Francesco Bavo

Francesco Bavo

Postdoc, Assistant Professor

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    1 - 10 out of 13Page size: 10
    1. 2019
    2. Published

      Discovery of 2-(Imidazo[1,2-b]pyridazin-2-yl)acetic Acid as a New Class of Ligands Selective for the γ-Hydroxybutyric Acid (GHB) High-Affinity Binding Sites

      Krall, J., Bavo, Francesco, Falk-Petersen, C. B., Jensen, C. H., Nielsen, J. O., Tian, Yongsong, Anglani, V., Kongstad, Kenneth Thermann, Petersen, Louise Piilgaard, Nielsen, Birgitte, Gloriam, David E., Kehler, J., Jensen, Anders A., Harpsøe, Kasper, Wellendorph, Petrine & Frølund, Bente, 14 Mar 2019, In: Journal of Medicinal Chemistry. 62, 5, p. 2798-2813

      Research output: Contribution to journal › Journal article › Research › peer-review

    3. Published

      Five-membered N-heterocyclic Scaffolds as Novel Amino Bioisosteres at gamma-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters

      Giraudo, A., Krall, J., Bavo, Francesco, Nielsen, Birgitte, Kongstad, Kenneth Thermann, Rolando, B., De Blasio, R., Gloriam, David E., Löffler, R., Thiesen, L., Harpsøe, Kasper, Frydenvang, Karla Andrea, Boschi, D., Wellendorph, Petrine, Lolli, M. L., Jensen, Anders A. & Frølund, Bente, 27 Jun 2019, In: Journal of Medicinal Chemistry. 62, 12, p. 5797-5809

      Research output: Contribution to journal › Journal article › Research › peer-review

    4. 2020
    5. Published

      Exploring the molecular determinants for subtype-selectivity of 2-amino-1,4,5,6-tetrahydropyrimidine-5-carboxylic acid analogs as betaine/GABA transporter 1 (BGT1) substrate-inhibitors

      Kickinger, S., Al-Khawaja, A., Haugaard, A. S., Lie, M. E. K., Bavo, Francesco, Loeffler, R., Damgaard, M., Ecker, G. F., Frølund, Bente & Wellendorph, Petrine, 2020, In: Scientific Reports. 10, 1, 15 p., 12992.

      Research output: Contribution to journal › Journal article › Research › peer-review

    6. Published

      Unraveling the Molecular Determinants for GABA Transporter Subtype Selectivity

      Kickinger, S., Al-Khawaja, A., Haugaard, A. S., Lie, M. E. K., Bavo, Francesco, Loffler, R., Damgaard, M., Frølund, Bente, Ecker, G. F. & Wellendorph, Petrine, 2020, p. 130A-130A.

      Research output: Contribution to conference › Conference abstract for conference › Research › peer-review

    7. Efficient One-Pot Reductive Aminations of Carbonyl Compounds with Aquivion-Fe as a Recyclable Catalyst and Sodium Borohydride

      Airoldi, V., Piccolo, O., Roda, G., Appiani, R., Bavo, Francesco, Tassini, R., Paganelli, S., Arnoldi, S., Pallavicini, M. & Bolchi, C., 16 Jan 2020, In: European Journal of Organic Chemistry. 2020, 2, p. 162-168 7 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    8. Behavioural and pharmacological profiles of zebrafish administrated pyrrolidinyl benzodioxanes and prolinol aryl ethers with high affinity for heteromeric nicotinic acetylcholine receptors

      Braida, D., Ponzoni, L., Moretti, M., Viani, P., Pallavicini, M., Bolchi, C., Appiani, R., Bavo, Francesco, Gotti, C. & Sala, M., 1 Aug 2020, In: Psychopharmacology. 237, 8, p. 2317-2326 10 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    9. 1,4-Benzodioxane, an evergreen, versatile scaffold in medicinal chemistry: A review of its recent applications in drug design

      Bolchi, C., Bavo, Francesco, Appiani, R., Roda, G. & Pallavicini, M., 15 Aug 2020, In: European Journal of Medicinal Chemistry. 200, 112419.

      Research output: Contribution to journal › Review › Research › peer-review

    10. Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype

      Bavo, Francesco, Pallavicini, M., Gotti, C., Appiani, R., Moretti, M., Colombo, S. F., Pucci, S., Viani, P., Budriesi, R., Renzi, M., Fucile, S. & Bolchi, C., 24 Dec 2020, In: Journal of Medicinal Chemistry. 63, 24, p. 15668-15692 25 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    11. 2021
    12. Published

      Determinants for α4β2 vs. α3β4 subtype selectivity of pyrrolidine-based nachrs ligands: A computational perspective with focus on recent cryo-em receptor structures

      Bavo, Francesco, Pallavicini, M., Appiani, R. & Bolchi, C., 2021, In: Molecules. 26, 12, 23 p., 3603.

      Research output: Contribution to journal › Journal article › Research › peer-review

    13. Published

      Structure-Activity Studies of 3,9-Diazaspiro[5.5]undecane-Based ?-Aminobutyric Acid Type A Receptor Antagonists with Immunomodulatory Effect

      Bavo, Francesco, De-Jong, H., Petersen, Jonas Odgaard, Falk-Petersen, C. B., Löffler, R., Sparrow, E., Rostrup, F., Eliasen, Jannik Nicklas, Wilhelmsen, K. S., Barslund, K., Bundgaard, C., Nielsen, Birgitte, Kristiansen, Uffe, Wellendorph, Petrine, Bogdanov, Y. & Frølund, Bente, 2021, In: Journal of Medicinal Chemistry. 64, 24, p. 17795-17812

      Research output: Contribution to journal › Journal article › Research › peer-review

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