Søren Brøgger Christensen

Søren Brøgger Christensen

Professor emeritus, Professor, emeritus

Member of:


    1. 1973
    2. Published

      Organic hydroxylamine derivatives. VII. Isoxazolin 5 ones. An investigation of a reaction sequence previously stated to give 3 hydroxyisoxazoles

      Krogsgaard-Larsen, Povl, Christensen, Søren Brøgger & Hjeds, H., 1 Jan 1973, In: Acta Chemica Scandinavica. 27, 8, p. 2802-2812 11 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    3. Published

      Organic hydroxylamine derivatives. VIII. Structural analogues of GABA of the isoxazole enol betaine type. Synthesis of 5,6,7,8 tetrahydro 4H isoxazolo[3,4 d]azepin 3 ol zwitterion and some derivatives

      Krogsgaard-Larsen, Povl, Hjeds, H. & Christensen, Søren Brøgger, 1 Jan 1973, In: Acta Chemica Scandinavica. 27, 9, p. 3251-3258 8 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    4. 1977
    5. Published

      Muscimol analogues. I. Syntheses of 4- and 8-aminocycloheptenol[1,2 d]isoxazol-3-ols and 4-(3-aminopropyl)-5-methyl-3-isoxazolol

      Krogsgaard-Larsen, Povl, Natova, L. & Christensen, Søren Brøgger, 1 Jan 1977, In: ACTA CHEM. SCAND.. B31, 7, p. 577-583 7 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    6. 1978
    7. Published

      Phytochemical and pharmacological investigations of the genus Thapsia (Apiaceae)

      Rasmussen, U., Christensen, Søren Brøgger & Sandberg, F., 1 Jan 1978, In: PLANTA MED.. 33, 3, p. 301-302 2 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    8. Published

      Thapsigargine and thapsigargicine, two new histamine liberators from Thapsia garganica L

      Rasmussen, U., Christensen, Søren Brøgger & Sandberg, F., 1 Jan 1978, In: Acta Pharmaceutica Suecica. 15, 2, p. 133-140 8 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    9. 1980
    10. Published

      Thapsigargin, constitution of a sesquiterpene lactone histamine liberator from thapsia garganica

      Christensen, Søren Brøgger, Rasmussen, U. & Christophersen, C., 1980, In: Tetrahedron Letters. 21, 39, p. 3829-3830 2 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    11. Published

      Preparations of deuterium labelled guvacine and isoguvacine

      Christensen, Søren Brøgger & Krogsgaard-Larsen, Povl, 1 Jan 1980, In: Journal of Labelled Compounds and Radiopharmaceuticals. 17, 2, p. 191-202 12 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    12. 1981
    13. Published

      Proacaciberin, A cyanogenic glycoside from Acacia sieberiana var. Woodii

      Nartey, F., Brimer, L. & Christensen, Søren Brøgger, 1981, In: Phytochemistry. 20, 6, p. 1311-1314 4 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    14. Published

      Structural elucidation and partial synthesis of 3-hydroxyheterodendrin, a cyanogenic glucoside from Acacia sieberiana var. woodii

      Brimer, L., Christensen, Søren Brøgger, Jaroszewski, J. W. & Nartey, F., 1981, In: Phytochemistry. 20, 9, p. 2221-2223 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    15. Published

      Phytochemistry of the genus Thapsia

      Rasmussen, U., Christensen, Søren Brøgger & Sandberg, F., 1 Jan 1981, In: Planta Medica. 43, 4, p. 336-341 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    16. 1982
    17. Published

      1-β-vicianosyl-(S)-2-methylbutyrate, a 1-O-acylglycoside from Acacia sieberana var. Woodii

      Christensen, Søren Brøgger, Brimer, L. & Nartey, F., 1982, In: Phytochemistry. 21, 11, p. 2683-2685 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    18. Published

      2-β-d-Glucopyranosyloxy-2-methylpropanol in Acacia sieberana var. woodii

      Brimer, L., Christensen, Søren Brøgger & Nartey, F., 1982, In: Phytochemistry. 21, 8, p. 2005-2007 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    19. Published

      Structure and biological activity of sesquiterpene lactones from Thapsia species and of analogue derivatives

      Rasmussen, U., Christensen, Søren Brøgger & Patkar, S. A., 1 Jan 1982, In: Planta Medica. 45, 3, p. P23

      Research output: Contribution to journalJournal articleResearchpeer-review

    20. 1984
    21. Published

      Structure of histamine releasing guaianolides from Thapsia species

      Christensen, Søren Brøgger, Norup, E., Rasmussen, U. & Øgaard Madsen, J., 1984, In: Phytochemistry. 23, 8, p. 1659-1663 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    22. 1985
    23. Published

