Fredrik Björkling

Fredrik Björkling

Emeritus


  1. Published

    Target enzyme mutations are the molecular basis for resistance towards pharmacological inhibition of nicotinamide phosphoribosyltransferase

    Olesen, U. H., Petersen, J. G., Garten, A., Kiess, W., Yoshino, J., Imai, S., Christensen, M. K., Fristrup, P., Thougaard, A. V., Björkling, Fredrik, Jensen, P. B., Nielsen, S. J. & Sehested, M., 10 Dec 2010, In: BMC Cancer. 10, p. 677 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Selected strategies to fight pathogenic bacteria

    Plotniece, A., Sobolev, A., Supuran, C. T., Carta, F., Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, J., Augustyns, K., Cos, P., De Vooght, L., Govaerts, M., Aizawa, J., Tammela, P. & Žalubovskis, R., 2023, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 38, 1, 27 p., 2155816.

    Research output: Contribution to journalReviewResearchpeer-review

  3. Published

    Optimized Synthesis of Fmoc/Boc-Protected PNA Monomers and their Assembly into PNA Oligomers.

    Shaikh, Ashif Yasin, Björkling, Fredrik, Nielsen, Peter E. & Franzyk, Henrik, 2021, In: European Journal of Organic Chemistry. 2021, 19, p. 2792-2801 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues

    Shaikh, Ashif Yasin, Björkling, Fredrik, Zabicka, D., Tomczak, M., Urbas, M., Domraceva, I., Kreicberga, A. & Franzyk, Henrik, 2023, In: Bioorganic Chemistry. 141, 11 p., 106876.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139

    Shehata, M. A., Jensen, A. C. N., Lissa, D., Bisig, C., Isberg, V., Andersen, K. B., Harpsøe, Kasper, Björkling, Fredrik, Bräuner, Hans & Gloriam, David E., 10 Nov 2016, In: Scientific Reports. 6, p. 1-13 13 p., 36681.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Triphenylcarbenium Tetrafluoroborate as an Efficient Catalyst in the Regioselective Reductive Ring Opening of Benzylidene Acetals of Carbohydrates

    Thota, N., Björkling, Fredrik & Kankala, S., 2019, In: ChemistrySelect. 4, 27, p. 7976-7980

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Prediction of drug efficacy for cancer treatment based on comparative analysis of chemosensitivity and gene expression data

    Wan, P., Li, Q., Larsen, J. E. P., Eklund, A. C., Parlesak, A., Rigina, O., Nielsen, S. J., Björkling, Fredrik & Jonsdottir, S. O., 2012, In: Bioorganic & Medicinal Chemistry. 20, 1, p. 167-176 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Evaluation of 1H-Triazole-1-[N,N'-Bis(tert-butoxycarbonyl)]carboxamidine in Solution-Phase and On-Resin Guanidinylation

    Wester, A., Björkling, Fredrik & Franzyk, Henrik, 2021, In: The Journal of Organic Chemistry. 86, 21, p. 14371–14380

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Non-natural Amino Acid and Peptoid Building Blocks for Optimization of the Cell-Penetrating (R-X-R)n Motif

    Wester, A., Björkling, Fredrik, Nieslen, P. & Franzyk, Henrik, Sep 2018, In: Journal of Peptide Science. 24, p. S94-S94

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  10. Published

    Discovery of Novel Non-Steroidal Cytochrome P450 17A1 Inhibitors as Potential Prostate Cancer Agents

    Wróbel, T. M., Rogova, O., Andersen, Kasper Langebjerg, Yadav, R., Brixius-Anderko, S., Scott, E. E., Olsen, L., Jørgensen, Flemming Steen & Björkling, Fredrik, 2020, In: International Journal of Molecular Sciences . 21, 14, p. 1-11 4868.

    Research output: Contribution to journalJournal articleResearchpeer-review

ID: 8863737