Anders Skov Kristensen

Anders Skov Kristensen

Associate Professor


  1. 2009
  2. Published

    Recent advances in the understanding of the interaction of antidepressant drugs with serotonin and norepinephrine transporters

    Andersen, J., Kristensen, Anders Skov, Bang-Andersen, B. & Strømgaard, Kristian, 2009, In: Chemical Communications. 25, p. 3677-3692

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Design and synthesis of highly potent and plasma-stable dimeric inhibitors of the PSD-95-NMDA receptor interaction

    Bach, Anders, Chi, C. N., Pang, G. F., Olsen, L., Kristensen, Anders Skov, Jemth, P. & Strømgaard, Kristian, 2009, In: Angewandte Chemie - International Edition. 48, 51, p. 9685-9689

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    The glutamate receptor GluR5 agonist (S)-2-amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid and the 8-methyl analogue: synthesis, molecular pharmacology, and biostructural characterization

    Clausen, Rasmus Prætorius, Naur, P., Kristensen, Anders Skov, Greenwood, J. R., Strange, M., Bräuner, Hans, Jensen, Anders A., Nielsen, A. S. T., Geneser, U., Ringgaard, L. M., Nielsen, Birgitte, Pickering, Darryl S, Brehm, L., Gajhede, Michael, Krogsgaard-Larsen, Povl & Kastrup, Jette Sandholm Jensen, 2009, In: Journal of Medicinal Chemistry. 52, 15, p. 4911-4922

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Detecting protein-protein interactions in living cells: development of a bioluminescence resonance energy transfer assay to evaluate the PSD-95/NMDA receptor interaction

    Gottschalk, M., Bach, Anders, Hansen, J. L., Krogsgaard-Larsen, Povl, Kristensen, Anders Skov & Strømgaard, Kristian, 2009, In: Neurochemical Research. 34, 10, p. 1729-1737

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Modulation of the dimer interface at ionotropic glutamate-like receptor d2 by D-serine and extracellular calcium

    Hansen, K. B., Naur, P., Kurtkaya, N. L., Kristensen, Anders Skov, Gajhede, Michael, Kastrup, Jette Sandholm Jensen & Traynelis, S. F., 2009, In: Journal of Neuroscience. 29, 4, p. 907-917

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Synthesis and biological activity of argiotoxin 636 and analogues: selective antagonists for ionotropic glutamate receptors

    Nelson, J. K., Frølund, S. U., Tikhonov, D. B., Kristensen, Anders Skov & Strømgaard, Kristian, 2009, In: Angewandte Chemie - International Edition. 48, 17, p. 3087-3091

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Skræddersyede proteiner: uden naturens begrænsninger

    Strømgaard, Kristian, Jensen, M. S. & Kristensen, Anders Skov, 2009, In: Lægemiddelforskning. p. 10-12

    Research output: Contribution to journalJournal articleCommunication

  9. 2008
  10. Published

    Protein-protein interaktion: et nyt mål for udvikling af lægemidler

    Bach, Anders, Gottschalk, M., Kristensen, Anders Skov & Strømgaard, Kristian, 2008, In: Lægemiddelforskning. p. 10-12

    Research output: Contribution to journalJournal articleCommunication

  11. Published

    From the selective serotonin transporter inhibitor citalopram to the selective norepinephrine transporter inhibitor talopram: Synthesis and structure-activity relationship studies

    Eildal, J. N. N., Andersen, J., Kristensen, Anders Skov, Jørgensen, A. M., Bang-Andersen, B., Jørgensen, M. & Strømgaard, Kristian, 2008, In: Journal of Medicinal Chemistry. 51, 10, p. 3045-3048

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Electrophysiological characterization of analogues of philanthotoxin-343 on ionotropic glutamate receptors

    Frølund, S. U., Ziegler, H. L., Franzyk, Henrik, Strømgaard, Kristian, Kristensen, Anders Skov & Jaroszewski, J. W., 2008.

    Research output: Contribution to conferencePosterResearch

  13. 2007
  14. Published

    Subunit-specific agonist activity at NR2A-, NR2B-, NR2C-, and NR2D-containing N-methyl-D-aspartate glutamate receptors

    Erreger, K., Geballe, M. T., Kristensen, Anders Skov, Chen, P. E., Hansen, K. B., Lee, C. J., Yuan, H., Le, P., Lyuboslavsky, P. N., Micale, N., Jørgensen, L., Clausen, Rasmus Prætorius, Wyllie, D. J. A., Snyder, J. P. & Traynelis, S. F., 2007, In: Molecular Pharmacology. 72, 4, p. 907-920

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Expressed protein ligation of ionotropic glutamate receptors

    Jensen, M. S., Kristensen, Anders Skov & Strømgaard, Kristian, 2007, In: Biopolymers. 88, 4, p. 602

    Research output: Contribution to journalConference abstract in journalResearch

  16. Published

    Structural correlates of ionotropic glutamate receptor function

    Kristensen, Anders Skov, Hansen, K. B., Wollmuth, L. P., Egebjerg, J. & Traynelis, S. F., 2007, The receptors: The glutamate receptors. Gereau, R. W. & Swanson, G. T. (eds.). 1. ed. Totowa N.J., USA: Humana Press, p. 247-299 42 p.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  17. Published

    Ionotropic glutamate-like receptor d2 binds D-serine and glycine.