      Absolute configurations of the histamine liberating sesquiterpene lactones thapsigargin and trilobolide

      Christensen, Søren Brøgger & Norup, E., 1985, In: Tetrahedron Letters. 26, 1, p. 107-110 4 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    24. Published

      The ability of thapsigargin and thapsigargicin to activate cells involved in the inflammatory response

      Ali, H., Christensen, Søren Brøgger, Foreman, J. C., Pearce, F. L., Piotrowski, W. & Thastrup, Ole, 1985, In: British Journal of Pharmacology. 85, 3, p. 705-12 8 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    25. Published

      Atriplex nummularia, a source for the two molluscicide saponins: Hederagenin-3-O-β-D-glucuronopyranoside and calenduloside E

      Christensen, Søren Brøgger & Omar, A. A., 1 Dec 1985, In: Journal of Natural Products. 48, 1, 1 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    26. 1986
    27. Published

      The potencies of thapsigargin and analogues as activators of rat peritoneal mast cells

      Norup, E., Smitt, U. W. & Christensen, Søren Brøgger, 1 Jan 1986, In: Planta Medica. NO. 4, p. 251-255 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    28. Published

      Thapsigargin, a histamine secretagogue, is a non-12-O-tetradecanolphorbol-13-acetate (TPA) type tumor promoter in two-stage mouse skin carcinogenesis

      Hakii, H., Fujiki, H., Suganuma, M., Nakayasu, M., Tahira, T., Sugimura, T., Scheuer, P. J. & Christensen, Søren Brøgger, 1 Jun 1986, In: Journal of Cancer Research and Clinical Oncology. 111, 3, p. 177-181 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    29. Published

      Synergistic stimulation of histamine release from rat peritoneal mast cells by 12-O-tetradecanoylphorbol 13-acetate (TPA)-type and non-TPA-type tumor promoters

      Ohuchi, K., Hirasawa, N., Takahashi, C., Watanabe, M., Tsurufuji, S., Fujiki, H., Suganuma, M., Hakii, H., Sugimura, T. & Christensen, Søren Brøgger, 16 Jun 1986, In: BBA - Molecular Cell Research. 887, 1, p. 94-99 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    30. Published

      Isorhamnetin3-(2,6-dirhamnosylgalactoside)-7-rhamnoside and 3-(6-rhamnosylgalactoside)-7-rhamnoside from Rhazya stricta

      Andersen, W. K., Omar, A. A. & Christensen, Søren Brøgger, 23 Dec 1986, In: Phytochemistry. 26, 1, p. 291-294 4 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    31. 1987
    32. Published

      The inflammatory and tumor-promoting sesquiterpene lactone, thapsigargin, activates platelets by selective mobilization of calcium as shown by protein phosphorylations

      Thastrup, Ole, Linnebjerg, H., Bjerrum, P. J., Knudsen, J. B. & Christensen, Søren Brøgger, 1987, In: BBA General Subjects. 927, 1, p. 65-73 9 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    33. Published

      Stimulation of arachidonic acid metabolism in rat peritoneal macrophages by thapsigargin, a non-(12-O-tetradecanoylphorbol-13-acetate) (TPA)-type tumor promoter

      Ohuchi, K., Sugawara, T., Watanabe, M., Hirasawa, N., Tsurufuji, S., Fujiki, H., Sugimura, T. & Christensen, Søren Brøgger, 1 Jun 1987, In: Journal of Cancer Research and Clinical Oncology. 113, 4, p. 319-324 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    34. Published

      A new sesquiterpene from laserpitium latifolium

      Moldt, P., Smitt, U. W. & Christensen, Søren Brøgger, 1 Sep 1987, In: Journal of Natural Products. 50, 5, p. 974-975 2 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    35. 1988
    36. Published

      Effect of thapsigargin on cytoplasmic Ca2+ and proliferation of human lymphocytes in relation to AIDS

      Scharff, O., Foder, B., Thastrup, Ole, Hofmann, B., Møller, J., Ryder, L. P., Jacobsen, K. D., Langhoff, E., Dickmeiss, E. & Christensen, Søren Brøgger, 1988, In: BBA General Subjects. 972, 3, p. 257-64 8 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    37. Published

      Effects of thapsigargin in isolated rat thoracic aorta

      Mikkelsen, E. O., Thastrup, Ole & Christensen, Søren Brøgger, 1988, In: Pharmacology & Toxicology. 62, 1, p. 7-11 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    38. Published

      Dimethyl sulfoxide decreases the fluorescence yield of the reaction between histamine and ortho-phthalaldehyde and may influence histamine release

      Moldt, P., Andersen, W. K. & Christensen, Søren Brøgger, 1 Jun 1988, In: Agents and Actions. 24, 1-2, p. 35-39 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    39. Published

