Matthias Manfred Herth
Professor
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- 2024
- Published
A facile synthesis of precursor for the σ-1 receptor PET radioligand [18F]FTC-146 and its radiofluorination
Marešová, A., Jurášek, M., Drašar, P. B., Dolenský, B., Prokudina, E. A., Shalgunov, Vladimir, Herth, Matthias Manfred, Cumming, P. & Popkov, A., 2024, In: Journal of Labelled Compounds and Radiopharmaceuticals. 67, 2, p. 59-66Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development and Preclinical Evaluation of [211At]PSAt-3-Ga: An Inhibitor for Targeted α-Therapy of Prostate Cancer.
El Fakiri, M., Ayada, N., Müller, Marius, Hvass, Lars, Gamzov, T. H., Clausen, Anne Skovsbo, Geis, N. M., Steinacker, N., Hansson, E., Lindegren, S., Aneheim, E., Jensen, H., Eder, A., Jensen, Andreas, Poulie, Christian Bernard Matthijs, Kjær, Andreas, Eder, M. & Herth, Matthias Manfred, 2024, In: Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 65, 4, p. 593-599Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Evaluation of F-537-Tetrazine in a model for brain pretargeting imaging. Comparison to N-(3-[18F] fluoro-5-(1,2,4,5-tetrazin-3-yl)benzyl)propan-1-amine
Shalgunov, Vladimir, van den Broek, S. L., Andersen, Ida Vang, Raval, N. R., Schäfer, G., Barz, M., Herth, Matthias Manfred & Battisti, Umberto Maria, 2024, In: Nuclear Medicine and Biology. 128-129, 12 p., 108877.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Investigation of imaging the somatostatin receptor by opening the blood-brain barrier with melittin – A feasibility study using positron emission tomography and [64Cu]Cu-DOTATATE
Andersen, Ida Vang, Bidesi, N. S. R., Shalgunov, Vladimir, Jørgensen, Jesper Tranekjær, Gustavsson, Karl Tobias, Strømgaard, Kristian, Ingemann Jensen, A. T., Kjær, Andreas & Herth, Matthias Manfred, 2024, In: Nuclear Medicine and Biology. 132-133, 5 p., 108905.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
Schlein, E., Rokka, J., Odell, L. R., van den Broek, S. L., Herth, Matthias Manfred, Battisti, Umberto Maria, Syvänen, S., Sehlin, D. & Eriksson, J., 2024, In: EJNMMI Radiopharmacy and Chemistry. 9, 1, 12 p., 21.Research output: Contribution to journal › Journal article › Research › peer-review
- 2023
- Published
A Fluorescent Probe as a Lead Compound for a Selective α-Synuclein PET Tracer: Development of a Library of 2-Styrylbenzothiazoles and Biological Evaluation of [18F]PFSB and [18F]MFSB
Di Nanni, A., Saw, R. S., Battisti, Umberto Maria, Bowden, G. D., Boeckermann, A., Bjerregaard-Andersen, K., Pichler, B. J., Herfert, K., Herth, Matthias Manfred & Maurer, A., 2023, In: ACS Omega. 8, 34, p. 31450–31467Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A SPECT-based method for dynamic imaging of the glymphatic system in rats
Sigurdsson, B., Hauglund, Natalie Linea, Lilius, T. O., Mogensen, F. L. H., Mortensen, K. N., Beschorner, Natalie, Klinger, L., Bærentzen, S. L., Rosenholm, Marko, Shalgunov, Vladimir, Herth, Matthias Manfred, Mori, Yuki & Nedergaard, Maiken, 2023, In: Journal of Cerebral Blood Flow and Metabolism. 43, 7, 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A nanobody recognizes a unique conserved epitope and potently neutralizes SARS-CoV-2 omicron variants
Modhiran, N., Lauer, S. M., Amarilla, A. A., Hewins, P., Lopes van den Broek, S. I., Low, Y. S., Thakur, N., Liang, B., Nieto, G. V., Jung, J., Paramitha, D., Isaacs, A., Sng, J. D. J., Song, D., Jørgensen, J. T., Cheuquemilla, Y., Bürger, J., Andersen, I. V., Himelreichs, J., Jara, R. & 18 others, , 2023, In: iScience. 26, 7, 26 p., 107085.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A pilot study of cerebral metabolism and serotonin 5-HT2A receptor occupancy in rats treated with the psychedelic tryptamine DMT in conjunction with the MAO inhibitor harmine
