Jesper Langgaard Kristensen
Professor
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- 2012
- Published
Total synthesis of ascididemin via anionic cascade ring closure
Petersen, I. N., Crestey, F. & Kristensen, Jesper Langgaard, 2012, In: Chemical Communications. 48, 72, p. 9092-9094Research output: Contribution to journal › Journal article › Research › peer-review
- 2011
- Published
Targeting histone lysine demethylases by truncating the histone 3 tail to obtain selective substrate-based inhibitors
Lohse, B., Nielsen, A. L., Kristensen, J. B. L., Helgstrand, C., Cloos, P. A. C., Olsen, L., Gajhede, Michael, Clausen, Rasmus Prætorius & Kristensen, Jesper Langgaard, 19 Sep 2011, In: Angewandte Chemie International Edition. 50, 39, p. 9100-9103Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of N-alkylated amino acids using fluorous-tagged hydroxylamines
Nielsen, S. D., Smith, G. P., Begtrup, M. & Kristensen, Jesper Langgaard, 22 Jul 2011, In: Tetrahedron. 67, 29, p. 5261-5267Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Enzyme kinetic studies of histone demethylases KDM4C and KDM6A: Towards understanding selectivity of inhibitors targeting oncogenic histone demethylases
Kristensen, J. B. L., Nielsen, A. L., Jørgensen, L., Kristensen, L. H., Helgstrand, C., Juknaite, L., Kristensen, Jesper Langgaard, Kastrup, Jette Sandholm Jensen, Clausen, Rasmus Prætorius, Olsen, L. & Gajhede, Michael, 23 Jun 2011, In: F E B S Letters. 585, 12, p. 1951-1956Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Radiosynthesis and in vivo evaluation of a series of substituted 11C-phenethylamines as 5-HT2A agonist PET tracers
Ettrup, A., Hansen, M., Santini, M. A., Paine, J. S., Gillings, N., Palner, M., Lehel, S., Herth, Matthias Manfred, Madsen, J., Kristensen, Jesper Langgaard, Begtrup, M. & Knudsen, Gitte Moos, 1 Apr 2011, In: European Journal of Nuclear Medicine and Molecular Imaging. 38, 4, p. 681-693Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Inhibitors of histone demethylases
Lohse, B., Kristensen, Jesper Langgaard, Kristensen, L. H., Agger, K., Helin, K., Gajhede, Michael & Clausen, Rasmus Prætorius, 1 Feb 2011, In: Bioorganic & Medicinal Chemistry. 19, 12, p. 3625-3636 11 p.Research output: Contribution to journal › Review › Research › peer-review
- Published
Development of New PET Radiotracers for In Vivo 5-HT7 Brain Imaging
Herth, Matthias Manfred, Hansen, H., Lehel, S., Ettrup, A., Paine, J., Madsen, J., Gillings, N., Kristensen, Jesper Langgaard & Knudsen, G., 2011, In: Journal of Labelled Compounds and Radiopharmaceuticals. 54, p. S277-S277Research output: Contribution to journal › Journal article › Research › peer-review
- 2010
- Published
Erratum: Aminolysis of resin-bound N-nosylaziridine-2-carboxylic acids (Organic Letters (2006) 8 (3371))
Olsen, Christian Adam, Christensen, C., Nielsen, Birgitte, Farah, M. M., Witt, M., Clausen, Rasmus Prætorius, Kristensen, Jesper Langgaard, Franzyk, Henrik & Jaroszewski, J. W., 15 Oct 2010, In: Organic Letters. 12, 20, p. 4708 1 p.Research output: Contribution to journal › Comment/debate › Research › peer-review
- Published
Amination of aryl iodides using a fluorous-tagged ammonia equivalent
Nielsen, S. D., Smith, G., Begtrup, M. & Kristensen, Jesper Langgaard, 2010, In: European Journal of Organic Chemistry. 2010, 19, p. 3704-3710Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Exploring the neuroleptic substituent in octoclothepin: potential ligands for positron emission tomography with subnanomolar affinity for alpha1-adrenoceptors
Kristensen, Jesper Langgaard, Pu¨schl, A., Jensen, M., Risgaard, R., Christoffersen, C. T., Bang-Andersen, B. & Balle, T., 2010, In: Journal of Medicinal Chemistry. 53, 19, p. 7021-7034Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Novel 4-(piperidin-4-yl)-1-hydroxypyrazoles as gamma-aminobutyric acidA receptor ligands: synthesis, pharmacology, and structure-activity relationships
Møller, H. A., Sander, T., Kristensen, Jesper Langgaard, Nielsen, Birgitte, Krall, J., Bergmann, M. L., Christiansen, B., Balle, T., Jensen, Anders A. & Frølund, Bente, 2010, In: Journal of Medicinal Chemistry. 53, 8, p. 3417-3421Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Ring opening of pymisyl-protected aziridines with organocuprates
Bornholdt, J., Felding, J., Clausen, Rasmus Prætorius & Kristensen, Jesper Langgaard, 2010, In: Chemistry: A European Journal. 16, 41, p. 12474-12480Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and application of a new fluorous-tagged ammonia equivalent
