Vladimir Shalgunov
Guest Researcher
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- Published
In Vivo Veritas - 18F-radiolabeled glycomimetics allow insights into the pharmacological fate of galectin-3 inhibitors
Bratteby, K., Torkelsson, E., Tampio L'Estrade, E., Peterson, K., Shalgunov, Vladimir, Xiong, M., Leffler, H., Zetterberg, F., Olsson, T. G., Gillings, N., Nilsson, U. J., Herth, Matthias Manfred & Erlandsson, M., 2020, In: Journal of Medicinal Chemistry. 63, 2, p. 747-755Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Insights into Elution of Anion Exchange Cartridges: Opening the Path toward Aliphatic 18F-Radiolabeling of Base-Sensitive Tracers
Bratteby, K., Shalgunov, Vladimir, Battisti, Umberto Maria, Petersen, I. N., Van Den Broek, S. L., Ohlsson, T., Gillings, N., Erlandsson, M. & Herth, Matthias Manfred, 2021, In: ACS Pharmacology and Translational Science. 4, 5, p. 1556–1566Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Investigation of imaging the somatostatin receptor by opening the blood-brain barrier with melittin – A feasibility study using positron emission tomography and [64Cu]Cu-DOTATATE
Andersen, Ida Vang, Bidesi, N. S. R., Shalgunov, Vladimir, Jørgensen, Jesper Tranekjær, Gustavsson, Karl Tobias, Strømgaard, Kristian, Ingemann Jensen, A. T., Kjær, Andreas & Herth, Matthias Manfred, 2024, In: Nuclear Medicine and Biology. 132-133, 5 p., 108905.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry
Steen, E. J. L., Jørgensen, Jesper Tranekjær, Denk, C., Battisti, Umberto Maria, Norregaard, K., Edem, P. E., Bratteby, K., Shalgunov, Vladimir, Wilkovitsch, M., Svatunek, D., Poulie, Christian Bernard Matthijs, Hvass, Lars, Simon, M., Wanek, T., Rossin, R., Robillard, M., Kristensen, Jesper Langgaard, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: ACS Pharmacology & Translational Science. 4, 2, p. 824-833 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Next generation fibroblast activation protein (FAP) targeting PET tracers : The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines
Poulie, Christian Bernard Matthijs, Shalgunov, Vladimir, Elvas, F., Van Rymenant, Y., Moon, E. S., Battisti, Umberto Maria, De Loose, J., De Meester, I., Rösch, F., Van Der Veken, P. & Herth, Matthias Manfred, 2023, In: European Journal of Medicinal Chemistry. 262, 10 p., 115862.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
On the consensus nomenclature rules for radiopharmaceutical chemistry - Reconsideration of radiochemical conversion
Herth, M. M., Ametamey, S., Antuganov, D., Bauman, A., Berndt, M., Brooks, A. F., Bormans, G., Choe, Y. S., Gillings, N., Hafeli, U. O., James, M. L., Kopka, K., Kramer, V., Krasikova, R., Madsen, J., Mu, L., Neumaier, B., Piel, M., Roesch, F., Ross, T. & 6 others, , 2021, In: Nuclear Medicine and Biology. 93, p. 19-21 3 p.Research output: Contribution to journal › Editorial › Research › peer-review
- Published
PET radiotracer translation from rats to higher species, using an increased-throughput in vivo evaluation strategy
L'Estrade, E. T., Xiong, M., Petersen, I., Shalgunov, Vladimir, Edgar, F. G., Hansen, H., Erlandsson, M., Ohlsson, T., Knudsen, Gitte Moos, Palner, M. & Herth, Matthias Manfred, May 2019, p. S389-S390.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
Preliminary Evaluation of (S)-7-[F-18]Fluorotryptophan as a Tracer for the Imaging of Serotonin Synthesis in Pig Brain
Shalgunov, Vladimir, Raval, N. R., Donovan, L. L., Nasser, A., Zlatopolskiy, B. D., Neumaier, B., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2020, In: European Journal of Nuclear Medicine and Molecular Imaging. 47, SUPPL 1, p. S639-S639 EP-267 .Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Preliminary Evaluation of (S)-7-[F-18]Fluorotryptophan as a Tracer for the Imaging of Tryptophan Metabolism Alterations in Tumor Xenografts
Hvass, L., Shalgunov, Vladimir, Jorgensen, J. T., Zlatopolskiy, B. D., Neumaier, B., Kjær, Andreas & Herth, Matthias Manfred, 2020, In: European Journal of Nuclear Medicine and Molecular Imaging. 47, SUPPL 1, p. S646-S647 Meeting Abstract: EP-282 .Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Pretargeted Imaging beyond the Blood–Brain Barrier: Utopia or Feasible?
