Vladimir Shalgunov

Vladimir Shalgunov

Guest Researcher


  1. Published

    F-18-Radiolabeling and in vivo evaluation of two diverse glycomimetics using PET

    Bratteby, K., Torkelsson, E., L'Estrade, E. T., Peterson, K., Shalgunov, Vladimir, Xiong, M., Leffer, H., Zetterberg, F., Ohlsson, T., Gillings, N., Nilsson, U., Herth, Matthias Manfred & Erlandsson, M., May 2019, p. S533-S534.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  2. Published

    Fragment-based labeling using condensation reactions of six potential 5-HT7R PET tracers

    Tampio L'Estrade, E., Shalgunov, Vladimir, Lehel, S., Nymann Petersen, I., Poulie, Christian Bernard Matthijs, Edgar, F. G., Volk, B., Ohlsson, T., Erlandsson, M., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2020, In: Journal of Radioanalytical and Nuclear Chemistry. 326, p. 1749-1762 14 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    High-throughput rat brain PET imaging and automatic spatial normalization of the dopamine D2/3 receptor ligand [F-18]fallypride

    Lange, D., Tejada, I. M., Xiong, M., Hillebrand, B., Noergaard, M., Baerentzen, S., Shalgunov, Vladimir, Herth, Matthias Manfred, Svarer, C. & Palner, M., 2019, In: Journal of Cerebral Blood Flow and Metabolism. 39, p. 588-589 2 p.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  4. Hunting for the high-affinity state of G-protein-coupled receptors with agonist tracers: Theoretical and practical considerations for positron emission tomography imaging

    Shalgunov, Vladimir, van Waarde, A., Booij, J., Michel, M. C., Dierckx, R. A. J. O. & Elsinga, P. H., May 2019, In: Medicinal Research Reviews. 39, 3, p. 1014-1052

    Research output: Contribution to journalReviewResearchpeer-review

  5. Published

    Improved radiosynthesis and preliminary in vivo evaluation of the 11 C-labeled tetrazine [ 11 C]AE-1 for pretargeted PET imaging

    Stéen, E. J. L., Jørgensen, Jesper Tranekjær, Petersen, I. N., Nørregaard, K., Lehel, S., Shalgunov, Vladimir, Birke, A., Edem, P. E., L'Estrade, E. T., Hansen, H. D., Villadsen, J., Erlandsson, M., Ohlsson, T., Yazdani, A., Valliant, J. F., Kristensen, Jesper Langgaard, Barz, M., Knudsen, Gitte Moos, Kjær, Andreas & Herth, Matthias Manfred, 1 Jan 2019, In: Bioorganic and Medicinal Chemistry Letters. 29, 8, p. 986-990

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    In Vivo Veritas - 18F-radiolabeled glycomimetics allow insights into the pharmacological fate of galectin-3 inhibitors

    Bratteby, K., Torkelsson, E., Tampio L'Estrade, E., Peterson, K., Shalgunov, Vladimir, Xiong, M., Leffler, H., Zetterberg, F., Olsson, T. G., Gillings, N., Nilsson, U. J., Herth, Matthias Manfred & Erlandsson, M., 2020, In: Journal of Medicinal Chemistry. 63, 2, p. 747-755

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Insights into Elution of Anion Exchange Cartridges: Opening the Path toward Aliphatic 18F-Radiolabeling of Base-Sensitive Tracers

    Bratteby, K., Shalgunov, Vladimir, Battisti, Umberto Maria, Petersen, I. N., Van Den Broek, S. L., Ohlsson, T., Gillings, N., Erlandsson, M. & Herth, Matthias Manfred, 2021, In: ACS Pharmacology and Translational Science. 4, 5, p. 1556–1566

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published
  9. Published

    Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry

    Steen, E. J. L., Jørgensen, Jesper Tranekjær, Denk, C., Battisti, Umberto Maria, Norregaard, K., Edem, P. E., Bratteby, K., Shalgunov, Vladimir, Wilkovitsch, M., Svatunek, D., Poulie, Christian Bernard Matthijs, Hvass, Lars, Simon, M., Wanek, T., Rossin, R., Robillard, M., Kristensen, Jesper Langgaard, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: ACS Pharmacology & Translational Science. 4, 2, p. 824-833 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Next generation fibroblast activation protein (FAP) targeting PET tracers : The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines

    Poulie, Christian Bernard Matthijs, Shalgunov, Vladimir, Elvas, F., Van Rymenant, Y., Moon, E. S., Battisti, Umberto Maria, De Loose, J., De Meester, I., Rösch, F., Van Der Veken, P. & Herth, Matthias Manfred, 2023, In: European Journal of Medicinal Chemistry. 262, 10 p., 115862.

    Research output: Contribution to journalJournal articleResearchpeer-review

ID: 185059116