Povl Krogsgaard-Larsen
Professor, emeritus
Medicinal Chemistry
Jagtvej 162
2100 København Ø
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(S)-homo-AMPA, a specific agonist at the mGlu6 subtype of metabotropic glutamic acid receptors
Ahmadian, H., Nielsen, Birgitte, Bräuner, Hans, Johansen, Tommy Nørskov, Stensbøl, T. B., Sløk, F. A., Sekiyama, N., Nakanishi, S., Krogsgaard-Larsen, Povl & Madsen, Ulf, 24 Oct 1997, In: Journal of Medicinal Chemistry. 40, 22, p. 3700-5Research output: Contribution to journal › Journal article › Research › peer-review
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Action of bicyclic isoxazole GABA analogues on GABA transporters and its relation to anticonvulsant activity
Bolvig, T., Larsson, O. M., Pickering, Darryl S, Nelson, N., Falch, E., Krogsgaard-Larsen, Povl, Schousboe, Arne & Pickering, Darryl S, 1999, In: European Journal of Pharmacology. 375, 1-3, p. 367-74 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Structure and pharmacology of 4,5,6,7-tetrahydroisothiazolo [5,4-c]pyridin-3-ol (Thio-THIP), an agonist/antagonist at GABA(A) receptors
Brehm, L., Ebert, B., Kristiansen, Uffe, Wafford, K. A., Kemp, J. A. & Krogsgaard-Larsen, Povl, 1997, In: European Journal of Medicinal Chemistry. 32, 4, p. 357-363 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
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(S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid, a potent and selective agonist at the GluR5 subtype of ionotropic glutamate receptors. Synthesis, modeling, and molecular pharmacology
Brehm, L., Greenwood, J. R., Hansen, K. B., Nielsen, Birgitte, Egebjerg, J., Stensbøl, T. B., Bräuner, Hans, Sløk, F. A., Kronborg, T. T. A. & Krogsgaard-Larsen, Povl, 10 Apr 2003, In: Journal of Medicinal Chemistry. 46, 8, p. 1350-8Research output: Contribution to journal › Journal article › Research › peer-review
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Crystal Structure and Quantum Chemical Ab Initio Calculations of Ibotenic Acid, an Excitatory Amino Acid Receptor Agonist
Brehm, L., Frydenvang, Karla Andrea, Krogsgaard-Larsen, Povl & Liljefors, T., 1998, In: Structural Chemistry. 9, 2, p. 149-155 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Structural and stereochemical requirements for interactions with subtypes of central excitatory amino acid receptors
Brehm, L., Christensen, I. T., Nielsen, Birgitte, Reinhardt, A., Ebert, B., Madsen, Ulf, Jørgensen, Flemming Steen, Hansen, J. J. & Krogsgaard-Larsen, Povl, 1990, Frontiers in Drug Research; Alfred Benzon Symposium 28. Jensen, B., Jørgensen, F. S. & Kofod, H. (eds.). Copenhagen: Munksgaard , p. 92-105 14 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
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Synthesis, theoretical and structural analyses, and enantiopharmacology of 3-carboxy homologs of AMPA
Brehm, L., Greenwood, J. R., Sløk, F. A., Holm, M. M., Nielsen, Birgitte, Geneser, U., Stensbøl, T. B., Bräuner, Hans, Begtrup, M., Egebjerg, J. & Krogsgaard-Larsen, Povl, Aug 2004, In: Chirality. 16, 7, p. 452-66Research output: Contribution to journal › Journal article › Research › peer-review
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Contrasting actions of philanthotoxin-343 and philanthotoxin-(12) on human muscle nicotinic acetylcholine receptors
Brier, T. J., Mellor, I. R., Tikhonov, D. B., Neagoe, I., Shao, Z., Brierley, M. J., Strømgaard, Kristian, Jaroszewski, J. W., Krogsgaard-Larsen, Povl & Usherwood, P. N. R., Oct 2003, In: Molecular Pharmacology. 64, 4, p. 954-964 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
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The agonist-binding domain of the calcium-sensing receptor is located at the amino-terminal domain
Bräuner, Hans, Jensen, Anders A., Sheppard, P. O., O'Hara, P. & Krogsgaard-Larsen, Povl, 1999, In: Journal of Biological Chemistry. 274, 26, p. 18382-6 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Cloning and characterization of a human orphan family C G-protein coupled receptor GPRC5D
Bräuner, Hans, Jensen, Anders A., Sheppard, P. O., Larsen, Birger Brodin, Krogsgaard-Larsen, Povl & O'Hara, P., 2001, In: BBA General Subjects. 1518, 3, p. 237-48 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Interaction of CPCCOEt with a chimeric mGlu1b and calcium sensing receptor
Bräuner, Hans, Jensen, Anders A. & Krogsgaard-Larsen, Povl, 1999, In: NeuroReport. 10, 18, p. 3923-5 3 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Ligands for glutamate receptors: design and therapeutic prospects
Bräuner, Hans, Egebjerg, J., Nielsen, E. O., Madsen, Ulf & Krogsgaard-Larsen, Povl, 13 Jul 2000, In: Journal of Medicinal Chemistry. 43, 14, p. 2609-45Research output: Contribution to journal › Journal article › Research › peer-review
