Fredrik Björkling
Emeritus
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- Published
Prediction of drug efficacy for cancer treatment based on comparative analysis of chemosensitivity and gene expression data
Wan, P., Li, Q., Larsen, J. E. P., Eklund, A. C., Parlesak, A., Rigina, O., Nielsen, S. J., Björkling, Fredrik & Jonsdottir, S. O., 2012, In: Bioorganic & Medicinal Chemistry. 20, 1, p. 167-176 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Selected strategies to fight pathogenic bacteria
Plotniece, A., Sobolev, A., Supuran, C. T., Carta, F., Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, J., Augustyns, K., Cos, P., De Vooght, L., Govaerts, M., Aizawa, J., Tammela, P. & Žalubovskis, R., 2023, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 38, 1, 27 p., 2155816.Research output: Contribution to journal › Review › Research › peer-review
- Published
Silver carbene complexes: An emerging class of anticancer agents
Kankala, S., Thota, N., Björkling, Fredrik, Taylor, M. K., Vadde, R. & Balusu, R., Mar 2019, In: Drug Development Research. 80, 2, p. 188-199Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structural Basis of Metallo-β-lactamase Inhibition by N-Sulfamoylpyrrole-2-carboxylates
Farley, A. J. M., Ermolovich, Y., Calvopiña, K., Rabe, P., Panduwawala, T., Brem, J., Björkling, Fredrik & Schofield, C. J., 2021, In: ACS Infectious Diseases. 7, 6, p. 1809–1817Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues
Shaikh, Ashif Yasin, Björkling, Fredrik, Zabicka, D., Tomczak, M., Urbas, M., Domraceva, I., Kreicberga, A. & Franzyk, Henrik, 2023, In: Bioorganic Chemistry. 141, 11 p., 106876.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Studies of antibacterial activity (in vitro and in vivo) and mode of action for des-acyl tridecaptins (DATs)
Couturier, C., Ronzon, Q., Lattanzi, G., Lingard, I., Coyne, S., Cazals, V., Dubarry, N., Yvon, S., Leroi-Geissler, C., Gracia, O. R., Teague, J., Sordello, S., Corbett, D., Bauch, C., Monlong, C., Payne, L., Taillier, T., Fuchs, H., Broenstrup, M., Harrison, P. H. & 10 others, , 2024, In: European Journal of Medicinal Chemistry. 265, 20 p., 116097.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and Structure–Activity Relationships of Novel Non-Steroidal CYP17A1 Inhibitors as Potential Prostate Cancer Agents
Wróbel, T. M., Rogova, O., Sharma, K., Velazquez, M. N. R., Pandey, A. V., Jørgensen, Flemming Steen, Arendrup, Frederic Schrøder, Andersen, Kasper Langebjerg & Björkling, Fredrik, 2022, In: Biomolecules. 12, 2, 165.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and antitumor effect in vitro and in vivo of substituted 1,3-dihydroindole-2-ones
Christensen, M. K., Erichsen, K. D., Trojel-Hansen, C., Tjørnelund, J., Nielsen, S. J., Frydenvang, Karla Andrea, Johansen, Tommy Nørskov, Nielsen, Birgitte, Sehested, M., Jensen, P. B., Ikaunieks, M., Zaichenko, A., Loza, E., Kalvinsh, I. & Björkling, Fredrik, 14 Oct 2010, In: Journal of Medicinal Chemistry. 53, 19, p. 7140-7145 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of novel fluorophenylpyrazole-picolinamide derivatives and determination of their anticancer activity
Kankala, S., Rama, K. R., Kesari, C., Björkling, Fredrik, Nerella, S., Gundepaka, P., Guguloth, H. & Thota, N., 2020, In: Synthetic Communications. 50, 19, p. 2997-3006 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of thiazole linked chalcones and their pyrimidine analogues as anticancer agents
Kesari, C., Rama, K. R., Sedighi, K., Stenvang, Jan, Björkling, Fredrik, Kankala, S. & Thota, N., 2021, In: Synthetic Communications. 51, 9, p. 1406-1416 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 8863737
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Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET
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1278
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Non-natural Amino Acid and Peptoid Building Blocks for Optimization of the Cell-Penetrating (R-X-R)n Motif
Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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279
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Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139
Research output: Contribution to journal › Journal article › Research › peer-review
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