Umberto Maria Battisti
Assistant Professor
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- 2022
- Published
Recent Advances in the Development of Tetrazine Ligation Tools for Pretargeted Nuclear Imaging
García-Vázquez, R., Battisti, Umberto Maria & Herth, Matthias Manfred, 2022, In: Pharmaceuticals. 15, 6, 25 p., 685.Research output: Contribution to journal › Review › Research › peer-review
- Published
[11C]Carboxylated Tetrazines for Facile Labeling of Trans-Cyclooctene-Functionalized PeptoBrushes
García-Vázquez, R., Battisti, Umberto Maria, Shalgunov, Vladimir, Schäfer, G., Barz, M. & Herth, Matthias Manfred, 2022, In: Macromolecular Rapid Communications. 43, 12, 7 p., 2100655.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development and evaluation of an 18F-labeled nanobody to target SARS-CoV-2's spike protein
Lopes van den Broek, S., García-Vázquez, R., Andersen, Ida Vang, Valenzuela-Nieto, G., Shalgunov, Vladimir, Battisti, Umberto Maria, Schwefel, D., Modhiran, N., Kramer, V., Cheuquemilla, Y., Jara, R., Salinas-Varas, C., Amarilla, A. A., Watterson, D., Rojas-Fernandez, A. & Herth, Matthias Manfred, 2022, In: Frontiers in Nuclear Medicine. 2, 1033697.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Benzothiadiazines derivatives as novel allosteric modulators of kainic acid receptors
Puja, G., Ravazzini, F., Losi, G., Bardoni, R., Battisti, Umberto Maria, Citti, C. & Cannazza, G., 2022, In: Journal of Physiology and Pharmacology. 73, 1, p. 19-28Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of the First Tritiated Tetrazine: Facilitating Tritiation of Proteins
Radjani Bidesi, N. S., Battisti, Umberto Maria, Lopes van de Broek, S., Shalgunov, Vladimir, Dall, A., Bøggild Kristensen, J., Sehlin, D., Syvänen, S., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2022, In: ChemBioChem. 23, 23, 7 p., e202200539.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Evaluation of the α-synuclein PET radiotracer (d3)-[11C]MODAG-001 in pigs
Raval, N. R., Madsen, C. A., Shalgunov, Vladimir, Nasser, A., Battisti, Umberto Maria, Beaman, Emily Eufaula, Juhl, M., Jørgensen, Louise Møller, Herth, Matthias Manfred, Hansen, H. D., Plavén-Sigray, P. & Knudsen, Gitte Moos, 2022, In: Nuclear Medicine and Biology. 114-115, p. 42-48Research output: Contribution to journal › Journal article › Research › peer-review
- 2023
- Accepted/In press
Labeling of highly reactive tetrazines using [ 18F]SuFEx
Battisti, Umberto Maria, Müller, Marius, García-Vázquez, R. & Herth, Matthias Manfred, 2023, (Accepted/In press) In: Synlett.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and radiolabeling of a polar [125 I]I-1,2,4,5-tetrazine
Bidesi, N., Shalgunov, Vladimir, Battisti, Umberto Maria, Hvass, Lars, Jørgensen, Jesper Tranekjær, Poulie, Christian Bernard Matthijs, Jensen, A. I., Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 1, p. 22-30Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A Fluorescent Probe as a Lead Compound for a Selective α-Synuclein PET Tracer: Development of a Library of 2-Styrylbenzothiazoles and Biological Evaluation of [18F]PFSB and [18F]MFSB
Di Nanni, A., Saw, R. S., Battisti, Umberto Maria, Bowden, G. D., Boeckermann, A., Bjerregaard-Andersen, K., Pichler, B. J., Herfert, K., Herth, Matthias Manfred & Maurer, A., 2023, In: ACS Omega. 8, 34, p. 31450–31467Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and in vivo evaluation of [11C]tucatinib for HER2-targeted PET imaging
Müller, Marius, Shalgunov, Vladimir, Hvass, Lars, Jørgensen, Jesper Tranekjær, Kramer, V., Staudt, Markus, Battisti, Umberto Maria, Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Bioorganic and Medicinal Chemistry Letters. 80, 5 p., 129088.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 210553848
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Development of18F-Labeled Bispyridyl Tetrazines for In Vivo Pretargeted PET Imaging
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
55
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Direct Cu-mediated aromatic18F-labeling of highly reactive tetrazines for pretargeted bioorthogonal PET imaging
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
36
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Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry
Research output: Contribution to journal › Journal article › Research › peer-review
Published