Employees – University of Copenhagen

Rasmus Prætorius Clausen

Rasmus Prætorius Clausen

Associate Professor


  1. 2019
  2. Accepted/In press

    Use of the 4-Hydroxy-Triazole Moiety as a Bioisosteric Tool for the Development of Ionotropic Glutamate Receptor Ligands. / Sainas, Stefano; Temperini, Piero; Farnsworth, Jill C; Yi, Feng; Møllerud, Stine; Jensen, Anders A.; Nielsen, Birgitte; Kastrup, Jette Sandholm Jensen; Hansen, Kasper B; Boschi, Donatella; Pickering, Darryl S; Clausen, Rasmus Prætorius; Lolli, Marco.

    In: Journal of Medicinal Chemistry, 2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. 2018
  4. Published

    Elucidation of fluorine's impact on pKa and in vitro Pgp-mediated efflux for a series of PDE9 inhibitors. / Fjelbye, Kasper; Marigo, Mauro; Clausen, Rasmus P.; Jørgensen, Erling B.; Christoffersen, Claus T.; Juhl, Karsten.

    In: MedChemComm, Vol. 9, No. 5, 2018, p. 893-896.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Inhibition of GABA transporters fails to afford significant protection following focal cerebral ischemia. / Lie, Maria Ek; Gowing, Emma K; Clausen, Rasmus P; Wellendorph, Petrine; Clarkson, Andrew N.

    In: Journal of Cerebral Blood Flow and Metabolism, Vol. 38, No. 1, 2018, p. 166-173.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. 2017
  7. Published

    Development of Non-GAT1-Selective Inhibitors : Challenges and Achievements. / Damgaard, Maria; Haugaard, Anne Stæhr; Kickinger, Stefanie; Al-Khawaja, Anas; Lie, Maria E K; Ecker, Gerhard F; Clausen, Rasmus Prætorius; Frølund, Bente.

    Advances in Neurobiology. Vol. 16 Springer, 2017. p. 315-332.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  8. Published

    Enantioselective Fluorination of Spirocyclic β-Prolinals Using Enamine Catalysis. / Fjelbye, Kasper; Marigo, Mauro; Clausen, Rasmus Prætorius; Juhl, Karsten.

    In: SYNLETT: Accounts and Rapid Communications in Chemical Synthesis, Vol. 28, No. 4, st-2016-b0535-l, 2017, p. 425-428.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Preparation of Spirocyclic β-Proline Esters : Geometrically Restricted Building Blocks for Medicinal Chemistry. / Fjelbye, Kasper; Marigo, Mauro; Clausen, Rasmus Prætorius; Juhl, Karsten.

    In: SYNLETT: Accounts and Rapid Communications in Chemical Synthesis, Vol. 28, No. 2, st-2016-b0534-l, 2017, p. 231-234.

    Research output: Contribution to journalReviewResearchpeer-review

  10. Published

    Radiosynthesis and Evaluation of [(11)C]3-Hydroxycyclopent-1-enecarboxylic Acid as Potential PET Ligand for the High-Affinity γ-Hydroxybutyric Acid Binding Sites. / Jensen, Claus H; Hansen, Hanne D; Bay, Tina; Vogensen, Stine B; Lehel, Szabolcs; Thiesen, Louise; Bundgaard, Christoffer; Clausen, Rasmus P; Knudsen, Gitte M; Herth, Matthias M; Wellendorph, Petrine; Frølund, Bente.

    In: A C S Chemical Neuroscience, Vol. 8, No. 1, 18.01.2017, p. 22-27.

    Research output: Contribution to journalLetterResearchpeer-review

  11. Published

    Identification of AICP as a GluN2C-Selective N-Methyl-d-Aspartate Receptor Superagonist at the GluN1 Glycine Site. / Jessen, Maja; Frederiksen, Kristen; Yi, Feng; Clausen, Rasmus P; Hansen, Kasper B; Bräuner-Osborne, Hans; Kilburn, John Paul; Damholt, Anders.

    In: Molecular Pharmacology, Vol. 92, No. 2, 08.2017, p. 151-161.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1). / Jørgensen, Lars; Al-Khawaja, Anas; Kickinger, Stefanie; Vogensen, Stine B; Skovgaard-Petersen, Jonas; Rosenthal, Emil; Borkar, Nrupa; Löffler, Rebekka; Madsen, Karsten K; Bräuner-Osborne, Hans; Schousboe, Arne; Ecker, Gerhard F; Wellendorph, Petrine; Clausen, Rasmus P.

    In: Journal of Medicinal Chemistry, Vol. 60, No. 21, 09.10.2017, p. 8834-8846.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Molecular Hybridization of Potent and Selective γ-Hydroxybutyric Acid (GHB) Ligands: Design, Synthesis, Binding Studies, and Molecular Modeling of Novel 3-Hydroxycyclopent-1-enecarboxylic Acid (HOCPCA) and trans-γ-Hydroxycrotonic Acid (T-HCA) Analogs. / Krall, Jacob; Jensen, Claus Hatt; Bavo, Francesco; Falk-Petersen, Christina Birkedahl; Haugaard, Anne Stæhr; Vogensen, Stine Byskov; Tian, Yongsong; Nittegaard-Nielsen, Mia; Sigurdardóttir, Sara Björk; Kehler, Jan; Kongstad, Kenneth Thermann; Gloriam, David E.; Clausen, Rasmus Prætorius; Harpsøe, Kasper; Wellendorph, Petrine; Frølund, Bente.

    In: Journal of Medicinal Chemistry, Vol. 60, No. 21, 2017, p. 9022-9039.

    Research output: Contribution to journalJournal articleResearchpeer-review

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