Emil Märcher-Rørsted

Emil Märcher-Rørsted

Guest researcher, Guest Researcher

Member of:


    Publication year:
    1. 2023
    2. Published

      In Vitro and In Vivo Evaluation of Pellotine: A Hypnotic Lophophora Alkaloid

      Poulie, C. B. M., Chan, C. B., Parka, A., Lettorp, M., Vos, J., Raaschou, A., Pottie, E., Bundgaard, M. S., Sørensen, L. M. E., Cecchi, C. R., Märcher-Rørsted, E., Bach, A., Herth, M. M., Decker, A., Jensen, A. A., Elfving, B., Kretschmann, A. C., Stove, C. P., Kohlmeier, K. A., Cornett, C. & 3 others, Janfelt, Christian, Kornum, Birgitte Rahbek & Kristensen, Jesper Langgaard, 2023, In: ACS Pharmacology & Translational Science. 6, 10, p. 1492-1507

      Research output: Contribution to journalJournal articlepeer-review

    3. Published

      Introducing Conformational Restraints on 25CN-NBOH: A Selective 5-HT2A Receptor Agonist

      Marcher, Emil, Nykodemová, J., Harpsøe, Kasper, Jensen, Anders A. & Kristensen, Jesper Langgaard, 2023, In: ACS Medicinal Chemistry Letters. 14, 3, p. 319–325

      Research output: Contribution to journalJournal articlepeer-review

    4. 2021
    5. Published

      25CN-NBOH: A selective agonist for in vitro and in vivo investigations of the serotonin 2A receptor

      Marcher, Emil, Jensen, Anders A. & Kristensen, Jesper Langgaard, 2021, In: ChemMedChem. 16, 21, p. 3263-3270

      Research output: Contribution to journalReviewpeer-review

    6. Published

      An improved, scalable synthesis of the selective serotonin 2A receptor agonist 25CN-NBOH

      Marcher, Emil, Nykodemova, J. & Kristensen, Jesper Langgaard, 2021, In: SynOpen. 5, 2, p. 158-160

      Research output: Contribution to journalJournal articlepeer-review

    7. Published

      Erythrina Alkaloid Analogues as nAChR Antagonists-A Flexible Platform for Leads in Drug Discovery

      Clementson, S., Matheu, S. A., Marcher, Emil, Pedersen, H., Jensen, Anders A., Clausen, Rasmus Prætorius, Vital, P., Glibstrup, E., Jessing, M. & Kristensen, Jesper Langgaard, 2021, In: The Journal of Organic Chemistry. 86, 12, p. 8248-8262

      Research output: Contribution to journalJournal articlepeer-review

    8. 2020
    9. Published

      Biased agonism of clinically approved μ-opioid receptor agonists and TRV130 is not controlled by binding and signaling kinetics

      Pedersen, M. F., Wrobel, T. M., Marcher, Emil, Pedersen, D. S., Møller, T. C., Gabriele, F., Pedersen, H., Matosiuk, D., Foster, S. R., Bouvier, M. & Bräuner, Hans, 2020, In: Neuropharmacology. 166, 13 p., 107718.

      Research output: Contribution to journalJournal articlepeer-review

    10. Published

      Investigation of the 2,5-dimethoxy motif in phenethylamine Serotonin 2A receptor agonists

      Marcher, Emil, Halberstadt, A. L., Klein, A. K., Chatha, M., Jademyr, S., Jensen, Anders A. & Kristensen, Jesper Langgaard, 2020, In: ACS Chemical Neuroscience. 11, p. 1238-1244

      Research output: Contribution to journalLetterpeer-review

    11. Published

      The selective 5-HT2A receptor agonist 25CN-NBOH: structure-activity relationship, in vivo pharmacology, and in vitro and ex vivo binding characteristics of [3H]25CN-NBOH

      Jensen, Anders A., Halberstadt, A. L., Marcher, Emil, Odland, Anna Ulstein, Chatha, M., Speth, N., Liebscher, G., Hansen, M., Bräuner, Hans, Palner, M., Andreasen T., Jesper & Kristensen, Jesper Langgaard, 2020, In: Biochemical Pharmacology. 177, 16 p., 113979.

      Research output: Contribution to journalJournal articlepeer-review

    12. 2019
    13. Published

      Probing the Existence of a Metastable Binding Site at the β2-Adrenergic Receptor with Homobivalent Bitopic Ligands

      Gaiser, B. I., Danielsen, M., Marcher, Emil, Røpke Jørgensen, K., Wróbel, T. M., Frykman, M., Johansson, H., Bräuner, Hans, Gloriam, David E., Mathiesen, Jesper M. & Sejer Pedersen, D., 12 Sep 2019, In: Journal of Medicinal Chemistry. 62, 17, p. 7806-7839 34 p.

      Research output: Contribution to journalJournal articlepeer-review

    14. 2013
    15. Published

    ID: 160190095