Christian Adam Olsen

Christian Adam Olsen

Professor


  1. Published

    Selectively N-protected enantiopure 2,5-disubstituted piperazines: Avoiding the pitfalls in solid-phase Fukuyama-Mitsunobu cyclizations

    Ottesen, L. K., Olsen, Christian Adam, Witt, M., Jaroszewski, J. W. & Franzyk, Henrik, 2009, In: Chemistry: A European Journal. 15, 12, p. 2966-2978

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Effect of co-inhabiting coagulase negative staphylococci on S. Aureus agr quorum sensing, host factor binding, and biofilm formation

    Peng, P., Baldry, M., Gless, B. H., Bojer, Martin Saxtorph, Espinosa-Gongora, C., Baig, S. J., Andersen, P. S., Olsen, Christian Adam & Ingmer, Hanne, 2019, In: Frontiers in Microbiology. 10, SEP, 14 p., 2212.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Modular total synthesis of lamellarin D

    Pla, D., Marchal, A., Olsen, Christian Adam, Albericio, F. & Álvarez, M., 20 Sep 2005, In: Journal of Organic Chemistry. 70, 20, p. 8231-8234 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Synthesis and structure-activity relationship study of potent cytotoxic analogues of the marine alkaloid lamellarin D

    Pla, D., Marchal, A., Olsen, Christian Adam, Francesch, A., Cuevas, C., Albericio, F. & Alvarez, M., 1 Jun 2006, In: Journal of Medicinal Chemistry. 49, 11, p. 3257-3268 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Mechanism-based Inhibitors of the Human Sirtuin 5 Deacylase: Structure-Activity Relationship, Biostructural, and Kinetic Insight

    Rajabi, N., Auth, M., Troelsen, K. R., Pannek, M., Bhatt, D., Fontenas, M., Hirschey, M., Steegborn, C., Madsen, A. S. & Olsen, Christian Adam, 20 Nov 2017, In: Angewandte Chemie, Int. Ed.. 56, 47, p. 14836-14841

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Targeting Sirtuins: Substrate Specificity and Inhibitor Design

    Rajabi, N., Galleano, I., Madsen, A. S. & Olsen, Christian Adam, 3 Feb 2018, Progress in Molecular Biology and Translational Science: Sirtuins in Health and Disease. Elsevier, p. 25-69 (Progress in Molecular Biology and Translational Science, Vol. 154).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  7. Published

    Investigation of Carboxylic Acid Isosteres and Prodrugs for Inhibition of the Human SIRT5 Lysine Deacylase Enzyme**

    Rajabi, N., Hansen, T. N., Nielsen, A. L., Nguyen, H. T., Bæk, M., Bolding, J. E., Bahlke, O., Petersen, S. E. G., Bartling, Christian Reinhard Otto, Strømgaard, Kristian & Olsen, Christian Adam, 2022, In: Angewandte Chemie - International Edition. 61, 22, 9 p., e202115805.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Dethioacylation by sirtuins 1–3: Considerations for drug design using mechanism-based sirtuin inhibition

    Rajabi, N., Nielsen, A. L. & Olsen, Christian Adam, 2020, In: A C S Medicinal Chemistry Letters. 11, 10, p. 1886-1892

    Research output: Contribution to journalLetterResearchpeer-review

  9. Published

    A Robust Proton Flux (pHlux) Assay for Studying the Function and Inhibition of the Influenza A M2 Proton Channel

    Santner, P., Martins, J. M. D. S., Laursen, J. S., Behrendt, L., Riber, Leise, Olsen, Christian Adam, Arkin, I. T., Winther, Jakob R., Willemoës, Martin & Lindorff-Larsen, Kresten, 2018, In: Biochemistry. 57, 41, p. 5949-5956

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Random mutagenesis analysis of the Influenza A M2 proton channel reveals novel resistance mutants

    Santner, P., Martins, J. M. D. S., Kampmeyer, Caroline, Hartmann-Petersen, Rasmus, Laursen, J. S., Stein, Amelie, Olsen, Christian Adam, Arkin, I. T., Winther, Jakob R., Willemoës, Martin & Lindorff-Larsen, Kresten, 2018, In: Biochemistry. 57, 41, p. 5957-5968

    Research output: Contribution to journalJournal articleResearchpeer-review

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