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A new structural class of subtype-selective inhibitor of cloned excitatory amino acid transporter, EAAT2
Bräuner, Hans, Hermit, M. B., Nielsen, Birgitte, Krogsgaard-Larsen, Povl & Johansen, Tommy Nørskov, 6 Oct 2000, In: European Journal of Pharmacology. 406, 1, p. 41-4Research output: Contribution to journal › Journal article › Research › peer-review
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Functional partial agonism at cloned human muscarinic acetylcholine receptors
Bräuner, Hans, Ebert, B., Brann, M. R., Falch, E. & Krogsgaard-Larsen, Povl, 10 Oct 1996, In: European Journal of Pharmacology. 313, 1-2, p. 145-50Research output: Contribution to journal › Journal article › Research › peer-review
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Annulated heterocyclic bioisosteres of norarecoline. Synthesis and molecular pharmacology at five recombinant human muscarinic acetylcholine receptors
Bräuner, Hans, Ebert, B., Brann, M. R., Falch, E. & Krogsgaard-Larsen, Povl, 9 Jun 1995, In: Journal of Medicinal Chemistry. 38, 12, p. 2188-95Research output: Contribution to journal › Journal article › Research › peer-review
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A new highly selective metabotropic excitatory amino acid agonist: 2-amino-4-(3-hydroxy-5-methylisoxazol-4-yl)butyric acid
Bräuner, Hans, Sløk, F. A., Skjaerbaek, N., Ebert, B., Sekiyama, N., Nakanishi, S. & Krogsgaard-Larsen, Povl, 2 Aug 1996, In: Journal of Medicinal Chemistry. 39, 16, p. 3188-94Research output: Contribution to journal › Journal article › Research › peer-review
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Sequence and expression pattern of a novel human orphan G-protein-coupled receptor, GPRC5B, a family C receptor with a short amino-terminal domain
Bräuner, Hans & Krogsgaard-Larsen, Povl, 15 Apr 2000, In: Genomics. 65, 2, p. 121-8Research output: Contribution to journal › Journal article › Research › peer-review
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Functional pharmacology of cloned heterodimeric GABA-B receptors expressed in mammalian cells
Bräuner, Hans & Krogsgaard-Larsen, Povl, Dec 1999, In: British Journal of Pharmacology. 128, 7, p. 1370-4Research output: Contribution to journal › Journal article › Research › peer-review
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Molecular pharmacology of 4-substituted glutamic acid analogues at ionotropic and metabotropic excitatory amino acid receptors
Bräuner, Hans, Nielsen, Birgitte, Stensbøl, T. B., Johansen, Tommy Nørskov, Skjaerbaek, N. & Krogsgaard-Larsen, Povl, 24 Sep 1997, In: European Journal of Pharmacology. 335, 2-3, p. R1-3Research output: Contribution to journal › Journal article › Research › peer-review
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Molecular pharmacology of homologues of ibotenic acid at cloned metabotropic glutamic acid receptors
Bräuner, Hans, Nielsen, Birgitte & Krogsgaard-Larsen, Povl, 5 Jun 1998, In: European Journal of Pharmacology. 350, 2-3, p. 311-6Research output: Contribution to journal › Journal article › Research › peer-review
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Pharmacology of (S)-homoquisqualic acid and (S)-2-amino-5-phosphonopentanoic acid [(S)-AP5] at cloned metabotropic glutamate receptors
Bräuner, Hans & Krogsgaard-Larsen, Povl, Jan 1998, In: British Journal of Pharmacology. 123, 2, p. 269-74Research output: Contribution to journal › Journal article › Research › peer-review
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Unprecedented migration of N-alkoxycarbonyl groups in protected pyroglutaminol
Bunch, Lennart, Norrby, P., Frydenvang, Karla Andrea, Krogsgaard-Larsen, Povl & Madsen, Ulf, 2001, In: Organic Letters. 3, 3, p. 433-5 3 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Synthesis and receptor binding affinity of new selective GluR5 ligands
Bunch, Lennart, Johansen, T. H., Bräuner, Hans, Stensbøl, T. B., Johansen, Tommy Nørskov, Krogsgaard-Larsen, Povl & Madsen, Ulf, Apr 2001, In: Bioorganic & Medicinal Chemistry. 9, 4, p. 875-9Research output: Contribution to journal › Journal article › Research › peer-review
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Subtype selective kainic acid receptor agonists: discovery and approaches to rational design
Bunch, Lennart & Krogsgaard-Larsen, Povl, 2009, In: Medicinal Research Reviews. 29, 1, p. 3-28Research output: Contribution to journal › Review › Research › peer-review
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Rational design, synthesis, and pharmacological evaluation of 2-azanorbornane-3-exo,5-endo-dicarboxylic acid: a novel conformationally restricted glutamic acid analogue
Bunch, Lennart, Liljefors, T., Greenwood, J. R., Frydenvang, Karla Andrea, Bräuner, Hans, Krogsgaard-Larsen, Povl & Madsen, Ulf, 2003, In: Journal of Organic Chemistry. 68, 4, p. 1489-95 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1303013