Vladimir Shalgunov
Guest Researcher
Medicinal Chemistry
Jagtvej 162
2100 København Ø
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Investigation of imaging the somatostatin receptor by opening the blood-brain barrier with melittin – A feasibility study using positron emission tomography and [64Cu]Cu-DOTATATE
Andersen, Ida Vang, Bidesi, N. S. R., Shalgunov, Vladimir, Jørgensen, Jesper Tranekjær, Gustavsson, Karl Tobias, Strømgaard, Kristian, Ingemann Jensen, A. T., Kjær, Andreas & Herth, Matthias Manfred, 2024, In: Nuclear Medicine and Biology. 132-133, 5 p., 108905.Research output: Contribution to journal › Journal article › Research › peer-review
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Development of the First Aliphatic 18F-Labeled Tetrazine Suitable for Pretargeted PET Imaging-Expanding the Bioorthogonal Tool Box
Battisti, Umberto Maria, Bratteby, K., Jørgensen, Jesper Tranekjær, Hvass, Lars, Shalgunov, Vladimir, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Journal of Medicinal Chemistry. 64, 20, p. 15297–15312Research output: Contribution to journal › Journal article › Research › peer-review
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Synthesis and radiolabeling of a polar [125 I]I-1,2,4,5-tetrazine
Bidesi, N., Shalgunov, Vladimir, Battisti, Umberto Maria, Hvass, Lars, Jørgensen, Jesper Tranekjær, Poulie, Christian Bernard Matthijs, Jensen, A. I., Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 1, p. 22-30Research output: Contribution to journal › Journal article › Research › peer-review
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The role of neuroimaging in Parkinson’s disease
Bidesi, N. S. R., Andersen, Ida Vang, Windhorst, A. D., Shalgunov, Vladimir & Herth, Matthias Manfred, 2021, In: Journal of Neurochemistry. 159, 4, p. 660-689Research output: Contribution to journal › Review › Research › peer-review
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F-18-Radiolabeling and in vivo evaluation of two diverse glycomimetics using PET
Bratteby, K., Torkelsson, E., L'Estrade, E. T., Peterson, K., Shalgunov, Vladimir, Xiong, M., Leffer, H., Zetterberg, F., Ohlsson, T., Gillings, N., Nilsson, U., Herth, Matthias Manfred & Erlandsson, M., May 2019, p. S533-S534.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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Aliphatic 18F-Radiofluorination: Recent Advances in the Labeling of Base-Sensitive Substrates**
Bratteby, K., Shalgunov, Vladimir & Herth, Matthias Manfred, 2021, In: ChemMedChem. 16, 17, p. 2612-2622Research output: Contribution to journal › Review › Research › peer-review
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Insights into Elution of Anion Exchange Cartridges: Opening the Path toward Aliphatic 18F-Radiolabeling of Base-Sensitive Tracers
Bratteby, K., Shalgunov, Vladimir, Battisti, Umberto Maria, Petersen, I. N., Van Den Broek, S. L., Ohlsson, T., Gillings, N., Erlandsson, M. & Herth, Matthias Manfred, 2021, In: ACS Pharmacology and Translational Science. 4, 5, p. 1556–1566Research output: Contribution to journal › Journal article › Research › peer-review
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In Vivo Veritas - 18F-radiolabeled glycomimetics allow insights into the pharmacological fate of galectin-3 inhibitors
Bratteby, K., Torkelsson, E., Tampio L'Estrade, E., Peterson, K., Shalgunov, Vladimir, Xiong, M., Leffler, H., Zetterberg, F., Olsson, T. G., Gillings, N., Nilsson, U. J., Herth, Matthias Manfred & Erlandsson, M., 2020, In: Journal of Medicinal Chemistry. 63, 2, p. 747-755Research output: Contribution to journal › Journal article › Research › peer-review
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The Chemogenetic Receptor Ligand Clozapine N-Oxide Induces in vivo Neuroreceptor Occupancy and Reduces Striatal Glutamate Levels
Bærentzen, S., Casado-Sainz, A., Lange, D., Shalgunov, Vladimir, Tejada, I. M., Xiong, M., L'Estrade, E. T., Edgar, F. G., Lee, H., Herth, Matthias Manfred & Palner, M., 2019, In: Frontiers in Neuroscience. 13, 7 p., 187.Research output: Contribution to journal › Journal article › Research › peer-review
