Fredrik Björkling
Emeritus
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- Published
Anticancer agents
Björkling, Fredrik & Jensen, L. H., 2010, Textbook of drug design and discovery. Krogsgaard-Larsen, P., Strømgaard, K. & Madsen, U. (eds.). 4 ed. Boca Raton: CRC Press, p. 375-392Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Education
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Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors
Brem, J., Panduwawala, T., Hansen, J. U., Hewitt, J., Liepins, E., Donets, P., Espina, L., Farley, A. J. M., Shubin, K., Campillos, G. G., Kiuru, P., Shishodia, S., Krahn, D., Leśniak, R. K., Schmidt (Adrian), J., Calvopiña, K., Turrientes, M. C., Kavanagh, M. E., Lubriks, D., Hinchliffe, P. & 41 others, , 2022, In: Nature Chemistry. 14, p. 15–24Research output: Contribution to journal › Journal article › Research › peer-review
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Synthesis and antitumor effect in vitro and in vivo of substituted 1,3-dihydroindole-2-ones
Christensen, M. K., Erichsen, K. D., Trojel-Hansen, C., Tjørnelund, J., Nielsen, S. J., Frydenvang, Karla Andrea, Johansen, Tommy Nørskov, Nielsen, Birgitte, Sehested, M., Jensen, P. B., Ikaunieks, M., Zaichenko, A., Loza, E., Kalvinsh, I. & Björkling, Fredrik, 14 Oct 2010, In: Journal of Medicinal Chemistry. 53, 19, p. 7140-7145 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Studies of antibacterial activity (in vitro and in vivo) and mode of action for des-acyl tridecaptins (DATs)
Couturier, C., Ronzon, Q., Lattanzi, G., Lingard, I., Coyne, S., Cazals, V., Dubarry, N., Yvon, S., Leroi-Geissler, C., Gracia, O. R., Teague, J., Sordello, S., Corbett, D., Bauch, C., Monlong, C., Payne, L., Taillier, T., Fuchs, H., Broenstrup, M., Harrison, P. H. & 10 others, , 2024, In: European Journal of Medicinal Chemistry. 265, 20 p., 116097.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents
Craig, A. J., Ermolovich, Y., Cameron, A., Rodler, A., Wang, H., Hawkes, J. A., Hubert, M., Björkling, Fredrik, Molchanova, N., Brimble, M. A., Moodie, L. W. K. & Svenson, J., 2023, In: ACS Medicinal Chemistry Letters. 14, 6, p. 802–809 8 p.Research output: Contribution to journal › Letter › Research › peer-review
- Published
[18F]FLT and [18F]FDG PET for non-invasive treatment monitoring of the nicotinamide phosphoribosyltransferase inhibitor APO866 in human xenografts
Erichsen, K. D., Johnbeck, C. B., Björkling, Fredrik, Madsen, J., Bzorek, M., Jensen, Peter, Højgaard, Liselotte, Sehested, M., Kjær, Andreas & Wessel, Mette Munk, 2013, In: P L o S One. 8, 1, p. 1-8 9 p., e53410.Research output: Contribution to journal › Journal article › Research › peer-review
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Structural Basis of Metallo-β-lactamase Inhibition by N-Sulfamoylpyrrole-2-carboxylates
Farley, A. J. M., Ermolovich, Y., Calvopiña, K., Rabe, P., Panduwawala, T., Brem, J., Björkling, Fredrik & Schofield, C. J., 2021, In: ACS Infectious Diseases. 7, 6, p. 1809–1817Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Jagten på kongens efterfølger
Franzyk, Henrik, Björkling, Fredrik, Nielsen, J. & Nielsen, Peter E., 2015, In: Lægemiddelforskning. 2015, p. 24-27 4 p.Research output: Contribution to journal › Journal article › Communication
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Peptide/β-Peptoid Hybrids with Ultrashort PEG-Like Moieties: Effects on Hydrophobicity, Antibacterial Activity and Hemolytic Properties
Frederiksen, N., Louka, S., Mudaliar, C., Domraceva, I., Kreicberga, A., Pugovics, O., Żabicka, D., Tomczak, M., Wygoda, W., Björkling, Fredrik & Franzyk, Henrik, 2021, In: International Journal of Molecular Sciences. 22, 13, 17 p., 7041.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Peptide/Peptoid Hybrid Oligomers: The Influence of Hydrophobicity and Relative Side-Chain Length on Antibacterial Activity and Cell Selectivity
Frederiksen, N., Hansen, Paul Robert, Björkling, Fredrik & Franzyk, Henrik, 4 Dec 2019, In: Molecules (Print Archive Edition). 24, 18 p., 4429.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 8863737
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Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET
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Non-natural Amino Acid and Peptoid Building Blocks for Optimization of the Cell-Penetrating (R-X-R)n Motif
Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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279
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Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139
Research output: Contribution to journal › Journal article › Research › peer-review
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