Umberto Maria Battisti
Assistant Professor
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- 2024
- Published
Evaluation of F-537-Tetrazine in a model for brain pretargeting imaging. Comparison to N-(3-[18F] fluoro-5-(1,2,4,5-tetrazin-3-yl)benzyl)propan-1-amine
Shalgunov, Vladimir, van den Broek, S. L., Andersen, Ida Vang, Raval, N. R., Schäfer, G., Barz, M., Herth, Matthias Manfred & Battisti, Umberto Maria, 2024, In: Nuclear Medicine and Biology. 128-129, 12 p., 108877.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
Schlein, E., Rokka, J., Odell, L. R., van den Broek, S. L., Herth, Matthias Manfred, Battisti, Umberto Maria, Syvänen, S., Sehlin, D. & Eriksson, J., 2024, In: EJNMMI Radiopharmacy and Chemistry. 9, 1, 12 p., 21.Research output: Contribution to journal › Journal article › Research › peer-review
- 2023
- Published
A Fluorescent Probe as a Lead Compound for a Selective α-Synuclein PET Tracer: Development of a Library of 2-Styrylbenzothiazoles and Biological Evaluation of [18F]PFSB and [18F]MFSB
Di Nanni, A., Saw, R. S., Battisti, Umberto Maria, Bowden, G. D., Boeckermann, A., Bjerregaard-Andersen, K., Pichler, B. J., Herfert, K., Herth, Matthias Manfred & Maurer, A., 2023, In: ACS Omega. 8, 34, p. 31450–31467Research output: Contribution to journal › Journal article › Research › peer-review
- Accepted/In press
Labeling of highly reactive tetrazines using [ 18F]SuFEx
Battisti, Umberto Maria, Müller, Marius, García-Vázquez, R. & Herth, Matthias Manfred, 2023, (Accepted/In press) In: Synlett.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Next generation fibroblast activation protein (FAP) targeting PET tracers : The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines
Poulie, Christian Bernard Matthijs, Shalgunov, Vladimir, Elvas, F., Van Rymenant, Y., Moon, E. S., Battisti, Umberto Maria, De Loose, J., De Meester, I., Rösch, F., Van Der Veken, P. & Herth, Matthias Manfred, 2023, In: European Journal of Medicinal Chemistry. 262, 10 p., 115862.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and in vivo evaluation of [11C]tucatinib for HER2-targeted PET imaging
Müller, Marius, Shalgunov, Vladimir, Hvass, Lars, Jørgensen, Jesper Tranekjær, Kramer, V., Staudt, Markus, Battisti, Umberto Maria, Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Bioorganic and Medicinal Chemistry Letters. 80, 5 p., 129088.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and radiolabeling of a polar [125 I]I-1,2,4,5-tetrazine
Bidesi, N., Shalgunov, Vladimir, Battisti, Umberto Maria, Hvass, Lars, Jørgensen, Jesper Tranekjær, Poulie, Christian Bernard Matthijs, Jensen, A. I., Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 1, p. 22-30Research output: Contribution to journal › Journal article › Research › peer-review
- 2022
- Published
Benzothiadiazines derivatives as novel allosteric modulators of kainic acid receptors
Puja, G., Ravazzini, F., Losi, G., Bardoni, R., Battisti, Umberto Maria, Citti, C. & Cannazza, G., 2022, In: Journal of Physiology and Pharmacology. 73, 1, p. 19-28Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development and evaluation of an 18F-labeled nanobody to target SARS-CoV-2's spike protein
Lopes van den Broek, S., García-Vázquez, R., Andersen, Ida Vang, Valenzuela-Nieto, G., Shalgunov, Vladimir, Battisti, Umberto Maria, Schwefel, D., Modhiran, N., Kramer, V., Cheuquemilla, Y., Jara, R., Salinas-Varas, C., Amarilla, A. A., Watterson, D., Rojas-Fernandez, A. & Herth, Matthias Manfred, 2022, In: Frontiers in Nuclear Medicine. 2, 1033697.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of the First Tritiated Tetrazine: Facilitating Tritiation of Proteins
Radjani Bidesi, N. S., Battisti, Umberto Maria, Lopes van de Broek, S., Shalgunov, Vladimir, Dall, A., Bøggild Kristensen, J., Sehlin, D., Syvänen, S., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2022, In: ChemBioChem. 23, 23, 7 p., e202200539.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 210553848
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Development of18F-Labeled Bispyridyl Tetrazines for In Vivo Pretargeted PET Imaging
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
55
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Direct Cu-mediated aromatic18F-labeling of highly reactive tetrazines for pretargeted bioorthogonal PET imaging
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
36
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Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry
Research output: Contribution to journal › Journal article › Research › peer-review
Published