Umberto Maria Battisti
Assistant Professor
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- Published
Direct Aromatic F-18-labeling of Tetrazines: A Rapid and Convenient Entry to Tetrazines for Pretargeted PET Imaging [Meeting Abstract]
Vazquez, R. G., Battisti, Umberto Maria, Stares, D. L., Petersen, I. N., Crestey, F., Svatunek, D., Mikula, H., Kristensen, Jesper Langgaard, Kjær, Andreas & Herth, Matthias Manfred, 2020, In: Journal of Nuclear Medicine. 61, Supl. 1, 2 p., 134.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry
Steen, E. J. L., Jørgensen, Jesper Tranekjær, Denk, C., Battisti, Umberto Maria, Norregaard, K., Edem, P. E., Bratteby, K., Shalgunov, Vladimir, Wilkovitsch, M., Svatunek, D., Poulie, Christian Bernard Matthijs, Hvass, Lars, Simon, M., Wanek, T., Rossin, R., Robillard, M., Kristensen, Jesper Langgaard, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: ACS Pharmacology & Translational Science. 4, 2, p. 824-833 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Spiroxatrine derivatives towards 5-HT1A receptor selectivity
Sorbi, C., Tait, A., Battisti, Umberto Maria & Brasili, L., 2020, In: Pharmacological Reports. 72, 2, p. 427-434 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Evaluation of F-537-Tetrazine in a model for brain pretargeting imaging. Comparison to N-(3-[18F] fluoro-5-(1,2,4,5-tetrazin-3-yl)benzyl)propan-1-amine
Shalgunov, Vladimir, van den Broek, S. L., Andersen, Ida Vang, Raval, N. R., Schäfer, G., Barz, M., Herth, Matthias Manfred & Battisti, Umberto Maria, 2024, In: Nuclear Medicine and Biology. 128-129, 12 p., 108877.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
Schlein, E., Rokka, J., Odell, L. R., van den Broek, S. L., Herth, Matthias Manfred, Battisti, Umberto Maria, Syvänen, S., Sehlin, D. & Eriksson, J., 2024, In: EJNMMI Radiopharmacy and Chemistry. 9, 1, 12 p., 21.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Evaluation of the α-synuclein PET radiotracer (d3)-[11C]MODAG-001 in pigs
Raval, N. R., Madsen, C. A., Shalgunov, Vladimir, Nasser, A., Battisti, Umberto Maria, Beaman, Emily Eufaula, Juhl, M., Jørgensen, Louise Møller, Herth, Matthias Manfred, Hansen, H. D., Plavén-Sigray, P. & Knudsen, Gitte Moos, 2022, In: Nuclear Medicine and Biology. 114-115, p. 42-48Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of the First Tritiated Tetrazine: Facilitating Tritiation of Proteins
Radjani Bidesi, N. S., Battisti, Umberto Maria, Lopes van de Broek, S., Shalgunov, Vladimir, Dall, A., Bøggild Kristensen, J., Sehlin, D., Syvänen, S., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2022, In: ChemBioChem. 23, 23, 7 p., e202200539.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Benzothiadiazines derivatives as novel allosteric modulators of kainic acid receptors
Puja, G., Ravazzini, F., Losi, G., Bardoni, R., Battisti, Umberto Maria, Citti, C. & Cannazza, G., 2022, In: Journal of Physiology and Pharmacology. 73, 1, p. 19-28Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Next generation fibroblast activation protein (FAP) targeting PET tracers : The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines
Poulie, Christian Bernard Matthijs, Shalgunov, Vladimir, Elvas, F., Van Rymenant, Y., Moon, E. S., Battisti, Umberto Maria, De Loose, J., De Meester, I., Rösch, F., Van Der Veken, P. & Herth, Matthias Manfred, 2023, In: European Journal of Medicinal Chemistry. 262, 10 p., 115862.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and in vivo evaluation of [11C]tucatinib for HER2-targeted PET imaging
Müller, Marius, Shalgunov, Vladimir, Hvass, Lars, Jørgensen, Jesper Tranekjær, Kramer, V., Staudt, Markus, Battisti, Umberto Maria, Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Bioorganic and Medicinal Chemistry Letters. 80, 5 p., 129088.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 210553848
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Development of18F-Labeled Bispyridyl Tetrazines for In Vivo Pretargeted PET Imaging
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
44
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Direct Cu-mediated aromatic18F-labeling of highly reactive tetrazines for pretargeted bioorthogonal PET imaging
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
34
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Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry
Research output: Contribution to journal › Journal article › Research › peer-review
Published