      Analysis of the stimulative effect of thapsigargin, a non‐TPA‐type tumour promoter, on arachidonic acid metabolism in rat peritoneal macrophages

      Ohuchi, K., Sugawara, T., Watanabe, M., Hirasawa, N., Tsurufuji, S., Fujiki, H., Christensen, Søren Brøgger & Sugimura, T., Jul 1988, In: British Journal of Pharmacology. 94, 3, p. 917-923 7 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    40. 1990
    41. Published

      HYDROINDENE SESQUITERPENES FROM THAPSIA-VILLOSA

      Smitt, U. W., Cornett, Claus, Norup, E. & Christensen, Søren Brøgger, 1990, In: Phytochemistry. 29, 3, p. 873-875 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    42. Published

      Inositol trisphosphate and thapsigargin discriminate endoplasmic reticulum stores of calcium in rat brain

      Verma, A., Hirsch, D. J., Hanley, M. R., Thastrup, O., Christensen, Søren Brøgger & Snyder, S. H., 1990, In: Biochemical and Biophysical Research Communications. 172, 2, p. 811-6 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    43. Published

      NEW PROAZULENE GUAIANOLIDES FROM THAPSIA-VILLOSA

      Smitt, U. W., Cornett, Claus, Andersen, A., Christensen, Søren Brøgger & Avato, P., 1990, In: Journal of Natural Products. 53, 6, p. 1479-1484 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    44. Published

      Ca2+ influx in human T lymphocytes is induced independently of inositol phosphate production by mobilization of intracellular Ca2+ stores. A study with the Ca2+ endoplasmic reticulum‐ATPase inhibitor thapsigargin

      Gouy, H., Cefai, D., Christensen, Søren Brøgger, Debré, P. & Bismuth, G., Oct 1990, In: European Journal of Immunology. 20, 10, p. 2269-2275 7 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    45. 1991
    46. Published

      Exciton Coupling in Circular Dichroic Spectroscopy as a Tool for Establishing the Absolute Configuration of alpha,beta-Unsaturated Esters of Allylic Alcohols

      Lauridsen, A., Cornett, Claus & Christensen, Søren Brøgger, 1991, In: Acta Chemica Scandinavica. Supplementum. 45, 1, p. 56-62 7 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    47. Published

      Novel Guaiane Esters from Thapsia villosa

      Lemmich, E., Smitt, U. W., Kastrup, Jette Sandholm Jensen & Christensen, Søren Brøgger, 1991, In: Phytochemistry. 30, p. 2987-2990 4 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    48. Published

      Nortrilobolide, a new potent guaianolide secretagogue from Thapsia garganica

      Smitt, U. W. & Christensen, Søren Brøgger, 25 Apr 1991, In: Planta Medica. 57, 2, p. 196-197 2 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    49. Published

      Thapsigargin-induced increase in cytoplasmic Ca2+concentration and aldosterone production in rat adrenal glomerulosa cells: Interaction with potassium and angiotensin-II

      Hajnóczky, G., Várnai, P., Holló, Z., Christensen, Søren Brøgger, Balla, T., Enyedi, P. & Spät, A., 1 May 1991, In: Endocrinology. 128, 5, p. 2639-2644 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    50. Published

      Cyclic AMP- and inositol phosphate-independent inhibition of Ca2+ influx by cholera toxin in CDS-stimulated jurkat T cells: A study with a cholera toxin-resistant cell variant and the Ca2+ endoplasmic reticulum-ATPase inhibitor thapsigargin

      Gouy, H., Cefai, D., Christensen, Søren Brøgger, Debre, P. & Bismuth, G., 1 Aug 1991, In: Journal of Immunology. 147, 3, p. 757-766 10 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    51. 1992
    52. Published

      The molluscicidal activity of coumarins from Ethulia conyzoides and of dicumarol

      Kady, M. M., Brimer, L., Furu, Peter, Lemmich, E., Nielsen, H. M., Thiilborg, S. T., Thastrup, Ole & Christensen, Søren Brøgger, 1992, In: Planta Medica. 58, 4, p. 334-7 4 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    53. Published

      Comparison of the Effects of Thapsigargin and BAY K 8644 on Spontaneous Mechanical Activity in Rat Portal Vein and Contractile Responses of Rat Cardiac Muscle

      Mikkelsen, E. O., Poulsen, S. H. & Christensen, Søren Brøgger, Feb 1992, In: Pharmacology & Toxicology. 70, 2, p. 152-156 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    54. Published

      Toxicodynamics of tumour promoters of mouse skin III. Specific binding of the tumour promoter thapsigargin as measured by the cold-acetone filter assay

