Francesco Bavo

Francesco Bavo

Postdoc, Assistant Professor

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    1 - 10 out of 13Page size: 10
    1. 2023
    2. Published

      Structural and stereochemical determinants for hGAT3 inhibition: development of novel conformationally constrained and substituted analogs of (S)-isoserine

      Bavo, Francesco, Kickinger, Stefanie, Lie, M. E. K., Avgerinos, Christos, Wilhelmsen, Kristine Sloth, Wellendorph, Petrine & Frølund, Bente, 2023, In: Medicinal Chemistry Research. 32, p. 2299–2324

      Research output: Contribution to journal › Journal article › Research › peer-review

    3. Published

      Subnanomolar Affinity and Selective Antagonism at alpha 7 Nicotinic Receptor by Combined Modifications of 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624)

      Bavo, Francesco, Pallavicini, M., Pucci, S., Appiani, R., Giraudo, A., Oh, H., Kneisley, D. L., Eaton, B., Lucero, L., Gotti, C., Clementi, F., Whiteaker, P. & Bolchi, C., 2023, In: Journal of Medicinal Chemistry. 66, 1, p. 306–332

      Research output: Contribution to journal › Journal article › Research › peer-review

    4. 2022
    5. Published

      From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human α9α10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue

      Bavo, Francesco, Pallavicini, M., Pucci, S., Appiani, R., Giraudo, A., Eaton, B., Lucero, L., Gotti, C., Moretti, M., Whiteaker, P. & Bolchi, C., 2022, In: Journal of Medicinal Chemistry. 65, 14, p. 10079-10097

      Research output: Contribution to journal › Journal article › Research › peer-review

    6. 2021
    7. Published

      Determinants for α4β2 vs. α3β4 subtype selectivity of pyrrolidine-based nachrs ligands: A computational perspective with focus on recent cryo-em receptor structures

      Bavo, Francesco, Pallavicini, M., Appiani, R. & Bolchi, C., 2021, In: Molecules. 26, 12, 23 p., 3603.

      Research output: Contribution to journal › Journal article › Research › peer-review

    8. Published

      Structure-Activity Studies of 3,9-Diazaspiro[5.5]undecane-Based ?-Aminobutyric Acid Type A Receptor Antagonists with Immunomodulatory Effect

      Bavo, Francesco, De-Jong, H., Petersen, Jonas Odgaard, Falk-Petersen, C. B., Löffler, R., Sparrow, E., Rostrup, F., Eliasen, Jannik Nicklas, Wilhelmsen, K. S., Barslund, K., Bundgaard, C., Nielsen, Birgitte, Kristiansen, Uffe, Wellendorph, Petrine, Bogdanov, Y. & Frølund, Bente, 2021, In: Journal of Medicinal Chemistry. 64, 24, p. 17795-17812

      Research output: Contribution to journal › Journal article › Research › peer-review

    9. 2020

    10. Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype

      Bavo, Francesco, Pallavicini, M., Gotti, C., Appiani, R., Moretti, M., Colombo, S. F., Pucci, S., Viani, P., Budriesi, R., Renzi, M., Fucile, S. & Bolchi, C., 24 Dec 2020, In: Journal of Medicinal Chemistry. 63, 24, p. 15668-15692 25 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    11. 1,4-Benzodioxane, an evergreen, versatile scaffold in medicinal chemistry: A review of its recent applications in drug design

      Bolchi, C., Bavo, Francesco, Appiani, R., Roda, G. & Pallavicini, M., 15 Aug 2020, In: European Journal of Medicinal Chemistry. 200, 112419.

      Research output: Contribution to journal › Review › Research › peer-review

    12. Behavioural and pharmacological profiles of zebrafish administrated pyrrolidinyl benzodioxanes and prolinol aryl ethers with high affinity for heteromeric nicotinic acetylcholine receptors

      Braida, D., Ponzoni, L., Moretti, M., Viani, P., Pallavicini, M., Bolchi, C., Appiani, R., Bavo, Francesco, Gotti, C. & Sala, M., 1 Aug 2020, In: Psychopharmacology. 237, 8, p. 2317-2326 10 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    13. Efficient One-Pot Reductive Aminations of Carbonyl Compounds with Aquivion-Fe as a Recyclable Catalyst and Sodium Borohydride

      Airoldi, V., Piccolo, O., Roda, G., Appiani, R., Bavo, Francesco, Tassini, R., Paganelli, S., Arnoldi, S., Pallavicini, M. & Bolchi, C., 16 Jan 2020, In: European Journal of Organic Chemistry. 2020, 2, p. 162-168 7 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    14. Published

      Exploring the molecular determinants for subtype-selectivity of 2-amino-1,4,5,6-tetrahydropyrimidine-5-carboxylic acid analogs as betaine/GABA transporter 1 (BGT1) substrate-inhibitors

      Kickinger, S., Al-Khawaja, A., Haugaard, A. S., Lie, M. E. K., Bavo, Francesco, Loeffler, R., Damgaard, M., Ecker, G. F., Frølund, Bente & Wellendorph, Petrine, 2020, In: Scientific Reports. 10, 1, 15 p., 12992.

      Research output: Contribution to journal › Journal article › Research › peer-review

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    ID: 220215448