Lopes van den Broek, S., Shalgunov, Vladimir, García Vázquez, R., Beschorner, Natalie, Bidesi, N. S. R., Nedergaard, Maiken, Knudsen, Gitte Moos, Sehlin, D., Syvänen, S. & Herth, Matthias Manfred, 2022, In: Pharmaceuticals. 15, 10, 13 p., 1191.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Pretargeting in nuclear imaging and radionuclide therapy: Improving efficacy of theranostics and nanomedicines
Stéen, E. J. L., Edem, P. E., Nørregaard, K., Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Kjær, Andreas & Herth, Matthias Manfred, Oct 2018, In: Biomaterials. 179, p. 209-245 37 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Radiolabeling of a polypeptide polymer for intratumoral delivery of alpha-particle emitter, 225Ac, and beta-particle emitter, 177Lu
Shalgunov, Vladimir, Engudar, G., Bohrmann, L., Wharton, L., Maskell, K., Johann, K., Barz, M., Schaffer, P., Herth, Matthias Manfred & Radchenko, V., 2022, In: Nuclear Medicine and Biology. 104-105, p. 11-21Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Radiosynthesis and preclinical evaluation of [11 C]Cimbi-701 - Towards the imaging of cerebral 5-HT7 receptors
L 'Estrade, E. T., Shalgunov, Vladimir, Edgar, F. G., Strebl-Bantillo, M. G., Xiong, M., Crestey, F., Neelamegam, R., Dyssegaard, A., Lehel, S., Erlandsson, M., Ohlsson, T., Hooker, J. M., Knudsen, Gitte Moos, Herth, Matthias Manfred & Hansen, H. D., 2020, In: Journal of Labelled Compounds and Radiopharmaceuticals. 63, p. 46-55Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Repeated low doses of psilocybin increase resilience to stress, lower compulsive actions, and strengthen cortical connections to the paraventricular thalamic nucleus in rats
Kiilerich, K. F., Lorenz, J., Scharff, M. B., Speth, N., Brandt, T. G., Czurylo, J., Xiong, M., Jessen, N. S., Casado-Sainz, A., Shalgunov, Vladimir, Kjærby, Celia, Satała, G., Bojarski, A. J., Jensen, Anders A., Herth, Matthias Manfred, Cumming, P., Overgaard, A. & Palner, M., 2023, In: Molecular Psychiatry. 28, 9, p. 3829-3841Research output: Contribution to journal › Journal article › Research › peer-review
- Published
SPECT imaging of the glymphatic pathway with In-111-labeled ovalbumin in the rat brain
Shalgunov, Vladimir, Lilius, T., Sigurosson, B., Baerentzen, S. L., Hauglund, Natalie Linea, Herth, Matthias Manfred, Palner, M. & Nedergaard, Maiken, 2019, In: Journal of Labelled Compounds and Radiopharmaceuticals. 62, Supplement 1, p. S404-S405 2 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Synthesis and in vivo evaluation of [11C]tucatinib for HER2-targeted PET imaging
Müller, Marius, Shalgunov, Vladimir, Hvass, Lars, Jørgensen, Jesper Tranekjær, Kramer, V., Staudt, Markus, Battisti, Umberto Maria, Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Bioorganic and Medicinal Chemistry Letters. 80, 5 p., 129088.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and radiolabeling of a polar [125 I]I-1,2,4,5-tetrazine
Bidesi, N., Shalgunov, Vladimir, Battisti, Umberto Maria, Hvass, Lars, Jørgensen, Jesper Tranekjær, Poulie, Christian Bernard Matthijs, Jensen, A. I., Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 1, p. 22-30Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis, Radiolabeling, and in Vitro and in Vivo Evaluation of [18F]ENL30: A Potential PET Radiotracer for the 5-HT7 Receptor