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A pilot study of cerebral metabolism and serotonin 5-HT2A receptor occupancy in rats treated with the psychedelic tryptamine DMT in conjunction with the MAO inhibitor harmine
Egger, K., Gudmundsen, F., Jessen, N. S., Baun, C., Poetzsch, S. N., Shalgunov, Vladimir, Herth, Matthias Manfred, Quednow, B. B., Martin-Soelch, C., Dornbierer, D., Scheidegger, M., Cumming, P. & Palner, M., 2023, In: Frontiers in Pharmacology. 14, 12 p., 1140656.Research output: Contribution to journal › Journal article › Research › peer-review
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Development of18F-Labeled Bispyridyl Tetrazines for In Vivo Pretargeted PET Imaging
García-Vázquez, R., Jørgensen, Jesper Tranekjær, Bratteby, K. E., Shalgunov, Vladimir, Hvass, Lars, Herth, Matthias Manfred, Kjær, Andreas & Battisti, Umberto Maria, 2022, In: Pharmaceuticals. 15, 2, 28 p., 245.Research output: Contribution to journal › Journal article › Research › peer-review
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Direct Cu-mediated aromatic18F-labeling of highly reactive tetrazines for pretargeted bioorthogonal PET imaging
García-Vázquez, R., Battisti, Umberto Maria, Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Hvass, Lars, Stares, D. L., Petersen, I. N., Crestey, F., Löffler, A., Svatunek, D., Kristensen, Jesper Langgaard, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Chemical Science. 12, 35, p. 11668-11675Research output: Contribution to journal › Journal article › Research › peer-review
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[11C]Carboxylated Tetrazines for Facile Labeling of Trans-Cyclooctene-Functionalized PeptoBrushes
García-Vázquez, R., Battisti, Umberto Maria, Shalgunov, Vladimir, Schäfer, G., Barz, M. & Herth, Matthias Manfred, 2022, In: Macromolecular Rapid Communications. 43, 12, 7 p., 2100655.Research output: Contribution to journal › Journal article › Research › peer-review
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On the consensus nomenclature rules for radiopharmaceutical chemistry - Reconsideration of radiochemical conversion
Herth, M. M., Ametamey, S., Antuganov, D., Bauman, A., Berndt, M., Brooks, A. F., Bormans, G., Choe, Y. S., Gillings, N., Hafeli, U. O., James, M. L., Kopka, K., Kramer, V., Krasikova, R., Madsen, J., Mu, L., Neumaier, B., Piel, M., Roesch, F., Ross, T. & 6 others, , 2021, In: Nuclear Medicine and Biology. 93, p. 19-21 3 p.Research output: Contribution to journal › Editorial › Research › peer-review
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Preliminary Evaluation of (S)-7-[F-18]Fluorotryptophan as a Tracer for the Imaging of Tryptophan Metabolism Alterations in Tumor Xenografts
Hvass, L., Shalgunov, Vladimir, Jorgensen, J. T., Zlatopolskiy, B. D., Neumaier, B., Kjær, Andreas & Herth, Matthias Manfred, 2020, In: European Journal of Nuclear Medicine and Molecular Imaging. 47, SUPPL 1, p. S646-S647 Meeting Abstract: EP-282 .Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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The polypharmacological profile of psilocybin and potential behavioural effects of very low doses
Kiilerich, K., Speth, N., Lorenz, J., Casado-Sainz, A., Shalgunov, Vladimir, Lange, D., Xiong, M., Herth, Matthias Manfred, Overgaard, A., Hansen, H. D. & Palner, M., 2019, In: European Neuropsychopharmacology. 29, Supplement 6, p. S175-S176 2 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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Repeated low doses of psilocybin increase resilience to stress, lower compulsive actions, and strengthen cortical connections to the paraventricular thalamic nucleus in rats
Kiilerich, K. F., Lorenz, J., Scharff, M. B., Speth, N., Brandt, T. G., Czurylo, J., Xiong, M., Jessen, N. S., Casado-Sainz, A., Shalgunov, Vladimir, Kjærby, Celia, Satała, G., Bojarski, A. J., Jensen, Anders A., Herth, Matthias Manfred, Cumming, P., Overgaard, A. & Palner, M., 2023, In: Molecular Psychiatry. 28, 9, p. 3829-3841Research output: Contribution to journal › Journal article › Research › peer-review
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Radiosynthesis and preclinical evaluation of [11 C]Cimbi-701 - Towards the imaging of cerebral 5-HT7 receptors
