Fredrik Björkling

Fredrik Björkling

Emeritus


  1. 2010
  2. Published

    Early detection of response to experimental chemotherapeutic Top216 with [18F]FLT and [18F]FDG PET in human ovary cancer xenografts in mice

    Wessel, Mette Munk, Erichsen, K. D., Björkling, Fredrik, Madsen, J., Jensen, P. B., Højgaard, Liselotte, Sehested, M. & Kjær, Andreas, 1 Jan 2010, In: P L o S One. 5, 9, p. e12965

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Synthesis and antitumor effect in vitro and in vivo of substituted 1,3-dihydroindole-2-ones

    Christensen, M. K., Erichsen, K. D., Trojel-Hansen, C., Tjørnelund, J., Nielsen, S. J., Frydenvang, Karla Andrea, Johansen, Tommy Nørskov, Nielsen, Birgitte, Sehested, M., Jensen, P. B., Ikaunieks, M., Zaichenko, A., Loza, E., Kalvinsh, I. & Björkling, Fredrik, 14 Oct 2010, In: Journal of Medicinal Chemistry. 53, 19, p. 7140-7145 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Target enzyme mutations are the molecular basis for resistance towards pharmacological inhibition of nicotinamide phosphoribosyltransferase

    Olesen, U. H., Petersen, J. G., Garten, A., Kiess, W., Yoshino, J., Imai, S., Christensen, M. K., Fristrup, P., Thougaard, A. V., Björkling, Fredrik, Jensen, P. B., Nielsen, S. J. & Sehested, M., 10 Dec 2010, In: BMC Cancer. 10, p. 677 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. 2012
  6. Published

    Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma brucei

    Kelly, J., Taylor, M. C., Horn, D., Loza, E., Kalvinsh, I. & Björkling, Fredrik, 2012, In: Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1886–1890 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Prediction of drug efficacy for cancer treatment based on comparative analysis of chemosensitivity and gene expression data

    Wan, P., Li, Q., Larsen, J. E. P., Eklund, A. C., Parlesak, A., Rigina, O., Nielsen, S. J., Björkling, Fredrik & Jonsdottir, S. O., 2012, In: Bioorganic & Medicinal Chemistry. 20, 1, p. 167-176 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published
  9. 2013
  10. Published

    Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET

    Wessel, Mette Munk, Erichsen, K. D., Björkling, Fredrik, Madsen, J., Jensen, Peter, Sehested, M., Højgaard, Liselotte & Kjær, Andreas, 2013, In: P L o S One. 8, 12, 9 p., e85126.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    [18F]FDG and [18F]FLT positron emission tomography imaging following treatment with belinostat in human ovary cancer xenografts in mice

    Wessel, Mette Munk, Erichsen, K. D., Johnbeck, C. B., Björkling, Fredrik, Madsen, J., Jensen, Peter, Sehested, M., Højgaard, Liselotte & Kjær, Andreas, 2013, In: B M C Cancer. 13, p. 1-9 10 p., 168.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    [18F]FLT and [18F]FDG PET for non-invasive treatment monitoring of the nicotinamide phosphoribosyltransferase inhibitor APO866 in human xenografts

    Erichsen, K. D., Johnbeck, C. B., Björkling, Fredrik, Madsen, J., Bzorek, M., Jensen, Peter, Højgaard, Liselotte, Sehested, M., Kjær, Andreas & Wessel, Mette Munk, 2013, In: P L o S One. 8, 1, p. 1-8 9 p., e53410.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. 2016
  14. Published

    Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139

    Shehata, M. A., Jensen, A. C. N., Lissa, D., Bisig, C., Isberg, V., Andersen, K. B., Harpsøe, Kasper, Björkling, Fredrik, Bräuner, Hans & Gloriam, David E., 10 Nov 2016, In: Scientific Reports. 6, p. 1-13 13 p., 36681.

    Research output: Contribution to journalJournal articleResearchpeer-review

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ID: 8863737