Egger, K., Gudmundsen, F., Jessen, N. S., Baun, C., Poetzsch, S. N., Shalgunov, Vladimir, Herth, Matthias Manfred, Quednow, B. B., Martin-Soelch, C., Dornbierer, D., Scheidegger, M., Cumming, P. & Palner, M., 2023, In: Frontiers in Pharmacology. 14, 12 p., 1140656.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Clearing and Masking Agents in Pretargeting Strategies
Staudt, Markus & Herth, Matthias Manfred, 2023, In: Pharmaceuticals. 16, 4, 15 p., 497.Research output: Contribution to journal › Review › Research › peer-review
- Published
Development of 11C-labeled CRANAD-102 for positron emission tomography imaging of soluble Aβ-species
Staudt, Markus, Shalgunov, Vladimir, Nedergaard, Maiken & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 12, p. 393-399Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Editorial: Prof. Frank Rösch's legacy in the radiopharmaceutical chemistry field
Poulie, Christian Bernard Matthijs, Piel, M., Neumaier, B., Ross, T. & Herth, Matthias Manfred, 2023, In: Frontiers in Nuclear Medicine. 3, 1336481.Research output: Contribution to journal › Editorial › Research › peer-review
- Published
In Vitro and In Vivo Evaluation of Pellotine: A Hypnotic Lophophora Alkaloid
Poulie, C. B. M., Chan, C. B., Parka, A., Lettorp, M., Vos, J., Raaschou, A., Pottie, E., Bundgaard, M. S., Sørensen, L. M. E., Cecchi, C. R., Märcher-Rørsted, E., Bach, A., Herth, M. M., Decker, A., Jensen, A. A., Elfving, B., Kretschmann, A. C., Stove, C. P., Kohlmeier, K. A., Cornett, C. & 3 others, , 2023, In: ACS Pharmacology & Translational Science. 6, 10, p. 1492-1507Research output: Contribution to journal › Journal article › Research › peer-review
- Accepted/In press
Labeling of highly reactive tetrazines using [ 18F]SuFEx
Battisti, Umberto Maria, Müller, Marius, García-Vázquez, R. & Herth, Matthias Manfred, 2023, (Accepted/In press) In: Synlett.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Next generation fibroblast activation protein (FAP) targeting PET tracers : The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines
Poulie, Christian Bernard Matthijs, Shalgunov, Vladimir, Elvas, F., Van Rymenant, Y., Moon, E. S., Battisti, Umberto Maria, De Loose, J., De Meester, I., Rösch, F., Van Der Veken, P. & Herth, Matthias Manfred, 2023, In: European Journal of Medicinal Chemistry. 262, 10 p., 115862.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Quantitative Evaluation of a Multimodal Aptamer-Targeted Long-Circulating Polymer for Tumor Targeting
Bohrmann, L., Burghardt, T., Rodríguez-Rodríguez, C., Herth, Matthias Manfred, Saatchi, K. & Häfeli, U. O., 2023, In: ACS Omega. 8, 12, p. 11003-11020Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Repeated low doses of psilocybin increase resilience to stress, lower compulsive actions, and strengthen cortical connections to the paraventricular thalamic nucleus in rats
Kiilerich, K. F., Lorenz, J., Scharff, M. B., Speth, N., Brandt, T. G., Czurylo, J., Xiong, M., Jessen, N. S., Casado-Sainz, A., Shalgunov, Vladimir, Kjærby, Celia, Satała, G., Bojarski, A. J., Jensen, Anders A., Herth, Matthias Manfred, Cumming, P., Overgaard, A. & Palner, M., 2023, In: Molecular Psychiatry. 28, 9, p. 3829-3841Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and in vivo evaluation of [11C]tucatinib for HER2-targeted PET imaging
Müller, Marius, Shalgunov, Vladimir, Hvass, Lars, Jørgensen, Jesper Tranekjær, Kramer, V., Staudt, Markus, Battisti, Umberto Maria, Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Bioorganic and Medicinal Chemistry Letters. 80, 5 p., 129088.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and radiolabeling of a polar [125 I]I-1,2,4,5-tetrazine
