Fredrik Björkling

Fredrik Björkling

Emeritus


  1. Published

    Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment

    Wróbel, T. M., Jørgensen, Flemming Steen, Pandey, A. V., Grudzińska, A., Sharma, K., Yakubu, J. & Björkling, Fredrik, 2023, In: Journal of Medicinal Chemistry. 66, 10, p. 6542–6566

    Research output: Contribution to journalReviewResearchpeer-review

  2. Published

    Non-natural Amino Acid and Peptoid Building Blocks for Optimization of the Cell-Penetrating (R-X-R)n Motif

    Wester, A., Björkling, Fredrik, Nieslen, P. & Franzyk, Henrik, Sep 2018, In: Journal of Peptide Science. 24, p. S94-S94

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  3. Published

    Microwave-assisted solid-phase synthesis of antisense acpP peptide nucleic acid-peptide conjugates active against colistin- and tigecycline-resistant E. coli and K. pneumoniae

    Hansen, A. M., Bonke, G., Hogendorf, W. F. J., Björkling, Fredrik, Nielsen, J., Kongstad, Kenneth Thermann, Zabicka, D., Tomczak, M., Urbas, M., Nielsen, Peter E. & Franzyk, Henrik, 2019, In: European Journal of Medicinal Chemistry. 168, p. 134-145 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Jagten på kongens efterfølger

    Franzyk, Henrik, Björkling, Fredrik, Nielsen, J. & Nielsen, Peter E., 2015, In: Lægemiddelforskning. 2015, p. 24-27 4 p.

    Research output: Contribution to journalJournal articleCommunication

  5. Published

    Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma brucei

    Kelly, J., Taylor, M. C., Horn, D., Loza, E., Kalvinsh, I. & Björkling, Fredrik, 2012, In: Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1886–1890 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors

    Brem, J., Panduwawala, T., Hansen, J. U., Hewitt, J., Liepins, E., Donets, P., Espina, L., Farley, A. J. M., Shubin, K., Campillos, G. G., Kiuru, P., Shishodia, S., Krahn, D., Leśniak, R. K., Schmidt (Adrian), J., Calvopiña, K., Turrientes, M. C., Kavanagh, M. E., Lubriks, D., Hinchliffe, P. & 41 others, Langley, G. W., Aboklaish, A. F., Eneroth, A., Backlund, M., Baran, A. G., Nielsen, E. I., Speake, M., Kuka, J., Robinson, J., Grinberga, S., Robinson, L., McDonough, M. A., Rydzik, A. M., Leissing, T. M., Jimenez-Castellanos, J. C., Avison, M. B., Da Silva Pinto, S., Pannifer, A. D., Martjuga, M., Widlake, E., Priede, M., Hopkins Navratilova, I., Gniadkowski, M., Belfrage, A. K., Brandt, P., Yli-Kauhaluoma, J., Bacque, E., Page, M. G. P., Björkling, Fredrik, Tyrrell, J. M., Spencer, J., Lang, P. A., Baranczewski, P., Cantón, R., McElroy, S. P., Jones, P. S., Baquero, F., Suna, E., Morrison, A., Walsh, T. R. & Schofield, C. J., 2022, In: Nature Chemistry. 14, p. 15–24

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET

    Wessel, Mette Munk, Erichsen, K. D., Björkling, Fredrik, Madsen, J., Jensen, Peter, Sehested, M., Højgaard, Liselotte & Kjær, Andreas, 2013, In: P L o S One. 8, 12, 9 p., e85126.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Exploring the Potential of Sulfur Moieties in Compounds Inhibiting Steroidogenesis

    Wróbel, T. M., Sharma, K., Mannella, I., Oliaro-Bosso, S., Nieckarz, P., Du Toit, T., Voegel, C. D., Rojas Velazquez, M. N., Yakubu, J., Matveeva, A., Therkelsen, S., Jørgensen, Flemming Steen, Pandey, A. V., Pippione, A. C., Lolli, M. L., Boschi, D. & Björkling, Fredrik, 2023, In: Biomolecules. 13, 9, 18 p., 1349.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Evaluation of 1H-Triazole-1-[N,N'-Bis(tert-butoxycarbonyl)]carboxamidine in Solution-Phase and On-Resin Guanidinylation

    Wester, A., Björkling, Fredrik & Franzyk, Henrik, 2021, In: The Journal of Organic Chemistry. 86, 21, p. 14371–14380

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Early detection of response to experimental chemotherapeutic Top216 with [18F]FLT and [18F]FDG PET in human ovary cancer xenografts in mice

    Wessel, Mette Munk, Erichsen, K. D., Björkling, Fredrik, Madsen, J., Jensen, P. B., Højgaard, Liselotte, Sehested, M. & Kjær, Andreas, 1 Jan 2010, In: P L o S One. 5, 9, p. e12965

    Research output: Contribution to journalJournal articleResearchpeer-review

ID: 8863737