Petrine Wellendorph

Petrine Wellendorph

Associate Professor


  1. 2019
  2. Published

    Five-membered N-heterocyclic Scaffolds as Novel Amino Bioisosteres at gamma-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters. / Giraudo, Alessandro; Krall, Jacob; Bavo, Francesco; Nielsen, Birgitte; Kongstad, Kenneth Thermann; Rolando, Barbara; De Blasio, Rosella; Gloriam, David E; Löffler, Rebekka; Thiesen, Louise; Harpsøe, Kasper; Frydenvang, Karla; Boschi, Donatella; Wellendorph, Petrine; Lolli, Marco L; Jensen, Anders A.; Frølund, Bente.

    In: Journal of Medicinal Chemistry, Vol. 62, No. 12, 27.06.2019, p. 5797-5809.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. E-pub ahead of print

    Structural and molecular aspects of betaine-GABA transporter 1 (BGT1) and its relation to brain function. / Kickinger, Stefanie; Hellsberg, Eva; Frølund, Bente; Schousboe, Arne; Ecker, Gerhard F; Wellendorph, Petrine.

    In: Neuropharmacology, 18.05.2019.

    Research output: Contribution to journalReviewResearchpeer-review

  4. Published

    Synthesis and Pharmacological Evaluation of [C-11]4-Methoxy-N-[2-(thiophen-2-yl) imidazo[1,2-a] pyridin-3-yl]benzamide as a Brain Penetrant PET Ligand Selective for the delta-Subunit-Containing gamma-Aminobutyric Acid Type A Receptors. / L'Estrade, Elina T.; Hansen, Hanne D.; Falk-Petersen, Christina; Haugaard, Anne; Griem-Krey, Nane; Jung, Sascha; Lueddens, Hartmut; Schirmeister, Tanja; Erlandsson, Maria; Ohlsson, Tomas; Knudsen, Gitte M.; Herth, Matthias M.; Wellendorph, Petrine; Frolund, Bente.

    In: ACS Omega, Vol. 4, No. 5, 05.2019, p. 8846-8851.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Lack of evidence for synaptic high-affinity γ-hydroxybutyric acid (GHB) transport in rat brain synaptosomes and 11 Na+ -dependent SLC neurotransmitter transporters. / Thiesen, Louise; Frølund, Bente; Wellendorph, Petrine.

    In: Journal of Neurochemistry, Vol. 149, No. 2, 04.2019, p. 195-210.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Discovery of 2-(Imidazo[1,2-b]pyridazin-2-yl)acetic Acid as a New Class of Ligands Selective for the γ-Hydroxybutyric Acid (GHB) High-Affinity Binding Sites. / Krall, Jacob; Bavo, Francesco; Falk-Petersen, Christina B; Jensen, Claus Hatt; Nielsen, Julie Olsson; Tian, Yongsong; Anglani, Valeria; Kongstad, Kenneth Thermann; Piilgaard, Louise; Nielsen, Birgitte; Gloriam, David E; Kehler, Jan; Jensen, Anders A.; Harpsøe, Kasper; Wellendorph, Petrine; Frølund, Bente.

    In: Journal of Medicinal Chemistry, Vol. 62, No. 5, 14.03.2019, p. 2798-2813.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Autoradiography as a Simple and Powerful Method for Visualization and Characterization of Pharmacological Targets. / Griem-Krey, Nane; Klein, Anders Bue; Herth, Matthias; Wellendorph, Petrine.

    In: Journal of visualized experiments : JoVE, No. 145, e58879, 12.03.2019.

    Research output: Contribution to journalJournal articleCommunication

  8. 2018
  9. Published

    Synthesis, pharmacological activity and molecular modeling studies of a series of 2-amino-1,4,5,6-tetrahydropyrimidine-5-carboxylic acid analogues as betaine/GABA transporter 1 (BGT1) substrate-inhibitors. / Kickinger, Stefanie; Al-Khawaja, Anas; Haugaard, Anne Staehr; Loeffler, Rebekka; Damgaard, Maria; Eckert, Gerhard; Frolund, Bente; Wellendorph, Petrine.

    2018. Abstract from 256th National Meeting and Exposition of the American-Chemical-Society (ACS) - Nanoscience, Nanotechnology and Beyond, United States.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  10. Published

    Inhibition of GABA transporters fails to afford significant protection following focal cerebral ischemia. / Lie, Maria Ek; Gowing, Emma K; Clausen, Rasmus P; Wellendorph, Petrine; Clarkson, Andrew N.

    In: Journal of Cerebral Blood Flow and Metabolism, Vol. 38, No. 1, 2018, p. 166-173.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Pharmacological Characterization of [3H]ATPCA as a Substrate for Studying the Functional Role of the Betaine/GABA Transporter 1 and the Creatine Transporter. / Al-Khawaja, Anas; Haugaard, Anne S; Marek, Ales; Löffler, Rebekka; Thiesen, Louise; Santiveri, Monica; Damgaard, Maria; Bundgaard, Christoffer; Frølund, Bente; Wellendorph, Petrine.

    In: A C S Chemical Neuroscience, Vol. 9, No. 3, 2018, p. 545–554.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. 2017
  13. Published

    GAT3 selective substrate l-isoserine upregulates GAT3 expression and increases functional recovery after a focal ischemic stroke in mice. / Lie, Maria Ek; Gowing, Emma K; Johansen, Nina B; Dalby, Nils Ole; Thiesen, Louise; Wellendorph, Petrine; Clarkson, Andrew N.

    In: Journal of Cerebral Blood Flow and Metabolism, 21.11.2017.

    Research output: Contribution to journalJournal articleResearchpeer-review

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ID: 1301791