Rasmus Prætorius Clausen

Rasmus Prætorius Clausen

Professor


  1. Published

    Preparation of Spirocyclic β-Proline Esters: Geometrically Restricted Building Blocks for Medicinal Chemistry

    Fjelbye, K., Marigo, M., Clausen, Rasmus Prætorius & Juhl, K., 2017, In: SYNLETT: Accounts and Rapid Communications in Chemical Synthesis. 28, 2, p. 231-234 4 p., st-2016-b0534-l.

    Research output: Contribution to journalReviewResearchpeer-review

  2. Published

    Elucidation of fluorine's impact on pKa and in vitro Pgp-mediated efflux for a series of PDE9 inhibitors

    Fjelbye, K., Marigo, M., Clausen, Rasmus Prætorius, Jørgensen, E. B., Christoffersen, C. T. & Juhl, K., 2018, In: MedChemComm. 9, 5, p. 893-896 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Biostructural and pharmacological studies of bicyclic analogues of the 3-isoxazolol glutamate receptor agonist ibotenic acid

    Frydenvang, Karla Andrea, Pickering, Darryl S, Greenwood, J. R., Krogsgaard-Larsen, N., Brehm, L., Nielsen, Birgitte, Vogensen, S. B., Hald, H., Kastrup, Jette Sandholm Jensen, Krogsgaard-Larsen, Povl & Clausen, Rasmus Prætorius, 10 Nov 2010, In: Journal of Medicinal Chemistry. 53, 23, p. 8354-8361

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    A novel selective γ-aminobutyric acid transport inhibitor demonstrates a functional role for GABA transporter subtype GAT2/BGT-1 in the CNS

    Frølund, Bente, Clausen, Rasmus Prætorius, Larsson, O. M., Schousboe, Arne, Krogsgaard-Larsen, Povl & White, H. S., 2006, In: Neurochemistry International. 48, p. 637–642

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Novel Approach toward 3,3-Difluoropiperidines from Easily Available Starting Materials and Synthesis of a New Phosphodiesterase Inhibitor

    Giacoboni, J., Clausen, Rasmus Prætorius & Marigo, M., Dec 2016, In: SYNLETT: Accounts and Rapid Communications in Chemical Synthesis. 27, 20, p. 2803-2806 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Tweaking agonist efficacy at N-methyl-D-aspartate receptors by site-directed mutagenesis

    Hansen, K. B., Clausen, Rasmus Prætorius, Bjerrum, E. J., Bechmann, C., Greenwood, J. R., Christensen, C., Kristensen, Jesper Langgaard, Egebjerg, J. & Bräuner, Hans, Dec 2005, In: Molecular Pharmacology. 68, 6, p. 1510-23

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Subunit-Specific Activation of NMDA Receptors

    Hansen, K. B., Burger, P., Vance, K. M., Snyder, J. P., Clausen, Rasmus Prætorius & Traynelis, S. F., Jan 2010, In: Biophysical Journal. 98, 3, suppl. 1, p. 525A-526A

    Research output: Contribution to journalConference abstract in journalResearch

  8. Published

    Structural determinants of agonist efficacy at the glutamate binding site of N-methyl-D-aspartate receptors

    Hansen, K. B., Tajima, N., Risgaard, R., Perszyk, R. E., Jørgensen, L., Vance, K. M., Ogden, K. K., Clausen, Rasmus Prætorius, Furukawa, H. & Traynelis, S. F., Jul 2013, In: Molecular Pharmacology. 84, 1, p. 114-127

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    MEDI 480-Novel lipophilic gamma-hydroxybutyrate (GHB) analogs with high affinity to GHB sites in rat brain

    Hog, S., Wellendorph, Petrine, Nielsen, Birgitte, Frølund, Bente & Clausen, Rasmus Prætorius, 10 Sep 2006, In: American Chemical Society. Abstracts of Papers (at the National Meeting). 232

    Research output: Contribution to journalConference abstract in journalResearch

  10. Published

    Hvordan virker Fantasy i hjernen?

    Høg, S., Wellendorph, Petrine, Greenwood, J. & Clausen, Rasmus Prætorius, 2005, In: Lægemiddelforskning. 2005, p. 16-17

    Research output: Contribution to journalJournal articleCommunication

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