Vladimir Shalgunov

Vladimir Shalgunov

Guest Researcher


  1. Published

    A SPECT-based method for dynamic imaging of the glymphatic system in rats

    Sigurdsson, B., Hauglund, Natalie Linea, Lilius, T. O., Mogensen, F. L. H., Mortensen, K. N., Beschorner, Natalie, Klinger, L., Bærentzen, S. L., Rosenholm, Marko, Shalgunov, Vladimir, Herth, Matthias Manfred, Mori, Yuki & Nedergaard, Maiken, 2023, In: Journal of Cerebral Blood Flow and Metabolism. 43, 7, 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    A facile synthesis of precursor for the σ-1 receptor PET radioligand [18F]FTC-146 and its radiofluorination

    Marešová, A., Jurášek, M., Drašar, P. B., Dolenský, B., Prokudina, E. A., Shalgunov, Vladimir, Herth, Matthias Manfred, Cumming, P. & Popkov, A., 2024, In: Journal of Labelled Compounds and Radiopharmaceuticals. 67, 2, p. 59-66

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    A pilot study of cerebral metabolism and serotonin 5-HT2A receptor occupancy in rats treated with the psychedelic tryptamine DMT in conjunction with the MAO inhibitor harmine

    Egger, K., Gudmundsen, F., Jessen, N. S., Baun, C., Poetzsch, S. N., Shalgunov, Vladimir, Herth, Matthias Manfred, Quednow, B. B., Martin-Soelch, C., Dornbierer, D., Scheidegger, M., Cumming, P. & Palner, M., 2023, In: Frontiers in Pharmacology. 14, 12 p., 1140656.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Aliphatic 18F-Radiofluorination: Recent Advances in the Labeling of Base-Sensitive Substrates**

    Bratteby, K., Shalgunov, Vladimir & Herth, Matthias Manfred, 2021, In: ChemMedChem. 16, 17, p. 2612-2622

    Research output: Contribution to journalReviewResearchpeer-review

  5. Published

    Bioorthogonal Click of Colloidal Gold Nanoparticles to Antibodies In vivo

    Poulie, Christian Bernard Matthijs, Sporer, E., Hvass, Lars, Jørgensen, Jesper Tranekjær, Kempen, Paul Joseph, Lopes van den Broek, S. I., Shalgunov, Vladimir, Kjær, Andreas, Jensen, A. I. & Herth, Matthias Manfred, 2022, In: Chemistry - A European Journal. 28, 61, 10 p., e202201847.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Blocking of efflux transporters in rats improves translational validation of brain radioligands

    Shalgunov, Vladimir, Xiong, M., L’Estrade, E. T., Raval, N. R., Andersen, Ida Vang, Edgar, F. G., Speth, N. R., Baerentzen, S. L., Hansen, H. D., Donovan, L. L., Nasser, A., Peitersen, S. T., Kjær, Andreas, Knudsen, Gitte Moos, Syvänen, S., Palner, M. & Herth, Matthias Manfred, 2020, In: EJNMMI Research. 10, 1, 11 p., 124.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Convenient Entry to 18 F-Labeled Amines through the Staudinger Reduction

    Stéen, E. J. L., Shalgunov, Vladimir, Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, 2019, In: European Journal of Organic Chemistry. 2019, 8, p. 1722-1725

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Convenient access to F-18-labeled amines through the Staudinger reduction

    Shalgunov, Vladimir, Steen, J., Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, May 2019, In: Journal of Labelled Compounds and Radiopharmaceuticals. 62, Supl. 1/SI, p. S205-S206 P-050.

    Research output: Contribution to journalConference abstract in journalResearch

  9. Published

    Cover Feature: Convenient Entry to 18 F-Labeled Amines through the Staudinger Reduction (Eur. J. Org. Chem. 8/2019)

    Stéen, E. J. L., Shalgunov, Vladimir, Denk, C., Mikula, H., Kjær, Andreas, Kristensen, Jesper Langgaard & Herth, Matthias Manfred, 28 Feb 2019, In: European Journal of Organic Chemistry. 2019, 8, p. 1686-1686

    Research output: Contribution to journalJournal articleCommunication

  10. Published

    Development and Evaluation of Two Potential 5-HT7 Receptor PET Tracers: [18F]ENL09 and [18F]ENL10

    Tampio L'Estrade, E., Xiong, M., Shalgunov, Vladimir, Edgar, F. G., Volk, B., Baerentzen, S. L., Palner, M., Erlandsson, M., Ohlsson, T., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2019, In: ACS Chemical Neuroscience. 10, 9, p. 3961-3968 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Development and evaluation of an 18F-labeled nanobody to target SARS-CoV-2's spike protein

    Lopes van den Broek, S., García-Vázquez, R., Andersen, Ida Vang, Valenzuela-Nieto, G., Shalgunov, Vladimir, Battisti, Umberto Maria, Schwefel, D., Modhiran, N., Kramer, V., Cheuquemilla, Y., Jara, R., Salinas-Varas, C., Amarilla, A. A., Watterson, D., Rojas-Fernandez, A. & Herth, Matthias Manfred, 2022, In: Frontiers in Nuclear Medicine. 2, 1033697.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Development of 11C-labeled CRANAD-102 for positron emission tomography imaging of soluble Aβ-species

    Staudt, Markus, Shalgunov, Vladimir, Nedergaard, Maiken & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 12, p. 393-399

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Development of Trans-Cyclooctene Modified Antibodies for Pretargeted Imaging within the Central Nervous System: [Meeting Abstract]

    van den Broek, S. L., Shalgunov, Vladimir, Sehlin, D., Syvanen, S. & Herth, Matthias Manfred, 2020, In: Journal of Nuclear Medicine. 61, Supl. 1, 3 p., 196.