    Naur, P., Hansen, K. B., Kristensen, Anders Skov, Dravid, S. M., Pickering, Darryl S, Olsen, L., Vestergaard, Bente, Egebjerg, J., Gajhede, Michael, Traynelis, S. F. & Kastrup, Jette Sandholm Jensen, 2007, In: Proceedings of the National Academy of Science of the United States of America. 104, 35, p. 14116-14121

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. 2006
  19. Published

    The structure of a mixed GluR2 ligand-binding core dimer in complex with (S)-glutamate and the antagonist (S)-NS1209

    Kasper, C., Pickering, Darryl S, Mirza, Osman Asghar, Olsen, L., Kristensen, Anders Skov, Greenwood, J. R., Liljefors, T., Schousboe, Arne, Wätjen, F., Gajhede, Michael, Sigurskjold, B. W. & Kastrup, Jette Sandholm Jensen, 2006, In: Journal of Molecular Biology. 357, 4, p. 1184-201 17 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Glutamate receptors: variation in structure-function coupling

    Kristensen, Anders Skov, Geballe, M. T., Snyder, J. P. & Traynelis, S. F., Feb 2006, In: Trends in Pharmacological Sciences. 27, 2, p. 65-9 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Glutamate receptors: variation in structure-function coupling

    Kristensen, Anders Skov, Geballe, M., Snyder, J. P. & Traynelis, S. F., Feb 2006, In: Trends in Pharmacological Sciences. 27, 2, p. 65-69 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. 2005
  23. Published

    Neuroscience: an intrusive chaperone

    Kristensen, Anders Skov & Traynelis, S. F., 23 Jun 2005, In: Nature. 435, 7045, p. 1042-3 2 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Neuroscience: an intrusive chaperone

    Kristensen, Anders Skov, 23 Jun 2005, In: Nature. 435, 7045, p. 1042-1043 2 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. 2004
  26. Published

    Mutational scanning of the human serotonin transporter reveals fast translocating serotonin transporter mutants

    Kristensen, Anders Skov, Larsen, M. B., Johnsen, L. B. & Wiborg, O., Mar 2004, In: European Journal of Neuroscience. 19, 6, p. 1513-23 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    On the neurotoxicity of glutaric, 3-hydroxyglutaric, and trans-glutaconic acids in glutaric acidemia type 1

    Lund, Trine Meldgaard, Christensen, E., Kristensen, Anders Skov, Schousboe, Arne & Lund, Allan Meldgaard, 2004, In: Journal of Neuroscience Research. 77, 1, p. 143-7 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Bioisosteric modifications of 2-arylureidobenzoic acids: selective noncompetitive antagonists for the homomeric kainate receptor subtype GluR5

    Valgeirsson, J., Nielsen, E. O., Peters, D., Mathiesen, C., Kristensen, Anders Skov & Madsen, Ulf, 30 Dec 2004, In: Journal of Medicinal Chemistry. 47, 27, p. 6948-57 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. 2003
  30. Published

    Design, synthesis, and pharmacology of a highly subtype-selective GluR1/2 agonist, (RS)-2-amino-3-(4-chloro-3-hydroxy-5-isoxazolyl)propionic acid (Cl-HIBO)

    Bjerrum, E. J., Kristensen, Anders Skov, Pickering, D. S., Greenwood, J. R., Nielsen, Birgitte, Liljefors, T., Schousboe, Arne, Bräuner, Hans, Madsen, Ulf & Pickering, Darryl S, 2003, In: Journal of Medicinal Chemistry. 46, 11, p. 2246-9 3 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    2-arylureidobenzoic acids: selective noncompetitive antagonists for the homomeric kainate receptor subtype GluR5

    Valgeirsson, J., Nielsen, E. Ø., Peters, D., Varming, T., Mathiesen, C., Kristensen, Anders Skov & Madsen, Ulf, 18 Dec 2003, In: Journal of Medicinal Chemistry. 46, 26, p. 5834-43 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Synthesis and in vitro pharmacology at AMPA and kainate preferring glutamate receptors of 4-heteroarylmethylidene glutamate analogues

    Valgeirsson, J., Christensen, J. K., Kristensen, Anders Skov, Pickering, Darryl S, Nielsen, Birgitte, Fischer, C., Bräuner, Hans, Nielsen, E. Ø., Krogsgaard-Larsen, Povl & Madsen, U., 2003, In: Bioorganic & Medicinal Chemistry. 11, 20, p. 4341-9 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. 2001
  34. Published

    Species-scanning mutagenesis of the serotonin transporter reveals residues essential in selective, high-affinity recognition of antidepressants

    Mortensen, O. V., Kristensen, Anders Skov & Wiborg, O., Oct 2001, In: Journal of Neurochemistry. 79, 2, p. 237-47 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. 1999
  36. Published

    Molecular cloning, expression and characterization of a bovine serotonin transporter

    Mortensen, O. V., Kristensen, Anders Skov, Rudnick, G. & Wiborg, O., 23 Jul 1999, In: Brain Research. 71, 1, p. 120-6 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

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