      Christensen, Søren Brøgger, Hergenhahn, M., Roeser, H. & Hecker, E., 1 May 1992, In: Journal of Cancer Research and Clinical Oncology. 118, 5, p. 344-348 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    55. 1993
    56. Published

      Licochalcone A, a novel antiparasitic agent with potent activity against human pathogenic protozoan species of Leishmania

      Chen, M., Christensen, Søren Brøgger, Blom, J., Lemmich, E., Nadelmann, L., Fich, K., Theander, Thor Grundtvig & Kharazmi, A., 1993, In: Antimicrobial Agents and Chemotherapy. 37, 12, p. 2550-6 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    57. Published

      Localization of the acyl groups in proazulene guaianolides from Thapsia transtagana and Thapsia garganica

      Avato, P., Cornett, Claus, Andersen, A., Smitt, U. W. & Christensen, Søren Brøgger, 1993, In: Journal of Natural Products. 56, 3, p. 411-415 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    58. Published

      Molluscicidal saponins from Phytolacca dodecandra

      Thiilborg, S. T., Christensen, Søren Brøgger, Cornett, Claus, Olsen, C. E. & Lemmich, E., 1993, In: Phytochemistry. 32, 5, p. 1167-1171 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    59. Published

      Calcium entry in Xenopus oocytes: effects of inositol trisphosphate, thapsigargin and DMSO

      Lupu-Meiri, M., Beit-Or, A., Christensen, Søren Brøgger & Oron, Y., Feb 1993, In: Cell Calcium. 14, 2, p. 101-110 10 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    60. Published

      An attempt to develop an ELISA against the sesquiterpene lactone thapsigargin

      Jager, A. K., Smitt, U. W., Nyman, U. & Christensen, Søren Brøgger, 1 Dec 1993, In: Planta Medica. 59, 7 SUPPL., p. A679

      Research output: Contribution to journalJournal articleResearchpeer-review

    61. Published

      Structure-activity relationships of thapsigargin

      Nielsen, S. F., Andersen, A., Olsen, C. E., Treimann, M., Thastrup, Ole & Christensen, Søren Brøgger, 1 Dec 1993, In: Planta Medica. 59, 7 SUPPL., p. A678-A679

      Research output: Contribution to journalJournal articleResearchpeer-review

    62. Published

      Derivatives of thapsigargin as probes of its binding site on endoplasmic reticulum Ca2+ ATPase. Stereoselectivity and important functional groups

      Christensen, Søren Brøgger, Andersen, A., Poulsen, J. C. J. & Treiman, M., 13 Dec 1993, In: FEBS Letters. 335, 3, p. 345-348 4 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    63. 1994
    64. Published

      An antileishmanial chalcone from Chinese licorice roots

      Christensen, Søren Brøgger, Ming, C., Andersen, L., Hjørne, U., Olsen, C. E., Cornett, Claus, Theander, Thor Grundtvig & Kharazmi, A., 1994, In: Planta Medica. 60, 2, p. 121-3 2 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    65. Published

      Antileishmanial activity of licochalcone A in mice infected with Leishmania major and in hamsters infected with Leishmania donovani

      Chen, M., Christensen, Søren Brøgger, Theander, Thor Grundtvig & Kharazmi, A., 1994, In: Antimicrobial Agents and Chemotherapy. 38, 6, p. 1339-44 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    66. Published

      CA2+-ATPASE INHIBITORY ACTIVITY OF A LOCKED ANALOG OF THAPSIGARGIN

      Andersen, A., Treiman, M., Poulsen, J. C. J., Cornett, Claus, Moldt, P., Olsen, C. E. & Christensen, Søren Brøgger, 1994, In: Bioorganic & Medicinal Chemistry Letters. 4, 5, p. 657-660 4 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    67. Published

      Ca2+-ATPase inhibitory activity of a locked analogue of thapsigargin

      Christensen, Søren Brøgger, Olsen, C. E., Moldt, P., Cornett, Claus, Poulsen, J. J., Treiman, M. & Andersen, A., 1994, In: Bioorganic & Medicinal Chemistry Letters.

