Tommy Nørskov Johansen
Associate Professor / Head of Studies
Medicinal Chemistry Research
Jagtvej 162, 2100 København Ø, 30, Building: 211
- 2019
- Published
N-(7-(1H-imidazol-1-yl)-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl)benzamide - a new kainate receptor selective antagonist and analgesic : Synthesis, X-ray crystallography, structure-affinity relationships, in vitro and in vivo pharmacology. / Møllerud, Stine; Hansen, Rie B; Pallesen, Jakob S; Temperini, Piero; Pasini, Diletta; Bornholdt, Jan; Nielsen, Birgitte; Mamedova, Esmira; Chalupnik, Paulina; Paternain, Ana V; Lerma, Juan; Del Castillo, Marta Diaz; Andreasen, Jesper T; Frydenvang, Karla; Kastrup, Jette Sandholm; Johansen, Tommy N; Pickering, Darryl S.
In: ACS Chemical Neuroscience, Vol. 10, 2019, p. 4685-4695.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
N1-Substituted Quinoxaline-2,3-diones as Kainate Receptor Antagonists: X-ray Crystallography, Structure-Affinity Relationships and in vitro Pharmacology. / Pallesen, Jakob Staun; Møllerud, Stine; Frydenvang, Karla Andrea; Pickering, Darryl S; Bornholt, Jan; Nielsen, Birgitte; Pasini, Diletta; Han, Liwei; Marconi, Laura; Kastrup, Jette Sandholm Jensen; Johansen, Tommy Nørskov.
In: A C S Chemical Neuroscience, Vol. 10, 20.03.2019, p. 1841-1853.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1302791