Icaro Ariel Simon

Icaro Ariel Simon

Postdoc

ORCID: 0000-0003-4550-4248

Publication year:
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1 - 9 out of 9Page size: 10
  1. 2024

  2. Pharmacological Characterization and Radiolabeling of VUF15485, a High-Affinity Small-Molecule Agonist for the Atypical Chemokine Receptor ACKR3

    Zarca, A. M., Adlere, I., Viciano, C. P., Arimont-Segura, M., Meyrath, M., Simon, I. A., Bebelman, J. P., Laan, D., Custers, H. G. J., Janssen, E., Versteegh, K. L., Buzink, M. C. M. L., Nesheva, D. N., Bosma, R., de Esch, I. J. P., Vischer, H. F., Wijtmans, M., Szpakowska, M., Chevigné, A., Hoffmann, C. & 5 others, de Graaf, C., Zarzycka, B. A., Windhorst, A. D., Smit, M. J. & Leurs, R., 2024, In: Molecular Pharmacology. 105, 4, p. 301-312 12 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  3. 2023
  4. Published

    Ligand selectivity hotspots in serotonin GPCRs

    Simon, Icaro A, Bjørn-Yoshimoto, Walden, Harpsøe, Kasper, Iliadis, S., Svensson, B., Jensen, Anders A. & Gloriam, David E., 2023, In: Trends in Pharmacological Sciences. 44, 12, p. 978-990

    Research output: Contribution to journal › Review › Research › peer-review

  5. PSW-Designer: An Open-Source Computational Platform for the Design and Virtual Screening of Photopharmacological Ligands

    Simon, Icaro A, Homan, E. J., Wijtmans, M., Sundström, M., Leurs, R., De Esch, I. J. P. & Zarzycka, B. A., 2023, In: Journal of Chemical Information and Modeling. 63, 21, p. 6696-6705 10 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  6. Published

    Structure–Activity Assessment and In-Depth Analysis of Biased Agonism in a Set of Phenylalkylamine 5-HT2A Receptor Agonists

    Pottie, E., Poulie, Christian Bernard Matthijs, Simon, Icaro A, Harpsøe, Kasper, D’Andrea, L., Komarov, I. V., Gloriam, David E., Jensen, Anders A., Kristensen, Jesper Langgaard & Stove, C. P., 2023, In: ACS Chemical Neuroscience. 14, 15, p. 2727–2742

    Research output: Contribution to journal › Journal article › Research › peer-review

  7. 2022
  8. Published

    Discovery of β-Arrestin-Biased 25CN-NBOH-Derived 5-HT2A Receptor Agonists

    Poulie, Christian Bernard Matthijs, Pottie, E., Simon, Icaro A, Harpsøe, Kasper, D'Andrea, L., Komarov, I. V., Gloriam, David E., Jensen, Anders A., Stove, C. P. & Kristensen, Jesper Langgaard, 2022, In: Journal of Medicinal Chemistry. 65, 18, p. 12031–12043

    Research output: Contribution to journal › Journal article › Research › peer-review

  9. Published

    GPCRs steer Gi and Gs selectivity via TM5-TM6 switches as revealed by structures of serotonin receptors

    Huang, S., Xu, P., Shen, D., Simon, Icaro A, Mao, C., Tan, Y., Zhang, H., Harpsøe, Kasper, Li, H., Zhang, Y., You, C., Yu, X., Jiang, Y., Zhang, Y., Gloriam, David E. & Xu, H. E., 2022, In: Molecular Cell. 82, 14, p. 2681-2695.e6 15 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  10. 2021
  11. Published

    Structural insights into the lipid and ligand regulation of serotonin receptors

    Xu, P., Huang, S., Zhang, H., Mao, C., Zhou, X. E., Cheng, X., Simon, Icaro A, Shen, D., Yen, H., Robinson, C. V., Harpsøe, Kasper, Svensson, B., Guo, J., Jiang, H., Gloriam, David E., Melcher, K., Jiang, Y., Zhang, Y. & Xu, H. E., 2021, In: Nature. 592, p. 469-473

    Research output: Contribution to journal › Journal article › Research › peer-review

  12. 2015

  13. CuO Nanofibers Immobilized on Paraffin-Impregnated Graphite Electrode and its Application in the Amperometric Detection of Glucose

    Simon, Icaro A, Medeiros, N. G., Garcia, K. C., Soares, R. M. D., Rosa, A. T. & Silva, J. A., Aug 2015, In: Journal of the Brazilian Chemical Society. 26, 8, p. 1710-1717

    Research output: Contribution to journal › Journal article › Research › peer-review

  14. 2013

  15. Electrochemical Behavior of Gold Nanoparticles Generated In Situ on 3-(1-Imidazolyl)propyl-silsesquioxane

    Simon, Icaro A, Vacaro, B. B., Nunes, M. R., Benvenutti, E. V., Dias, S. L. P., Gushikem, Y. & Arguello, J., Nov 2013, In: Electroanalysis. 25, 11, p. 2501-2506

    Research output: Contribution to journal › Journal article › Research › peer-review

ID: 345280972