      Research output: Contribution to journalJournal articleResearchpeer-review

    68. Published

      Licochalcone A, a new antimalarial agent, inhibits in vitro growth of the human malaria parasite Plasmodium falciparum and protects mice from P. yoelii infection

      Chen, M., Theander, Thor Grundtvig, Christensen, Søren Brøgger, Hviid, Lars, Zhai, L. & Kharazmi, A., 1994, In: Antimicrobial Agents and Chemotherapy. 38, 7, p. 1470-5 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    69. Published

      Molluscicidal saponins from a Zimbabwean strain of Phytolacca dodecandra

      Thiilborg, S. T., Christensen, Søren Brøgger, Cornett, Claus, Olsen, C. E. & Lemmich, E., 1994, In: Phytochemistry. 36, 3, p. 753-759 7 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    70. Published

      SELECTIVE TRANSFORMATIONS OF THE CA-2+ PUMP INHIBITOR THAPSIGARGIN

      Andersen, A., Cornett, Claus, Lauridsen, A., Olsen, C. E. & Christensen, Søren Brøgger, 1994, In: Acta Chemica Scandinavica. Supplementum. 48, 4, p. 340-346 7 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    71. Published

      Thapsigargin: a novel molecular probe for studying intracellular calcium release and storage

      Thastrup, Ole, Dawson, A. P., Scharff, O., Foder, B., Cullen, P. J., Drøbak, B. K., Bjerrum, P. J., Christensen, Søren Brøgger & Hanley, M. R., 1994, In: Agents and Actions. 43, 3-4, p. 187-93 7 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    72. 1995
    73. Published

      Structure-activity relationships of analogues of thapsigargin modified at O-11 and O-12

      Nielsen, S. F., Thastrup, Ole, Pedersen, R., Olsen, C. E. & Christensen, Søren Brøgger, 1995, In: Journal of Medicinal Chemistry. 38, 2, p. 272-6 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    74. Published

      Synthesis of antiparasitic licorice chalcones

      Nielsen, S. F., Chen, M., Theander, Thor Grundtvig, Kharazmi, A. & Christensen, Søren Brøgger, 1995, In: Bioorganic & Medicinal Chemistry Letters. 5, p. 449-452 4 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    75. Published

      The antileishmanial agent licochalcone A interferes with the function of parasite mitochondria

      Zhai, L., Blom, J., Chen, M., Christensen, Søren Brøgger & Kharazmi, A., 1995, In: Antimicrobial Agents and Chemotherapy. 39, 12, p. 2742-8 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    76. 1996
    77. Published

      Syntheses of 11-hydroxylated guaianolides

      Lauridsen, A., Cornett, Claus, Vulpius, T., Moldt, P. & Christensen, Søren Brøgger, 1996, In: Acta Chemica Scandinavica. Supplementum. 50, 2, p. 150-157 8 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    78. 1997
    79. Published

      Discovery of oxygenated chalcoes as novel antimalarial agents

      Kharazmi, A., Chen, M., Theander, Thor Grundtvig & Christensen, Søren Brøgger, 1997, In: Annals of Tropical Medicine and Parasitology. 91, p. S91-S95 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    80. Published

      Discovery of oxygentade chalcones as novel antimalarial agents

      Kharazmi, A., Chen, M., Theander, Thor Grundtvig & Christensen, Søren Brøgger, 1997, In: Annals of Tropical Medicine and Parasitology. 91, SUPPL. 1, p. S91-S95

      Research output: Contribution to journalJournal articleResearchpeer-review

    81. Published

      Sesquiterpenoids from Thapsia species and medicinal chemistry of the thapsigargins.

      Christensen, Søren Brøgger, Andersen, A. & Smitt, U. W., 1997, In: Fortschritte der Chemie organischer Naturstoffe. Progress in the chemistry of organic natural products. Progrès dans la chimie des substances organiques naturelles. 71, p. 129-167 39 p.

      Research output: Contribution to journalReviewResearchpeer-review

    82. Published

      Synthesis, isolation and identification of glucuronides and mercapturic acids of a novel antiparasitic agent, licochalcone A

      Nadelmann, L., Tjornelund, J., Hansen, S. H., Cornett, Claus, Sidelmann, U. G., Braumann, U., Christensen, E. & Christensen, Søren Brøgger, 1997, In: Xenobiotica. 27, 7, p. 667-680 14 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    83. Published

      The novel oxygenated chalcone, 2,4-dimethoxy-4'-butoxychalcone, exhibits potent activity against human malaria parasite Plasmodium falciparum in vitro and rodent parasites Plasmodium berghei and Plasmodium yoelii in vivo

      Chen, M., Christensen, Søren Brøgger, Zhai, L., Rasmussen, M. H., Theander, Thor Grundtvig, Frøkjær, Sven, Steffansen, B., Davidsen, J. & Kharazmi, A., 1997, In: Journal of Infectious Diseases. 176, 5, p. 1327-33 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    84. Published

      Two new antiprotozoal 5-methylcoumarins from Vernonia brachycalyx

      Oketch-Rabah, H. A., Lemmich, E., Dossaji, S. F., Theander, Thor Grundtvig, Olsen, C. E., Cornett, Claus, Kharazmi, A. & Christensen, Søren Brøgger, 1997, In: Journal of Natural Products. 60, 5, p. 458-61 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    85. 1998
    86. Published