Nielsen, S. D., Smith, G., Begtrup, M. & Kristensen, Jesper Langgaard, 2010, In: Chemistry: A European Journal. 16, 15, p. 4557-4566Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of enantiopure 3-substituted morpholines
Bornholdt, J., Felding, J. & Kristensen, Jesper Langgaard, 2010, In: Journal of Organic Chemistry. 75, 21, p. 7454-7457Research output: Contribution to journal › Journal article › Research › peer-review
- 2009
- Published
Heterocyclic pentafluorophenyl sulfonate esters as shelf stable alternatives to sulfonyl chlorides
Bornholdt, J., Fjære, K. W., Felding, J. & Kristensen, Jesper Langgaard, 2009, In: Tetrahedron. 65, 45, p. 9280-9284Research output: Contribution to journal › Journal article › Research › peer-review
- 2008
- Published
N-Hydroxypyrazolyl glycine derivatives as selective N-methyl-D-aspartic acid receptor ligands
Clausen, Rasmus Prætorius, Christensen, C., Hansen, K. B., Greenwood, J. R., Jørgensen, L., Micale, N., Madsen, J. C., Nielsen, Birgitte, Egebjerg, J., Bräuner, Hans, Traynelis, S. F. & Kristensen, Jesper Langgaard, 2008, In: Journal of Medicinal Chemistry. 51, 14, p. 4179-87Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of RHPS4 via an anionic ring closing cascade
Kristensen, Jesper Langgaard, 2008, In: Tetrahedron Letters. 49, 15, p. 2351-2354Research output: Contribution to journal › Journal article › Research › peer-review
- 2006
- Published
Synthesis, cross-coupling, and anionic cyclization of ortho-substituted naphthaleneboronic esters
Lysén, M., Madden, M., Kristensen, Jesper Langgaard, Vedsø, P., Zöllner, C. & Begtrup, M., 17 Oct 2006, In: Synthesis. 20, p. 3478-3484 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of substituted 2-cyanoarylboronic esters
Lysén, M., Hansen, H. M., Begtrup, M. & Kristensen, Jesper Langgaard, 17 Mar 2006, In: Journal of Organic Chemistry. 71, 6, p. 2518-20 3 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Aminolysis of resin-bound N-nosylaziridine-2-carboxylic acids
Olsen, Christian Adam, Christensen, C., Nielsen, Birgitte, Farah, M. M., Mohamed, F. M., Witt, M., Clausen, Rasmus Prætorius, Kristensen, Jesper Langgaard, Franzyk, Henrik & Jaroszewski, J. W., 2006, In: Organic Letters. 8, 15, p. 3371-4 4 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2005
- Published
Tweaking agonist efficacy at N-methyl-D-aspartate receptors by site-directed mutagenesis
Hansen, K. B., Clausen, Rasmus Prætorius, Bjerrum, E. J., Bechmann, C., Greenwood, J. R., Christensen, C., Kristensen, Jesper Langgaard, Egebjerg, J. & Bräuner, Hans, Dec 2005, In: Molecular Pharmacology. 68, 6, p. 1510-23Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and binding studies of 2-arylapomorphines
Søndergaard, K., Kristensen, Jesper Langgaard, Palner, M., Gillings, N., Knudsen, Gitte Moos, Roth, B. & Begtrup, M., 21 Nov 2005, In: Organic & Biomolecular Chemistry. 3, 22, p. 4077-4081 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of azaphenanthridines via anionic ring closure
Hansen, H. M., Lysén, M., Begtrup, M. & Kristensen, Jesper Langgaard, 17 Oct 2005, In: Tetrahedron. 61, 42, p. 9955-9960 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of (R)-(-)-2-fluoronorapomorphine - A precursor for the synthesis of (R)-(-)-2-fluoro-N-[C]propylnorapomorphine for evaluation as a dopamine D agonist ligand for PET investigations
Søndergaard, K., Kristensen, Jesper Langgaard, Gillings, N. & Begtrup, M., 14 Oct 2005, In: European Journal of Organic Chemistry. 20, p. 4428-4433 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of tertiary benzamides via Pd-catalyzed coupling of arylboronic esters and carbamoyl chlorides
Lysén, M., Kelleher, S., Begtrup, M. & Kristensen, Jesper Langgaard, 24 Jun 2005, In: Journal of Organic Chemistry. 70, 13, p. 5342-5343 2 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1305029
Most downloads
-
551
downloads
Convenient access to F-18-labeled amines through the Staudinger reduction
Research output: Contribution to journal › Conference abstract in journal › Research
Published -
331
downloads
A strategic approach to [6,6]-bicyclic lactones: application towards the CD fragment of DHβE
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
223
downloads
Substrate- and Cofactor-independent Inhibition of Histone Demethylase KDM4C
Research output: Contribution to journal › Journal article › Research › peer-review
Published