L 'Estrade, E. T., Shalgunov, Vladimir, Edgar, F. G., Strebl-Bantillo, M. G., Xiong, M., Crestey, F., Neelamegam, R., Dyssegaard, A., Lehel, S., Erlandsson, M., Ohlsson, T., Hooker, J. M., Knudsen, Gitte Moos, Herth, Matthias Manfred & Hansen, H. D., 2020, In: Journal of Labelled Compounds and Radiopharmaceuticals. 63, p. 46-55Research output: Contribution to journal › Journal article › Research › peer-review
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PET radiotracer translation from rats to higher species, using an increased-throughput in vivo evaluation strategy
L'Estrade, E. T., Xiong, M., Petersen, I., Shalgunov, Vladimir, Edgar, F. G., Hansen, H., Erlandsson, M., Ohlsson, T., Knudsen, Gitte Moos, Palner, M. & Herth, Matthias Manfred, May 2019, p. S389-S390.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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High-throughput rat brain PET imaging and automatic spatial normalization of the dopamine D2/3 receptor ligand [F-18]fallypride
Lange, D., Tejada, I. M., Xiong, M., Hillebrand, B., Noergaard, M., Baerentzen, S., Shalgunov, Vladimir, Herth, Matthias Manfred, Svarer, C. & Palner, M., 2019, In: Journal of Cerebral Blood Flow and Metabolism. 39, p. 588-589 2 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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Development and evaluation of an 18F-labeled nanobody to target SARS-CoV-2's spike protein
Lopes van den Broek, S., García-Vázquez, R., Andersen, Ida Vang, Valenzuela-Nieto, G., Shalgunov, Vladimir, Battisti, Umberto Maria, Schwefel, D., Modhiran, N., Kramer, V., Cheuquemilla, Y., Jara, R., Salinas-Varas, C., Amarilla, A. A., Watterson, D., Rojas-Fernandez, A. & Herth, Matthias Manfred, 2022, In: Frontiers in Nuclear Medicine. 2, 1033697.Research output: Contribution to journal › Journal article › Research › peer-review
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Pretargeted Imaging beyond the Blood–Brain Barrier: Utopia or Feasible?
Lopes van den Broek, S., Shalgunov, Vladimir, García Vázquez, R., Beschorner, Natalie, Bidesi, N. S. R., Nedergaard, Maiken, Knudsen, Gitte Moos, Sehlin, D., Syvänen, S. & Herth, Matthias Manfred, 2022, In: Pharmaceuticals. 15, 10, 13 p., 1191.Research output: Contribution to journal › Journal article › Research › peer-review
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A facile synthesis of precursor for the σ-1 receptor PET radioligand [18F]FTC-146 and its radiofluorination
Marešová, A., Jurášek, M., Drašar, P. B., Dolenský, B., Prokudina, E. A., Shalgunov, Vladimir, Herth, Matthias Manfred, Cumming, P. & Popkov, A., 2024, In: Journal of Labelled Compounds and Radiopharmaceuticals. 67, 2, p. 59-66Research output: Contribution to journal › Journal article › Research › peer-review
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Synthesis and in vivo evaluation of [11C]tucatinib for HER2-targeted PET imaging
Müller, Marius, Shalgunov, Vladimir, Hvass, Lars, Jørgensen, Jesper Tranekjær, Kramer, V., Staudt, Markus, Battisti, Umberto Maria, Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Bioorganic and Medicinal Chemistry Letters. 80, 5 p., 129088.Research output: Contribution to journal › Journal article › Research › peer-review
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Evaluation of [Cu-64]Cu-NOTA-PEG7-H-Tz for Pretargeted Imaging in LS174T Xenografts-Comparison to [111In-111]In-DOTA-PEG11-BisPy-Tz
Poulie, Christian Bernard Matthijs, Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Kougioumtzoglou, G., Jeppesen, T. E., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Molecules. 26, 3, 9 p., 544.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 185059116
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SPECT imaging of the glymphatic pathway with In-111-labeled ovalbumin in the rat brain
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Convenient access to F-18-labeled amines through the Staudinger reduction
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369
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Pretargeting in nuclear imaging and radionuclide therapy: Improving efficacy of theranostics and nanomedicines
Research output: Contribution to journal › Journal article › Research › peer-review
Published