      Alkamides from Phyllanthus fraternus

      Sittie, A. A., Lemmich, E., Olsen, C. E., Hviid, Lars & Christensen, Søren Brøgger, 1998, In: Planta Medica. 64, 2, p. 192-3 1 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    87. Published

      Antiprotozoal properties of 16,17-dihydrobrachycalyxolide from Vernonia brachycalyx

      Oketch-Rabah, H. A., Christensen, Søren Brøgger, Frydenvang, Karla Andrea, Dossaji, S. F., Theander, Thor Grundtvig, Cornett, Claus, Watkins, W. M., Kharazmi, A. & Lemmich, E., 1998, In: Planta Medica. 64, 6, p. 559-62 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    88. Published

      Limonoids from Khaya senegalensis

      Khalid, S., Friedrichsen, G., Kharazmi, A., Theander, Thor Grundtvig, Olsen, C. & Christensen, Søren Brøgger, 1998, In: Phytochemistry. 49, 6, p. 1769-1772 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    89. Published

      Modifications of the alpha,beta-double bond in chalcones only marginally affect the antiprotozoal activities

      Nielsen, S. F., Kharazmi, A. & Christensen, Søren Brøgger, 1998, In: Bioorganic & Medicinal Chemistry. 6, 7, p. 937-45 8 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    90. Published

      A tool coming of age: Thapsigargin as an inhibitor of sarco-endoplasmic reticulum Ca2+-ATPases

      Treiman, M., Caspersen, C. & Christensen, Søren Brøgger, 1 Jan 1998, In: Trends in Pharmacological Sciences. 19, 4, p. 131-135 5 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    91. 1999
    92. Published

      Structure-activity studies: in vitro antileishmanial and antimalarial activities of anthraquinones from Morinda lucida

      Sittie, A. A., Lemmich, E., Olsen, C. E., Hviid, Lars, Kharazmi, A., Nkrumah, F. K. & Christensen, Søren Brøgger, 1999, In: Planta Medica. 65, 3, p. 259-61 2 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    93. Published

      The antileishmanial activity of novel oxygenated chalcones and their mechanism of action

      Zhai, L., Chen, M., Blom, J., Theander, Thor Grundtvig, Christensen, Søren Brøgger & Kharazmi, A., 1999, In: Journal of Antimicrobial Chemotherapy. 43, 6, p. 793-803 10 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    94. 2000
    95. Published

      Absolute configuration and antiprotozoal activity of minquartynoic acid

      Rasmussen, H. B., Christensen, Søren Brøgger, Kvist, L. P., Kharazmi, A. & Huansi, A. G., 2000, In: Journal of Natural Products. 63, 9, p. 1295-6 1 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    96. Published

      A simple and efficient separation of the curcumins, the antiprotozoal constituents of Curcuma longa

      Rasmussen, H. B., Christensen, Søren Brøgger, Kvist, L. P. & Karazmi, A., 22 Jun 2000, In: Planta Medica. 66, 4, p. 396-398 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    97. 2001
    98. Published

      Inhibition of fumarate reductase in Leishmania major and L. donovani by chalcones

      Chen, M., Zhai, L., Christensen, Søren Brøgger, Theander, Thor Grundtvig & Kharazmi, A., 2001, In: Antimicrobial Agents and Chemotherapy. 45, 7, p. 2023-9 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    99. Published

      Isolation of tow high-polar fractions from 'Banlangen', root of isatis tinctoria L. and its activity

      Qin, Q., He, H. P., Christensen, Søren Brøgger, Rasmussen, H. B., Kharazmi, A. & Chen, M., 1 Jan 2001, In: Chinese Pharmacological Bulletin. 17, 6, p. 714-715 2 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    100. 2002
    101. Published

      Hydrophilic carboxylic acids and iridoid glycosides in the juice of American and European cranberries (Vaccinium macrocarpon and V. oxycoccos), lingonberries (V. vitis-idaea), and blueberries (V. myrtillus)

      Jensen, H. D., Krogfelt, K. A., Cornett, Claus, Hansen, S. H. & Christensen, Søren Brøgger, 2002, In: Journal of Agricultural and Food Chemistry. 50, 23, p. 6871-4 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    102. Published

      Incorporation of the Cross Fire Beilstein database in the organic chemistry curriculum at the Royal Danish School of Pharmacy

      Christensen, Søren Brøgger, Franzyk, Henrik, Frølund, Bente, Jaroszewski, J. W., Stærk, Dan & Vedsø, P., 2002, In: Journal of Chemical Education. 79, p. 765-768

      Research output: Contribution to journalJournal articleResearch

    103. Published

      Incorporation of the crossfire Beilstein database into the organic chemistry curriculum at the Royal Danish School of Pharmacy