Bidesi, N., Shalgunov, Vladimir, Battisti, Umberto Maria, Hvass, Lars, Jørgensen, Jesper Tranekjær, Poulie, Christian Bernard Matthijs, Jensen, A. I., Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 1, p. 22-30Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The Alzheimer's disease 5xFAD mouse model is best suited to investigate pretargeted imaging approaches beyond the blood-brain barrier
Lopes van den Broek, S. I., Sehlin, D., Andersen, Jens Velde, Aldana, Blanca, Beschorner, Natalie, Nedergaard, Maiken, Knudsen, Gitte Moos, Syvanen, S. & Herth, Matthias Manfred, 2023, In: Frontiers in Nuclear Medicine. 2, 7 p., 1001722.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The Structural Combination of SIL and MODAG Scaffolds Fails to Enhance Binding to α-Synuclein but Reveals Promising Affinity to Amyloid β
Di Nanni, A., Saw, R. S., Bowden, G. D., Bidesi, N. S. R., Bjerregaard-Andersen, K., Korat, Š., Herth, Matthias Manfred, Pichler, B. J., Herfert, K. & Maurer, A., 2023, In: Molecules. 28, 10, 20 p., 4001.Research output: Contribution to journal › Journal article › Research › peer-review
- 2022
- Published
Bioorthogonal Click of Colloidal Gold Nanoparticles to Antibodies In vivo
Poulie, Christian Bernard Matthijs, Sporer, E., Hvass, Lars, Jørgensen, Jesper Tranekjær, Kempen, Paul Joseph, Lopes van den Broek, S. I., Shalgunov, Vladimir, Kjær, Andreas, Jensen, A. I. & Herth, Matthias Manfred, 2022, In: Chemistry - A European Journal. 28, 61, 10 p., e202201847.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Covalent core-radiolabeling of polymeric micelles with125I/211At for theranostic radiotherapy
Sporer, E., Poulie, Christian Bernard Matthijs, Bäck, T., Lindegren, S., Jensen, H., Kempen, Paul Joseph, Kjær, Andreas, Herth, Matthias Manfred & Jensen, A. I., 2022, In: Nanotheranostics. 6, 4, p. 388-399Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development and evaluation of an 18F-labeled nanobody to target SARS-CoV-2's spike protein
Lopes van den Broek, S., García-Vázquez, R., Andersen, Ida Vang, Valenzuela-Nieto, G., Shalgunov, Vladimir, Battisti, Umberto Maria, Schwefel, D., Modhiran, N., Kramer, V., Cheuquemilla, Y., Jara, R., Salinas-Varas, C., Amarilla, A. A., Watterson, D., Rojas-Fernandez, A. & Herth, Matthias Manfred, 2022, In: Frontiers in Nuclear Medicine. 2, 1033697.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of the First Tritiated Tetrazine: Facilitating Tritiation of Proteins
Radjani Bidesi, N. S., Battisti, Umberto Maria, Lopes van de Broek, S., Shalgunov, Vladimir, Dall, A., Bøggild Kristensen, J., Sehlin, D., Syvänen, S., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2022, In: ChemBioChem. 23, 23, 7 p., e202200539.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 33147568
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573
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SPECT imaging of the glymphatic pathway with In-111-labeled ovalbumin in the rat brain
Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
Published -
543
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Convenient access to F-18-labeled amines through the Staudinger reduction
Research output: Contribution to journal › Conference abstract in journal › Research
Published -
361
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Pretargeting in nuclear imaging and radionuclide therapy: Improving efficacy of theranostics and nanomedicines
Research output: Contribution to journal › Journal article › Research › peer-review
Published