    Research output: Contribution to journalConference abstract in journalResearch

  14. Published

    Development of the First Aliphatic 18F-Labeled Tetrazine Suitable for Pretargeted PET Imaging-Expanding the Bioorthogonal Tool Box

    Battisti, Umberto Maria, Bratteby, K., Jørgensen, Jesper Tranekjær, Hvass, Lars, Shalgunov, Vladimir, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Journal of Medicinal Chemistry. 64, 20, p. 15297–15312

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Development of the First Tritiated Tetrazine: Facilitating Tritiation of Proteins

    Radjani Bidesi, N. S., Battisti, Umberto Maria, Lopes van de Broek, S., Shalgunov, Vladimir, Dall, A., Bøggild Kristensen, J., Sehlin, D., Syvänen, S., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2022, In: ChemBioChem. 23, 23, 7 p., e202200539.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Development of18F-Labeled Bispyridyl Tetrazines for In Vivo Pretargeted PET Imaging

    García-Vázquez, R., Jørgensen, Jesper Tranekjær, Bratteby, K. E., Shalgunov, Vladimir, Hvass, Lars, Herth, Matthias Manfred, Kjær, Andreas & Battisti, Umberto Maria, 2022, In: Pharmaceuticals. 15, 2, 28 p., 245.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Direct Cu-mediated aromatic18F-labeling of highly reactive tetrazines for pretargeted bioorthogonal PET imaging

    García-Vázquez, R., Battisti, Umberto Maria, Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Hvass, Lars, Stares, D. L., Petersen, I. N., Crestey, F., Löffler, A., Svatunek, D., Kristensen, Jesper Langgaard, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Chemical Science. 12, 35, p. 11668-11675

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Evaluation of F-537-Tetrazine in a model for brain pretargeting imaging. Comparison to N-(3-[18F] fluoro-5-(1,2,4,5-tetrazin-3-yl)benzyl)propan-1-amine

    Shalgunov, Vladimir, van den Broek, S. L., Andersen, Ida Vang, Raval, N. R., Schäfer, G., Barz, M., Herth, Matthias Manfred & Battisti, Umberto Maria, 2024, In: Nuclear Medicine and Biology. 128-129, 12 p., 108877.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Evaluation of [Cu-64]Cu-NOTA-PEG7-H-Tz for Pretargeted Imaging in LS174T Xenografts-Comparison to [111In-111]In-DOTA-PEG11-BisPy-Tz

    Poulie, Christian Bernard Matthijs, Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Kougioumtzoglou, G., Jeppesen, T. E., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Molecules. 26, 3, 9 p., 544.

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Evaluation of the α-synuclein PET radiotracer (d3)-[11C]MODAG-001 in pigs

    Raval, N. R., Madsen, C. A., Shalgunov, Vladimir, Nasser, A., Battisti, Umberto Maria, Beaman, Emily Eufaula, Juhl, M., Jørgensen, Louise Møller, Herth, Matthias Manfred, Hansen, H. D., Plavén-Sigray, P. & Knudsen, Gitte Moos, 2022, In: Nuclear Medicine and Biology. 114-115, p. 42-48

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    F-18-Radiolabeling and in vivo evaluation of two diverse glycomimetics using PET

    Bratteby, K., Torkelsson, E., L'Estrade, E. T., Peterson, K., Shalgunov, Vladimir, Xiong, M., Leffer, H., Zetterberg, F., Ohlsson, T., Gillings, N., Nilsson, U., Herth, Matthias Manfred & Erlandsson, M., May 2019, p. S533-S534.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  22. Published

    Fragment-based labeling using condensation reactions of six potential 5-HT7R PET tracers

    Tampio L'Estrade, E., Shalgunov, Vladimir, Lehel, S., Nymann Petersen, I., Poulie, Christian Bernard Matthijs, Edgar, F. G., Volk, B., Ohlsson, T., Erlandsson, M., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2020, In: Journal of Radioanalytical and Nuclear Chemistry. 326, p. 1749-1762 14 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    High-throughput rat brain PET imaging and automatic spatial normalization of the dopamine D2/3 receptor ligand [F-18]fallypride

    Lange, D., Tejada, I. M., Xiong, M., Hillebrand, B., Noergaard, M., Baerentzen, S., Shalgunov, Vladimir, Herth, Matthias Manfred, Svarer, C. & Palner, M., 2019, In: Journal of Cerebral Blood Flow and Metabolism. 39, p. 588-589 2 p.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  24. Hunting for the high-affinity state of G-protein-coupled receptors with agonist tracers: Theoretical and practical considerations for positron emission tomography imaging

    Shalgunov, Vladimir, van Waarde, A., Booij, J., Michel, M. C., Dierckx, R. A. J. O. & Elsinga, P. H., May 2019, In: Medicinal Research Reviews. 39, 3, p. 1014-1052

    Research output: Contribution to journalReviewResearchpeer-review

  25. Published

    Improved radiosynthesis and preliminary in vivo evaluation of the 11 C-labeled tetrazine [ 11 C]AE-1 for pretargeted PET imaging

    Stéen, E. J. L., Jørgensen, Jesper Tranekjær, Petersen, I. N., Nørregaard, K., Lehel, S., Shalgunov, Vladimir, Birke, A., Edem, P. E., L'Estrade, E. T., Hansen, H. D., Villadsen, J., Erlandsson, M., Ohlsson, T., Yazdani, A., Valliant, J. F., Kristensen, Jesper Langgaard, Barz, M., Knudsen, Gitte Moos, Kjær, Andreas & Herth, Matthias Manfred, 1 Jan 2019, In: Bioorganic and Medicinal Chemistry Letters. 29, 8, p. 986-990

    Research output: Contribution to journalJournal articleResearchpeer-review

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ID: 185059116