      Christensen, Søren Brøgger, Franzyk, Henrik, Frølund, Bente, Jaroszewski, J. W., Stærk, Dan & Vedsø, P., 1 Jun 2002, In: Journal of Chemical Education. 79, 6, 1 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    104. Published

      An antiplasmodial lignan from Euterpe precatoria

      Jensen, J. F., Kvist, L. P. & Christensen, Søren Brøgger, 1 Dec 2002, In: Journal of Natural Products. 65, 12, p. 1915-1917 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    105. 2003
    106. Published

      Ancistrotanzanine A, the first 5,3’-coupled naphtylisoquinoline alkaloid, and two further, 5,8’-linked related compounds from the newly described species Ancistrocladus tanzaniensis

      Bringmann, G., Dreyer, M., Faber, J. H., Dalsgaard, P. W., Stærk, Dan, Jaroszewski, J. W., Ndangalasi, H., Mbago, F., Brun, R., Reichert, M., Maksimenka, K. & Christensen, Søren Brøgger, 2003, In: Journal of Natural Products. 66, p. 1159-1165

      Research output: Contribution to journalJournal articleResearchpeer-review

    107. Published

      An antiinflammatory galactolipid from rose hip (Rosa canina) that inhibits chemotaxis of human peripheral blood neutrophils in vitro

      Larsen, Erik, Kharazmi, A., Christensen, L. P. & Christensen, Søren Brøgger, 1 Jul 2003, In: Journal of Natural Products. 66, 7, p. 994-995 2 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    108. Published

      Prostate-specific antigen-activated thapsigargin prodrug as targeted therapy for prostate cancer

      Denmeade, S. R., Jakobsen, C. M., Janssen, S., Khan, S. R., Garrett, E. S., Lilja, H., Christensen, Søren Brøgger & Isaacs, J. T., 2 Jul 2003, In: National Cancer Institute. Journal (Online). 95, 13, p. 990-1000 11 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    109. 2004
    110. Published

      Ancistrotanzanine C and related 5,1’- and 7,3’- coupled naphtylisoquinoline alkaloids from Ancistrocladus tanzaniensis

      Bringmann, G., Dreyer, M., Faber, J. H., Dalsgaard, P. W., Stærk, Dan, Jaroszewski, J. W., Ndangalasi, H., Mbago, F., Brun, R. & Christensen, Søren Brøgger, 2004, In: Journal of Natural Products. 67, p. 743-748

      Research output: Contribution to journalJournal articleResearchpeer-review

    111. Published

      The antiparasitic compound Licochalcon A is a potent echinocytogenic agent that modifies erythrocyte membrane in the concentration region where the antiplasmodial activity is observed

      Ziegler, H. L., Hansen, Harald S., Stærk, Dan, Christensen, Søren Brøgger, Hägerstrand, H. & Jaroszewski, J. W., 2004, In: Antimicrobial Agents and Chemotherapy. 48, p. 4067-4071

      Research output: Contribution to journalJournal articleResearchpeer-review

    112. Published

      Antiplasmodial Constituents of Cajanus cajan

      Duker-Eshun, G., Jaroszewski, J. W., Asomaning, W. A., Oppong-Boachie, F. & Christensen, Søren Brøgger, 1 Feb 2004, In: Phytotherapy Research. 18, 2, p. 128-130 3 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    113. Published

      Synthesis of the thapsigargins

      Ley, S. V., Antonello, A., Balskus, E. P., Booth, D. T., Christensen, Søren Brøgger, Cleator, E., Gold, H., Högenauer, K., Hünger, U., Myers, R. M., Oliver, S. F., Simic, O., Smith, M. D., Søhoel, H. & Woolford, A. J. A., 17 Aug 2004, In: Proceedings of the National Academy of Sciences of the United States of America. 101, 33, p. 12073-12078 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    114. Published

      Screening a combinatorial peptide library to develop a human glandular kallikrein 2-activated prodrug as targeted therapy for prostate cancer

      Janssen, S., Jakobsen, C. M., Rosen, D. M., Ricklis, R. M., Reineke, U., Christensen, Søren Brøgger, Lilja, H. & Denmeade, S. R., 1 Nov 2004, In: Molecular Cancer Therapeutics. 3, 11, p. 1439-1450 12 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    115. 2005
    116. Published

      Applying linear interaction energy method for rational design of noncompetitive allosteric inhibitors of the sarco- and endoplasmic reticulum calcium-ATPase

      Singh, P., Mhaka, A. M., Christensen, Søren Brøgger, Gray, J. J., Denmeade, S. R. & Isaacs, J. T., 21 Apr 2005, In: Journal of Medicinal Chemistry. 48, 8, p. 3005-3014 10 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    117. 2006
    118. Published

