Kristian Strømgaard
Professor
Biopharmaceuticals
Jagtvej 162
2100 København Ø
- Published
Energetic pathway sampling in a protein interaction domain
Hultqvist, G., Haq, S. R., Punekar, A. S., Chi, C. N., Engström, A., Bach, Anders, Strømgaard, Kristian, Selmer, M., Gianni, S. & Jemth, P., 25 Jun 2013, In: Structure. 21, 7, p. 1193-1202Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Evaluation of PhTX-74 as Subtype-Selective Inhibitor of GluA2-Containing AMPA Receptors
Poulsen, Mette Homann, Lucas, S., Strømgaard, Kristian & Kristensen, Anders Skov, Feb 2014, In: Molecular Pharmacology. 85, 2, p. 261-268 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Expedient synthesis of 1,3-substituted benzene peptidomimetics
Bach, Anders & Strømgaard, Kristian, 8 Feb 2011, In: Synthesis. 2011, 5, p. 807-815Research output: Contribution to journal › Journal article › Research › peer-review
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Expressed protein ligation of ionotropic glutamate receptors
Jensen, M. S., Kristensen, Anders Skov & Strømgaard, Kristian, 2007, In: Biopolymers. 88, 4, p. 602Research output: Contribution to journal › Conference abstract in journal › Research
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Facile synthesis of α-hydroxy carboxylic acids from the corresponding α-amino acids
Stuhr-Hansen, N., Padrah, S. & Strømgaard, Kristian, 2014, In: Tetrahedron Letters. 55, 30, p. 4149-4151 3 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Facilitating the structural characterisation of non-canonical amino acids in biomolecular NMR
Kuschert, S., Stroet, M., Chin, Y. K. Y., Conibear, A. C., Jia, X., Lee, T., Bartling, Christian Reinhard Otto, Strømgaard, Kristian, Güntert, P., Rosengren, K. J., Mark, A. E. & Mobli, M., 2023, In: Magnetic Resonance. 4, 1, p. 57-72Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Fatty acid derivatives of dimeric inhibitors of PSD-95
Strømgaard, Kristian, Bach, Anders & Nissen, K. B., 4 Jun 2015, IPC No. A61K38/17 , Patent No. WO2015/078477A1, Priority date 1 Dec 2013, Priority No. DK/2013/70735Research output: Patent
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From the selective serotonin transporter inhibitor citalopram to the selective norepinephrine transporter inhibitor talopram: Synthesis and structure-activity relationship studies
Eildal, J. N. N., Andersen, J., Kristensen, Anders Skov, Jørgensen, A. M., Bang-Andersen, B., Jørgensen, M. & Strømgaard, Kristian, 2008, In: Journal of Medicinal Chemistry. 51, 10, p. 3045-3048Research output: Contribution to journal › Journal article › Research › peer-review
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GLP-1-directed NMDA receptor antagonism for obesity treatment
Petersen, J., Ludwig, M. Q., Juozaityte, V., Ranea-Robles, P., Svendsen, C., Hwang, E., Kristensen, A. W., Fadahunsi, N., Lund, J., Breum, A. W., Mathiesen, C. V., Sachs, L., Moreno-Justicia, R., Rohlfs, R., Ford, J. C., Douros, J. D., Finan, B., Portillo, B., Grose, K., Petersen, J. E. & 13 others, , 2024, In: Nature. 629, 8014, p. 1133–1141Research output: Contribution to journal › Journal article › Research › peer-review
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General synthesis of β-alanine-containing spider polyamine toxins and discovery of nephila polyamine toxins 1 and 8 as highly potent inhibitors of ionotropic glutamate receptors
Lucas, S., Poulsen, Mette Homann, Nørager, N. G., Barslund, A. F., Bach, T. B., Kristensen, Anders Skov & Strømgaard, Kristian, 26 Nov 2012, In: Journal of Medicinal Chemistry. 55, 22, p. 10297-10301 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Genetically encoded photocrosslinkers locate the high-affinity binding site of antidepressant drugs in the human serotonin transporter
Rannversson, H., Andersen, J., Hall, L. S., Bang-Andersen, B., Park, M., Huber, T., Sakmar, T. P. & Strømgaard, Kristian, 19 Apr 2016, In: Nature Communications. 7, p. 1-9 9 p., 11261.Research output: Contribution to journal › Journal article › Research › peer-review
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Gephyrin-binding peptides visualize postsynaptic sites and modulate neurotransmission
Maric, H. M., Hausrat, T. J., Neubert, F., Dalby, N. O., Doose, S., Sauer, M., Kneussel, M. & Strømgaard, Kristian, 2017, In: Nature Chemical Biology. 13, p. 153-160 11 p., 2246.Research output: Contribution to journal › Journal article › Research › peer-review
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Giftstoffer fra hvepse og edderkopper i forskning og lægemiddeludvikling
