Kristian Strømgaard
Professor
Medicinal Chemistry Research
Jagtvej 162, 2100 København Ø, 30, Building: 240
- 2016
- Published
Interrogating the Molecular Basis for Substrate Recognition in Serotonin and Dopamine Transporters with High-Affinity Substrate-Based Bivalent Ligands. / Andersen, Jacob; Ladefoged, Lucy Kate; Kristensen, Trine N Bjerre; Munro, Lachlan; Grouleff, Julie; Stuhr-Hansen, Nicolai; Kristensen, Anders S; Schiøtt, Birgit; Strømgaard, Kristian.
In: A C S Chemical Neuroscience, Vol. 7, No. 10, 19.10.2016, p. 1406-1417.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Importance of a Conserved Lys/Arg Residue for Ligand/PDZ Domain Interactions as Examined by Protein Semisynthesis. / Pedersen, Søren W; Moran, Griffin E; Sereikaité, Vita; Kedström, Linda Maria Haugaard; Strømgaard, Kristian.
In: ChemBioChem, Vol. 17, No. 20, 17.10.2016, p. 1936-1944.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Precise Somatotopic Thalamocortical Axon Guidance Depends on LPA-Mediated PRG-2/Radixin Signaling. / Cheng, Jin; Sahani, Sadhna; Hausrat, Torben Johann; Yang, Jenq-Wei; Ji, Haichao; Schmarowski, Nikolai; Endle, Heiko; Liu, Xinfeng; Li, Yunbo; Böttche, Rahel; Radyushkin, Konstantin; Maric, Hans M; Hoerder-Suabedissen, Anna; Molnár, Zoltán; Prouvot, Pierre-Hugues; Trimbuch, Thorsten; Ninnemann, Olaf; Huai, Jisen; Fan, Wei; Visentin, Barbara; Sabbadini, Roger; Strømgaard, Kristian; Stroh, Albrecht; Luhmann, Heiko J; Kneussel, Matthias; Nitsch, Robert; Vogt, Johannes.
In: Neuron, Vol. 92, No. 1, 05.10.2016, p. 126-142.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Effects of the dimeric PSD-95 inhibitor UCCB01-144 in mouse models of pain, cognition and motor function. / Andreasen, Jesper T; Nasser, Arafat; Caballero-Puntiverio, Maitane; Sahlholt, Maj; Bach, Anders; Gynther, Mikko; Strømgaard, Kristian; Pickering, Darryl S.
In: European Journal of Pharmacology, Vol. 780, 05.06.2016, p. 166-73.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Ligand binding to the PDZ domains of postsynaptic density protein 95. / Toto, Angelo; Pedersen, Søren W; Karlsson, O Andreas; Moran, Griffin E; Andersson, Eva; Chi, Celestine N; Strømgaard, Kristian; Gianni, Stefano; Jemth, Per.
In: Protein Engineering Design and Selection (Print), Vol. 29, No. 5, 05.2016, p. 169-75.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Genetically encoded photocrosslinkers locate the high-affinity binding site of antidepressant drugs in the human serotonin transporter. / Rannversson, Hafsteinn; Andersen, Jacob; Hall, Lena Sørensen; Bang-Andersen, Benny; Park, Minyoung; Huber, Thomas; Sakmar, Thomas P; Strømgaard, Kristian.
In: Nature Communications, Vol. 7, 11261, 19.04.2016, p. 1-9.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structure-activity relationship studies of citalopram derivatives : examining substituents conferring selectivity for the allosteric site in the serotonin transporter. / Larsen, M Andreas B; Plenge, Per; Andersen, Jacob; Eildal, Jonas Nii Nortey; Kristensen, Anders S; Bøgesø, Klaus P; Gether, Ulrik; Strømgaard, Kristian; Bang-Andersen, Benny; Loland, Claus J.
In: British Journal of Pharmacology, Vol. 173, No. 5, 03.2016, p. 925-936.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design and synthesis of triazole-based peptidomimetics of a PSD-95 PDZ domain inhibitor. / Bach, Anders; Pedersen, Thomas B.; Strømgaard, Kristian.
In: MedChemComm, Vol. 7, No. 3, 2016, p. 531-536.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of symmetrical and non-symmetrical bivalent neurotransmitter ligands. / Stuhr-Hansen, Nicolai; Andersen, Jacob; Thygesen, Mikkel Boas; Strømgaard, Kristian.
In: ChemistrySelect, Vol. 1, No. 3, 2016, p. 407-413.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Total synthesis and structure–activity relationship studies of a series of selective G protein inhibitors. / Xiong, Xiaofeng; Zhang, Hang; Underwood, Christina R.; Harpsøe, Kasper; Gardella, Thomas J.; Wöldike, Mie F.; Mannstadt, Michael; Gloriam, David E.; Bräuner-osborne, Hans; Strømgaard, Kristian.
In: Nature Chemistry, Vol. 8, No. 11, 2016, p. 1035-1041.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1302559
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PDZ domain-mediated interactions of G protein-coupled receptors with postsynaptic density protein 95: quantitative characterization of interactions
Research output: Contribution to journal › Journal article › Research › peer-review
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