      Cytotoxic phenylpropanoids and an additional thapsigargin analogue isolated from Thapsia garganica

      Liu, Huizhen, Jensen, K. G., Tran, L. M., Chen, M., Zhai, L., Olsen, C. E., Søhoel, H., Denmeade, S. R., Issacs, J. T. & Christensen, Søren Brøgger, 2006, In: Phytochemistry. 67, 24, p. 2651-2658 8 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    119. Published

      Sesquiterpenes from Thapsia nitida var. meridionalis and Thapsia nitida var. nitida

      Rubal, J. J., Guerra, F. M., Moreno-Dorado, F. J., Jorge, Z. D., Massanet, G. M., Søhoel, H., Smitt, U. W., Frydenvang, Karla Andrea, Christensen, Søren Brøgger, Nielsen, C. & Eriksson, M., 2006, In: Journal of Natural Products. 69, 11, p. 1566-71 6 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    120. Published

      Pharmacokinetics, biodistribution, and antitumor efficacy of a human glandular kallikrein 2 (hK2)-activated thapsigargin prodrug

      Janssen, S., Rosen, D. M., Ricklis, R. M., Dionne, C. A., Lilja, H., Christensen, Søren Brøgger, Isaacs, J. T. & Denmeade, S. R., 1 Mar 2006, In: Prostate. 66, 4, p. 358-368 11 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    121. Published

      Identification and evaluation of Peruvian plants used to treat malaria and leishmaniasis

      Kvist, L. P., Christensen, Søren Brøgger, Rasmussen, H. B., Mejia, K. & Gonzalez, Ana Valeria, 19 Jul 2006, In: Journal of Ethnopharmacology. 106, 3, p. 390-402 13 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    122. Published

      Ancistrocladinium A and B, the first N,C-coupled naphthyldihydroisoquinoline alkaloids, from a Congolese Ancistrocladus species

      Bringmann, G., Kajahn, I., Reichert, M., Pedersen, S. E. H., Faber, J. H., Gulder, T., Brun, R., Christensen, Søren Brøgger, Ponte-Sucre, A., Moll, H., Heubl, G. & Mudogo, V., 8 Dec 2006, In: Journal of Organic Chemistry. 71, 25, p. 9348-9356 9 p.

      Research output: Contribution to journalJournal articleResearchpeer-review

    123. 2007
    124. Published

      Cytotoxic kurubasch aldehyde from Trichilia emetica

      Traore, M., Zhai, L., Chen, M., Olsen, C. E., Odile, N., Pierres, G. I., Bosco, O. J., Robert, G. T. & Christensen, Søren Brøgger, 2007, In: Natural Product Reports. 21, 1, p. 13-17

      Research output: Contribution to journalJournal articleResearchpeer-review

    125. Published

      Identification of natural products using HPLC-SPE combined with CapNMR

      Lambert, M., Wolfender, J., Stærk, Dan, Christensen, Søren Brøgger, Hostettmann, K. & Jaroszewski, J. W., 2007, In: Analytical Chemistry. 79, 2, p. 727-735

      Research output: Contribution to journalJournal articleResearchpeer-review

    126. Published

      Isolation and characterization of pristimerin as the antiplasmodial and antileishmanial agent of Maytenus senegalensis (Lam.) Exell.

      Khalid, S. A., Friedrichsen, G. M., Christensen, Søren Brøgger, El Tahir, A. & Satti, G. M., 2007, In: Arkivoc. ix, p. 129-134

      Research output: Contribution to journalJournal articleResearchpeer-review

    127. Published

      Noter til bioorganisk kemi M23-1

      Franzyk, Henrik, Christensen, Søren Brøgger & Jaroszewski, J. W., 2007, København: Københavns Universitet, Det Farmaceutiske Fakultet, Institut for Medicinalkemi.

      Research output: Book/ReportCompendium/lecture notesEducation

    128. Published

      Prenylated acetophenones from Melicope obscura and Melicope obtusifolia ssp. obtusifolia var. arborea and their distribution in Rutaceae

      Adsersen, A., Smitt, U. W., Simonsen, H. T., Christensen, Søren Brøgger & Jaroszewski, J. W., 2007, In: Biochemical Systematics and Ecology. 35, 7, p. 447-453

      Research output: Contribution to journalJournal articleResearchpeer-review

    129. Published

      Psychotropic constituents of Mentha aquatica L.

      van Staden, J., Stafford, G. I., Almqvist, J. P., Vangsøe, S. A. K., Olsen, H. T., Christensen, Søren Brøgger, Adsersen, A. & Jäger, A. K., 2007.

      Research output: Contribution to conferencePosterResearch

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