Strømgaard, Kristian, 2008, In: Carlsbergfondet. Aarsskrift. p. 42-47Research output: Contribution to journal › Journal article › Communication
Ginkgolide derivatives for photolabeling studies: preparation and pharmacological evaluation
Strømgaard, Kristian, Saito, D. R., Shindou, H., Ishii, S., Shimizu, T. & Nakanishi, K., 29 Aug 2002, In: Journal of Medicinal Chemistry. 45, 18, p. 4038-4046 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
Ginkgolides: selective acetylations, translactonization, and biological evaluation
Jaracz, S., Strømgaard, Kristian & Nakanishi, K., 28 Jun 2002, In: Journal of Organic Chemistry. 67, 13, p. 4623-4626 4 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Ginkgolides and glycine receptors: a structure-activity relationship study
Jaracz, S., Nakanishi, K., Jensen, Anders A. & Strømgaard, Kristian, 2004, In: Chemistry: A European Journal. 10, 6, p. 1507-18 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Heparin promotes fibrillation of most phenol-soluble modulin virulence peptides from Staphylococcus aureus
Najarzadeh, Z., Zaman, M., Sereikaité, Vita, Strømgaard, Kristian, Andreasen, M. & Otzen, D. E., 2021, In: Journal of Biological Chemistry. 297, 2, 14 p., 100953.Research output: Contribution to journal › Journal article › Research › peer-review
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Heterotrimeric G Proteins as Therapeutic Targets in Drug Discovery
Li, J., Ge, Y., Huang, J., Strømgaard, Kristian, Zhang, X. & Xiong, X., 2020, In: Journal of Medicinal Chemistry. 63, 10, p. 5013-5030 18 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Submitted
High-affinity, dimeric inhibitors of PSD-95 as efficient neuroprotectants against ischemic brain damage and for treatment of pain
Bach, Anders & Strømgaard, Kristian, 2012, (Submitted) Patent No. WO2012/156308 (Granted: EP2707014B1; US9139615B2)Research output: Patent
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Human Fibrinogen Inhibits Amyloid Assembly of Most Phenol-Soluble Modulins from Staphylococcus aureus
Najarzadeh, Z., Nielsen, J., Farzadfard, A., Sereikaité, Vita, Strømgaard, Kristian, Meyer, R. L. & Otzen, D. E., 2021, In: ACS Omega. 6, 34, p. 21960-21970Research output: Contribution to journal › Journal article › Research › peer-review
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Identification and characterization of a small-molecule inhibitor of death-associated protein kinase 1
Wilbek, T. S., Skovgaard, T., Sorrell, F. J., Knapp, S., Berthelsen, J. & Strømgaard, Kristian, 2 Jan 2015, In: ChemBioChem. 16, 1, p. 59-63 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Identification of GDF15 peptide fragments inhibiting GFRAL receptor signaling
Alexopoulou, Flora, Buch-Månson, N., Pedersen, S. L., Vrang, N., Fink, L. N. & Strømgaard, Kristian, 2023, In: Peptides. 168, 7 p., 171063.Research output: Contribution to journal › Journal article › Research › peer-review
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Identification of a small-molecule inhibitor of the PICK1 PDZ domain that inhibits hippocampal LTP and LTD
Thorsen, T. S., Madsen, Kenneth Lindegaard, Rebola, N., Rathje, Mette, Anggono, V., Bach, Anders, Moreira, I. S., Stuhr-Hansen, N., Dyhring, T., Peters, D., Beuming, T., Huganir, R., Weinstein, H., Mulle, C., Strømgaard, Kristian, Rønn, L. C. B. & Gether, Ulrik, 2010, In: Proceedings of the National Academy of Science of the United States of America. 107, 1, p. 413-8 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Importance of a Conserved Lys/Arg Residue for Ligand/PDZ Domain Interactions as Examined by Protein Semisynthesis
Pedersen, S. W., Moran, G. E., Sereikaité, Vita, Kedström, L. M. H. & Strømgaard, Kristian, 17 Oct 2016, In: ChemBioChem. 17, 20, p. 1936-1944 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Importance of the Extracellular Loop 4 in the Human Serotonin Transporter for Inhibitor Binding and Substrate Translocation
Rannversson, H., Wilson, P., Kristensen, K. B., Sinning, S., Kristensen, Anders Skov, Strømgaard, Kristian & Andersen, J., 5 Jun 2015, In: The Journal of Biological Chemistry. 290, 23, p. 14582-94 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1302559
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PDZ domain-mediated interactions of G protein-coupled receptors with postsynaptic density protein 95: quantitative characterization of interactions
Research output: Contribution to journal › Journal article › Research › peer-review
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