamela; Kristensen, Kristina Birch; Sinning, Steffen; Kristensen, Anders Skov; Strømgaard, Kristian; Andersen, Jacob.
In: The Journal of Biological Chemistry, Vol. 290, No. 23, 05.06.2015, p. 14582-94.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Fatty acid derivatives of dimeric inhibitors of PSD-95. / Strømgaard, Kristian (Inventor); Bach, Anders (Inventor); Nissen, Klaus Bertram (Inventor).
IPC No.: A61K38/17 . Patent No.: WO2015/078477A1.Research output: Patent
- Published
Identification and characterization of a small-molecule inhibitor of death-associated protein kinase 1. / Wilbek, Theis S; Skovgaard, Tine; Sorrell, Fiona J; Knapp, Stefan; Berthelsen, Jens; Strømgaard, Kristian.
In: ChemBioChem, Vol. 16, No. 1, 02.01.2015, p. 59-63.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Polyamine toxins from spiders and wasps : Polyamine toxins from spiders and wasps. / Xiong, Xiaofeng; Strømgaard, Kristian.
Polyamines: A Universal Molecular Nexus for Growth, Survival, and Specialized Metabolism. Springer, Japan, 2015. p. 201-214.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
ID: 1302559
Most downloads
-
2912
downloads
PDZ domain-mediated interactions of G protein-coupled receptors with postsynaptic density protein 95: quantitative characterization of interactions
Research output: Contribution to journal › Journal article › Research › peer-review
Published