Albert J. Kooistra

Albert J. Kooistra

Associate Professor


  1. 2019
  2. Published

    Aminergic GPCR-Ligand Interactions: A Chemical and Structural Map of Receptor Mutation Data

    Vass, M., Podlewska, S., De Esch, I. J. P., Bojarski, A. J., Leurs, R., Kooistra, Albert J. & De Graaf, C., 2019, In: Journal of Medicinal Chemistry. 62, 8, p. 3784-3839 56 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. 2018
  4. Development of novel fluorescent histamine H1-receptor antagonists to study ligand-binding kinetics in living cells

    Stoddart, L. A., Vernall, A. J., Bouzo-Lorenzo, M., Bosma, R., Kooistra, Albert J., De Graaf, C., Vischer, H. F., Leurs, R., Briddon, S. J., Kellam, B. & Hill, S. J., 1 Dec 2018, In: Scientific Reports. 8, 1, 1572.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Structural insights into serotonin receptor ligands polypharmacology

    Podlewska, S., Kafel, R., Lacivita, E., Satała, G., Kooistra, Albert J., Vass, M., de Graaf, C., Leopoldo, M., Bojarski, A. J. & Mordalski, S., 10 May 2018, In: European Journal of Medicinal Chemistry. 151, p. 797-814 18 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Chemical Diversity in the G Protein-Coupled Receptor Superfamily

    Vass, M., Kooistra, Albert J., Yang, D., Stevens, R. C., Wang, M. W. & de Graaf, C., 1 May 2018, In: Trends in Pharmacological Sciences. 39, 5, p. 494-512 19 p.

    Research output: Contribution to journalReviewResearchpeer-review

  7. Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology

    Hauwert, N. J., Mocking, T. A. M., Da Costa Pereira, D., Kooistra, Albert J., Wijnen, L. M., Vreeker, G. C. M., Verweij, E. W. E., De Boer, A. H., Smit, M. J., De Graaf, C., Vischer, H. F., De Esch, I. J. P., Wijtmans, M. & Leurs, R., 28 Mar 2018, In: Journal of the American Chemical Society. 140, 12, p. 4232-4243 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. 3D-e-Chem: Structural Cheminformatics Workflows for Computer-Aided Drug Discovery

    Kooistra, Albert J., Vass, M., McGuire, R., Leurs, R., de Esch, I. J. P., Vriend, G., Verhoeven, S. & de Graaf, C., 20 Mar 2018, In: ChemMedChem. 13, 6, p. 614-626 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    A Structural Framework for GPCR Chemogenomics: What’s In a Residue Number?

    Vass, M., Kooistra, Albert J., Verhoeven, S., Gloriam, David E., de Esch, I. J. P. & de Graaf, C., 1 Jan 2018, Methods in Molecular Biology. Humana Press, p. 73-113 41 p. (Methods in Molecular Biology, Vol. 1705).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  10. 2017
  11. Structural Chemogenomics Databases to Navigate Protein-Ligand Interaction Space

    Kanev, G. K., Kooistra, Albert J., de Esch, I. J. P. & de Graaf, C., 3 Jun 2017, The Future of Drug Discovery. Elsevier Science Inc., Vol. 1-8. p. 444-471 28 p.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  12. 3D-e-Chem-VM: Structural Cheminformatics Research Infrastructure in a Freely Available Virtual Machine

    McGuire, R., Verhoeven, S., Vass, M., Vriend, G., De Esch, I. J. P., Lusher, S. J., Leurs, R., Ridder, L., Kooistra, Albert J., Ritschel, T. & De Graaf, C., 27 Feb 2017, In: Journal of Chemical Information and Modeling. 57, 2, p. 115-121 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Kinase-Centric Computational Drug Development

    Kooistra, Albert J. & Volkamer, A., 1 Jan 2017, Annual Reports in Medicinal Chemistry. Academic Press, p. 263-299 37 p. (Annual Reports in Medicinal Chemistry, Vol. 50).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

ID: 196033213