Povl Krogsgaard-Larsen
Professor, emeritus
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- 1991
- Published
Conformational and pharmacological characterization of 4-AHCP, a bicyclic homologue of the excitatory amino acid receptor agonist AMPA
Lund, Trine Meldgaard, Madsen, Ulf, Ebert, B., Jørgensen, Flemming Steen & Krogsgaard-Larsen, Povl, 1991, In: Med. Chem. Res. 1, p. 136-141 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Excitatory amino acid receptors: multiplicity and structural requirements for activation and blockade
Krogsgaard-Larsen, Povl, Lund, Trine Meldgaard, Jørgensen, Flemming Steen & Brehn, L., 1991, Excitatory amino acids and synaptic function. Wheal, H. & Thomson, A. (eds.). London: Academic Press, p. 1-17 17 p. (Excitatory Amino Acids and Synaptic Transmission, Academic Press, London).Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- Published
Novel (Gamma-Aminobutyric Acid)A Agonists and Partial Agonists
Krogsgaard-Larsen, Povl, Frølund, Bente, Kristiansen, Uffe, Lambert, J. D. C., Falch, E. & Curtis, D. R., 1991, Transmitter Amino Acid Receptors. Barnard, E. A. & Costa, E. (eds.). Raven Press, p. 237–249Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- 1990
- Published
AMPA receptor agonists, design, synthesis and molecular pharmacology
Lund, Trine Meldgaard, Christensen, I. T., Madsen, Ulf, Ebert, B., Brehm, L. & Krogsgaard-Larsen, Povl, 1990, In: Neurochemistry International. 16 suppl 1, 51, p. 51 1 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- Published
Excitatory Amino acid receptor agonists: enantiomeric resolutions by use of enzymes and chiral HPLC
Hansen, J. J., Nielsen, Birgitte, Reinhardt, A. & Krogsgaard-Larsen, Povl, 1990, In: Acta Pharmaceutica Nordica. 2, p. 185-192 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Relationship between structure, conformational flexibility, and biological activity of agonists and antagonists at the N-methyl-D-aspartic acid subtype of excitatory amino acid receptors
Madsen, Ulf, Brehm, L., Schaumburg, K., Jørgensen, Flemming Steen & Krogsgaard-Larsen, Povl, 1990, In: Journal of Medicinal Chemistry. 33, 1, p. 374-80 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structural and stereochemical requirements for interactions with subtypes of central excitatory amino acid receptors
Brehm, L., Christensen, I. T., Nielsen, Birgitte, Reinhardt, A., Ebert, B., Madsen, Ulf, Jørgensen, Flemming Steen, Hansen, J. J. & Krogsgaard-Larsen, Povl, 1990, Frontiers in Drug Research; Alfred Benzon Symposium 28. Jensen, B., Jørgensen, F. S. & Kofod, H. (eds.). Copenhagen: Munksgaard , p. 92-105 14 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- Published
Structural, stereochemical and conformational requirements for activation and blockade of central glutamic acid receptors
Krogsgaard-Larsen, Povl, Madsen, Ulf, Brehm, L., Christensen, I. T., Nielsen, Birgitte, Reinhardt, A., Ebert, B. & Hansen, J. J., 1990, Problems and Wonders of Chirale Molecules. Simonyi, M. (ed.). Budapest: Akadémiai Kiadó, p. 205-225 21 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- 1989
- Published
Heterocyclic muscarinic agonists: Structural and therapeutic aspects
Krogsgaard-Larsen, Povl, Jensen, B., Falch, E. & Jørgensen, Flemming Steen, 1 Jan 1989, In: Drugs of the Future. 14, 6, p. 541-561 21 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Excitatory Amino acid agonists and parital agonists
Christensen, I. T., Reinhardt, A., Nielsen, Birgitte, Ebert, B., Madsen, Ulf, Nielsen, E. Ø., Brehm, L. & Krogsgaard-Larsen, Povl, 1989, In: drug design and delivery. 5, p. 57-71 15 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Excitatory Amino acid agonists: Enzymic resolution, X-ray structure, and enantioselective activities of (R)- and (S)-bromohomoibotenic acid
Hansen, J. J., Nielsen, Birgitte, Krogsgaard-Larsen, Povl, Brehm, L., Nielsen, E. Ø. & Curtis, D. R., 1989, In: Journal of Medicinal Chemistry. 32, p. 2254-2260 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Excitatory amino acid agonists and partial agonists
Christensen, I. T., Reinhardt, A., Nielsen, B., Ebert, B., Madsen, Ulf, Nielsen, E. O., Brehm, L. & Krogsgaard-Larsen, Povl, 1989, In: Drug Design and Delivery. 5, 1, p. 57-71 15 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Isoxazole amino acids as glutamic acid receptor agonists: conformational and stereochemical aspects
Hansen, J. J., Madsen, Ulf, Nielsen, E. Ø., Nielsen, Birgitte, Brehm, L. & Krogsgaard-Larsen, Povl, 1989, New Methods in Drug Research. Makriayannis, A. (ed.). Barcelona: Prous Scientific Publishers, Vol. 3. p. 73-101 29 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- Published
Medicinal chemical and pharmacological focus on GABA and glutamic acid receptors in neurodegenerative disorders
Krogsgaard-Larsen, Povl, Hedegaard, A., Nielsen, L., Nielsen, Birgitte, Madsen, Ulf, Brehm, L., Falch, E., Hjeds, H. & Hansen, J. J., 1989, Trends in Medicinal Chemistry '88. van der Goot, H., Domány, G., Pallos, L. & Timmerman, H. (eds.). Elsevier, Amsterdam, p. 429-452 24 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- 1987
- Published
Molecular pharmacology of excitatory amino acid receptors: conformational and stereochemical requirements
Krogsgaard-Larsen, Povl, Madsen, Ulf, Nielsen, Birgitte, Hansen, J. J., Nielsen, E. Ø., Brehm, L. & Curtis, D. R., 1987, Proceedings of the X'th International Congress of Pharmacology. Rand, M. J. & Raper, C. (eds.). Elsevier, p. 113-116 4 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- 1980
- Published
Preparations of deuterium labelled guvacine and isoguvacine
Christensen, Søren Brøgger & Krogsgaard-Larsen, Povl, 1 Jan 1980, In: Journal of Labelled Compounds and Radiopharmaceuticals. 17, 2, p. 191-202 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 1977
- Published
Muscimol analogues. I. Syntheses of 4- and 8-aminocycloheptenol[1,2 d]isoxazol-3-ols and 4-(3-aminopropyl)-5-methyl-3-isoxazolol
Krogsgaard-Larsen, Povl, Natova, L. & Christensen, Søren Brøgger, 1 Jan 1977, In: ACTA CHEM. SCAND.. B31, 7, p. 577-583 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 1973
- Published
Organic hydroxylamine derivatives. VII. Isoxazolin 5 ones. An investigation of a reaction sequence previously stated to give 3 hydroxyisoxazoles
Krogsgaard-Larsen, Povl, Christensen, Søren Brøgger & Hjeds, H., 1 Jan 1973, In: Acta Chemica Scandinavica. 27, 8, p. 2802-2812 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Organic hydroxylamine derivatives. VIII. Structural analogues of GABA of the isoxazole enol betaine type. Synthesis of 5,6,7,8 tetrahydro 4H isoxazolo[3,4 d]azepin 3 ol zwitterion and some derivatives
Krogsgaard-Larsen, Povl, Hjeds, H. & Christensen, Søren Brøgger, 1 Jan 1973, In: Acta Chemica Scandinavica. 27, 9, p. 3251-3258 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1303013