Fredrik Björkling

Fredrik Björkling

Emeritus


  1. Published

    Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues

    Shaikh, Ashif Yasin, Björkling, Fredrik, Zabicka, D., Tomczak, M., Urbas, M., Domraceva, I., Kreicberga, A. & Franzyk, Henrik, 2023, In: Bioorganic Chemistry. 141, 11 p., 106876.

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Selected strategies to fight pathogenic bacteria

    Plotniece, A., Sobolev, A., Supuran, C. T., Carta, F., Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, J., Augustyns, K., Cos, P., De Vooght, L., Govaerts, M., Aizawa, J., Tammela, P. & Žalubovskis, R., 2023, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 38, 1, 27 p., 2155816.

    Research output: Contribution to journalReviewResearchpeer-review

  3. Published

    Target enzyme mutations are the molecular basis for resistance towards pharmacological inhibition of nicotinamide phosphoribosyltransferase

    Olesen, U. H., Petersen, J. G., Garten, A., Kiess, W., Yoshino, J., Imai, S., Christensen, M. K., Fristrup, P., Thougaard, A. V., Björkling, Fredrik, Jensen, P. B., Nielsen, S. J. & Sehested, M., 10 Dec 2010, In: BMC Cancer. 10, p. 677 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Antisense PNA antibiotics against multiresistant Gram-negative bacteria

    Nielsen, Peter E., Björkling, Fredrik & Franzyk, Henrik, 2017, In: International Journal of Molecular Medicine. 40, Suppl. 1, p. S22 1 p., Abstract 169.

    Research output: Contribution to journalConference abstract in journalResearch

  5. Published

    Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET

    Wessel, Mette Munk, Erichsen, K. D., Björkling, Fredrik, Madsen, J., Jensen, Peter, Sehested, M., Højgaard, Liselotte & Kjær, Andreas, 2013, In: P L o S One. 8, 12, 9 p., e85126.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Synthesis of thiazole linked chalcones and their pyrimidine analogues as anticancer agents

    Kesari, C., Rama, K. R., Sedighi, K., Stenvang, Jan, Björkling, Fredrik, Kankala, S. & Thota, N., 2021, In: Synthetic Communications. 51, 9, p. 1406-1416 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma brucei

    Kelly, J., Taylor, M. C., Horn, D., Loza, E., Kalvinsh, I. & Björkling, Fredrik, 2012, In: Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1886–1890 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Synthesis of novel fluorophenylpyrazole-picolinamide derivatives and determination of their anticancer activity

    Kankala, S., Rama, K. R., Kesari, C., Björkling, Fredrik, Nerella, S., Gundepaka, P., Guguloth, H. & Thota, N., 2020, In: Synthetic Communications. 50, 19, p. 2997-3006 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Silver carbene complexes: An emerging class of anticancer agents

    Kankala, S., Thota, N., Björkling, Fredrik, Taylor, M. K., Vadde, R. & Balusu, R., Mar 2019, In: Drug Development Research. 80, 2, p. 188-199

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Polymyxins with Potent Antibacterial Activity against Colistin-Resistant Pathogens: Fine-Tuning Hydrophobicity with Unnatural Amino Acids

    Jørgensen, Johan Storm, Harifi Mood, Elnaz, Knap, A. S. H., Nielsen, S. E., Nielsen, Peter E., Żabicka, D., Matias, C., Domraceva, I., Björkling, Fredrik & Franzyk, Henrik, 2024, In: Journal of Medicinal Chemistry. 67, 2, p. 1370–1383

    Research output: Contribution to journalJournal articleResearchpeer-review

ID: 8863737