Tampio L'Estrade, E., Edgar, F. G., Xiong, M., Shalgunov, Vladimir, Baerentzen, S. L., Erlandsson, M., Ohlsson, T. G., Palner, M., Knudsen, Gitte Moos & Herth, Matthias Manfred, 23 Apr 2019, In: ACS Omega. 4, 4, p. 7344-7353Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The Chemogenetic Receptor Ligand Clozapine N-Oxide Induces in vivo Neuroreceptor Occupancy and Reduces Striatal Glutamate Levels
Bærentzen, S., Casado-Sainz, A., Lange, D., Shalgunov, Vladimir, Tejada, I. M., Xiong, M., L'Estrade, E. T., Edgar, F. G., Lee, H., Herth, Matthias Manfred & Palner, M., 2019, In: Frontiers in Neuroscience. 13, 7 p., 187.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The polypharmacological profile of psilocybin and potential behavioural effects of very low doses
Kiilerich, K., Speth, N., Lorenz, J., Casado-Sainz, A., Shalgunov, Vladimir, Lange, D., Xiong, M., Herth, Matthias Manfred, Overgaard, A., Hansen, H. D. & Palner, M., 2019, In: European Neuropsychopharmacology. 29, Supplement 6, p. S175-S176 2 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
The role of neuroimaging in Parkinson’s disease
Bidesi, N. S. R., Andersen, Ida Vang, Windhorst, A. D., Shalgunov, Vladimir & Herth, Matthias Manfred, 2021, In: Journal of Neurochemistry. 159, 4, p. 660-689Research output: Contribution to journal › Review › Research › peer-review
- Published
Trans-Cyclooctene-Functionalized PeptoBrushes with Improved Reaction Kinetics of the Tetrazine Ligation for Pretargeted Nuclear Imaging
Stéen, E. J. L., Jørgensen, Jesper Tranekjær, Johann, K., Norregaard, K., Sohr, B., Svatunek, D., Birke, A., Shalgunov, Vladimir, Edem, P. E., Rossin, R., Seidl, C., Schmid, F., Robillard, M. S., Kristensen, Jesper Langgaard, Mikula, H., Barz, M., Kjær, Andreas & Herth, Matthias Manfred, 2020, In: ACS Nano. 14, 1, p. 568-584Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Transport of nanomedicines across the blood-brain barrier: Challenges and opportunities for imaging and therapy
van den Broek, S. L., Shalgunov, Vladimir & Herth, Matthias Manfred, 2022, In: Biomaterials Advances. 141, 11 p., 213125.Research output: Contribution to journal › Review › Research › peer-review
- Published
[11C]Carboxylated Tetrazines for Facile Labeling of Trans-Cyclooctene-Functionalized PeptoBrushes
García-Vázquez, R., Battisti, Umberto Maria, Shalgunov, Vladimir, Schäfer, G., Barz, M. & Herth, Matthias Manfred, 2022, In: Macromolecular Rapid Communications. 43, 12, 7 p., 2100655.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 185059116
Most downloads
-
580
downloads
SPECT imaging of the glymphatic pathway with In-111-labeled ovalbumin in the rat brain
Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
Published -
551
downloads
Convenient access to F-18-labeled amines through the Staudinger reduction
Research output: Contribution to journal › Conference abstract in journal › Research
Published -
368
downloads
Pretargeting in nuclear imaging and radionuclide therapy: Improving efficacy of theranostics and nanomedicines
Research output: Contribution to journal › Journal article › Research › peer-review
Published